WO2007003295A3 - Verfahren zur herstellung von 3-arylmethylthio- und 3-heteroarylmethylthio-4,5- dihydro-isoxazolin-derivaten - Google Patents

Verfahren zur herstellung von 3-arylmethylthio- und 3-heteroarylmethylthio-4,5- dihydro-isoxazolin-derivaten Download PDF

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Publication number
WO2007003295A3
WO2007003295A3 PCT/EP2006/006123 EP2006006123W WO2007003295A3 WO 2007003295 A3 WO2007003295 A3 WO 2007003295A3 EP 2006006123 W EP2006006123 W EP 2006006123W WO 2007003295 A3 WO2007003295 A3 WO 2007003295A3
Authority
WO
WIPO (PCT)
Prior art keywords
heteroarylmethylthio
arylmethylthio
dihydro
producing
isoxazoline derivatives
Prior art date
Application number
PCT/EP2006/006123
Other languages
English (en)
French (fr)
Other versions
WO2007003295A2 (de
Inventor
Wolfgang Schaper
Hendrik Helmke
Original Assignee
Bayer Cropscience Ag
Wolfgang Schaper
Hendrik Helmke
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag, Wolfgang Schaper, Hendrik Helmke filed Critical Bayer Cropscience Ag
Priority to JP2008519823A priority Critical patent/JP2008544996A/ja
Priority to BRPI0612729-0A priority patent/BRPI0612729A2/pt
Priority to CA002614239A priority patent/CA2614239A1/en
Priority to EP06776077A priority patent/EP1902038A2/de
Publication of WO2007003295A2 publication Critical patent/WO2007003295A2/de
Publication of WO2007003295A3 publication Critical patent/WO2007003295A3/de
Priority to IL188431A priority patent/IL188431A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/08—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

Verfahren zur Herstellung von 3-Arylmethylthio- und 3-Heteroarylmethylthio-4,5- dihydro-isoxazolin-Derivaten Die Erfindung betrifft ein Verfahren zur Herstellung von von 3-Arylmethylthio- und 3- Heteroarylmethylthio-4,5-dihydro-isoxazolin-Derivaten der allgemeinen Formel (I) durch ein Eintopfverfahren, in dem korrespondierende Arylmethyl- und Heteroarylmethyl-isothiuroniumsalze in Gegenwart einer wässrigen Alkali- oder Erdalkalibase mit einem Isoxazolin-Derivat zu den entsprechenden 3-Arylmethylthio- und 3-Heteroarylmethylthio-4,5-dihydro-isoxazolin-Derivaten umgesetzt werden.
PCT/EP2006/006123 2005-07-06 2006-06-24 Verfahren zur herstellung von 3-arylmethylthio- und 3-heteroarylmethylthio-4,5- dihydro-isoxazolin-derivaten WO2007003295A2 (de)

Priority Applications (5)

Application Number Priority Date Filing Date Title
JP2008519823A JP2008544996A (ja) 2005-07-06 2006-06-24 ３−アリールメチルチオ−及び３−ヘテロアリールメチルチオ−４，５−ジヒドロイソオキサゾリン誘導体の製造方法
BRPI0612729-0A BRPI0612729A2 (pt) 2005-07-06 2006-06-24 Método para a produção de derivados de 3-arilmetiltio- e 3 - heteroarilmetiltio-4,5-dihdroisoxazolina
CA002614239A CA2614239A1 (en) 2005-07-06 2006-06-24 Method for producing 3-arylmethylthio- and 3-heteroarylmethylthio-4,5-dihydro-isoxazoline derivatives
EP06776077A EP1902038A2 (de) 2005-07-06 2006-06-24 Verfahren zur herstellung von 3-arylmethylthio- und 3-heteroarylmethylthio-4,5- dihydro-isoxazolin-derivaten
IL188431A IL188431A0 (en) 2005-07-06 2007-12-26 Process for preparing 3-arylmethylthio-and 3-heteroarylmethylthio-4,5-dihydro-

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102005031583A DE102005031583A1 (de) 2005-07-06 2005-07-06 Verfahren zur Herstellung von von 3-Arylmethylthio- und 3-Heteroarylmethylthio-4,5-dihydro-isoxazolin-Derivaten
DE102005031583.6 2005-07-06

Publications (2)

Publication Number Publication Date
WO2007003295A2 WO2007003295A2 (de) 2007-01-11
WO2007003295A3 true WO2007003295A3 (de) 2007-07-19

Family

ID=37530083

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2006/006123 WO2007003295A2 (de) 2005-07-06 2006-06-24 Verfahren zur herstellung von 3-arylmethylthio- und 3-heteroarylmethylthio-4,5- dihydro-isoxazolin-derivaten

Country Status (10)

Country Link
US (1) US20070015805A1 (de)
EP (1) EP1902038A2 (de)
JP (1) JP2008544996A (de)
KR (1) KR20080030605A (de)
CN (1) CN101213181A (de)
BR (1) BRPI0612729A2 (de)
CA (1) CA2614239A1 (de)
DE (1) DE102005031583A1 (de)
IL (1) IL188431A0 (de)
WO (1) WO2007003295A2 (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1799657B1 (de) * 2004-10-05 2009-12-02 Syngenta Limited Isoxazolinderivate und ihre verwendung als herbizide
GB0526044D0 (en) * 2005-12-21 2006-02-01 Syngenta Ltd Novel herbicides
DE102007012168A1 (de) 2007-03-12 2008-09-18 Bayer Cropscience Ag 2-[Heteroarylalkyl-sulfonyl]-thiazol-Derivate und 2-[Heteroarylalkyl-sulfinyl]-thiazol-Derivate, Verfahren zu deren Herstellung, sowie deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren
EP2065374A1 (de) 2007-11-30 2009-06-03 Bayer CropScience AG 2-(Benzyl- und 1H-pyrazol-4-ylmethyl)sulfinyl-Thiazol-Derivate als Herbizide und Pflanzenwachstumsregulatoren
EP2065373A1 (de) 2007-11-30 2009-06-03 Bayer CropScience AG Chirale 3-(Benzylsulfinyl)-5,5-dimethyl-4,5-dihydroisoxazol-Derivate und 5,5-Dimethyl-3-[(1H-pyrazol-4-ylmethyl) sulfinyl]-4,5-dihydroisoxazol-Derivate, Verfahren zu deren Herstellung sowie deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren
EP2112143A1 (de) 2008-04-22 2009-10-28 Bayer CropScience AG 2-(Benzylsulfonyl)-Oxazol-Derivate, chirale 2-(Benzylsulfinyl)-Oxazol-Derivate 2-(Benzylsulfanyl-Oxazol Derivate, Verfahren zu deren Herstellung sowie deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren
EP2112149A1 (de) 2008-04-22 2009-10-28 Bayer CropScience Aktiengesellschaft 2-[(1h-Pyrazol-4-ylmethyl)-sulfonyl]-Oxazol-Derivate, 2-[(1H-Pyrazol-4-ylmethyl)-sulfanyl]-Oxazol-Derivate und chirale 2-[(1H-Pyrazol-4-ylmethyl)-sulfinyl]-Oxazol-Derivate, Verfahren zu deren Herstellung sowie deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren
EP2272846A1 (de) * 2009-06-23 2011-01-12 Bayer CropScience AG Thiazolylpiperidin Derivate als Fungizide
CN103145626B (zh) * 2013-02-28 2015-02-11 山东大学 一种合成4-氨基-2-甲巯基嘧啶-5-甲醛的方法
IL292532B1 (en) 2019-10-31 2024-04-01 Kumiai Chemical Industry Co Process for the production of herbicide and its intermediates
CN113754648B (zh) * 2020-06-02 2023-02-17 山东润博生物科技有限公司 一种砜吡草唑及其中间体的制备方法
CN112110912B (zh) * 2020-07-31 2022-07-05 绍兴贝斯美化工股份有限公司 一种合成硫醚类中间体的方法
CN114075149A (zh) * 2020-08-20 2022-02-22 宁夏苏融达化工有限公司 含二氟苯基的杂环化合物及其应用
AU2022280405A1 (en) * 2021-05-27 2023-11-30 Upl Limited Novel intermediate for preparation of pyroxasulfone
WO2023194957A1 (en) * 2022-04-08 2023-10-12 Upl Limited A process for preparation of 3-[5-(difluoromethoxy)-1- methyl-3-(trifluoromethyl)pyrazol-4- ylmethylsulfonyl]-4,5-dihydro-5,5-dimethyl-1,2-oxazole and its intermediates

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004013106A1 (ja) * 2002-08-01 2004-02-12 Ihara Chemical Industry Co., Ltd. ピラゾール誘導体及びその製造方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU769834B2 (en) * 1999-08-10 2004-02-05 Ihara Chemical Industry Co. Ltd. Isoxazoline derivatives and herbicides containing the same as the active ingredient
JP4465133B2 (ja) * 2001-02-08 2010-05-19 クミアイ化学工業株式会社 イソオキサゾリン誘導体及びこれを有効成分とする除草剤
JP4317445B2 (ja) * 2001-06-21 2009-08-19 クミアイ化学工業株式会社 イソオキサゾリン誘導体及び除草剤

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004013106A1 (ja) * 2002-08-01 2004-02-12 Ihara Chemical Industry Co., Ltd. ピラゾール誘導体及びその製造方法
EP1541561A1 (de) * 2002-08-01 2005-06-15 IHARA CHEMICAL INDUSTRY Co., Ltd. Pyrazolderivate und verfahren zu deren herstellung

Also Published As

Publication number Publication date
JP2008544996A (ja) 2008-12-11
KR20080030605A (ko) 2008-04-04
BRPI0612729A2 (pt) 2010-11-30
DE102005031583A1 (de) 2007-01-25
US20070015805A1 (en) 2007-01-18
CA2614239A1 (en) 2007-01-11
WO2007003295A2 (de) 2007-01-11
EP1902038A2 (de) 2008-03-26
CN101213181A (zh) 2008-07-02
IL188431A0 (en) 2008-11-03

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