UY32353A - Compuestos de soluciones oculares tópicas para suministrar concentraciones efectivas del agente activo al segmento posterior del ojo - Google Patents

Compuestos de soluciones oculares tópicas para suministrar concentraciones efectivas del agente activo al segmento posterior del ojo

Info

Publication number
UY32353A
UY32353A UY0001032353A UY32353A UY32353A UY 32353 A UY32353 A UY 32353A UY 0001032353 A UY0001032353 A UY 0001032353A UY 32353 A UY32353 A UY 32353A UY 32353 A UY32353 A UY 32353A
Authority
UY
Uruguay
Prior art keywords
active agent
effective concentrations
eye segment
back eye
supply effective
Prior art date
Application number
UY0001032353A
Other languages
English (en)
Inventor
Masood A Chowhan
Original Assignee
Alcon Res Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alcon Res Ltd filed Critical Alcon Res Ltd
Publication of UY32353A publication Critical patent/UY32353A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Ophthalmology & Optometry (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Compuestos farmacéuticos que contienen tandospirona para la administración ocular tópica. Los compuestos son útiles para suministrar tandospirona al segmento posterior del ojo, a efecto de tratar desordenes que afectan dichos tejidos.
UY0001032353A 2008-12-22 2009-12-21 Compuestos de soluciones oculares tópicas para suministrar concentraciones efectivas del agente activo al segmento posterior del ojo UY32353A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13970108P 2008-12-22 2008-12-22

Publications (1)

Publication Number Publication Date
UY32353A true UY32353A (es) 2010-04-30

Family

ID=41559537

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032353A UY32353A (es) 2008-12-22 2009-12-21 Compuestos de soluciones oculares tópicas para suministrar concentraciones efectivas del agente activo al segmento posterior del ojo

Country Status (15)

Country Link
US (1) US20100160342A1 (es)
EP (1) EP2367528A1 (es)
JP (1) JP2012513393A (es)
KR (1) KR20110099044A (es)
CN (1) CN102264344A (es)
AR (1) AR074828A1 (es)
AU (1) AU2009330517A1 (es)
BR (1) BRPI0923502A2 (es)
CA (1) CA2747917A1 (es)
CL (1) CL2009002197A1 (es)
MX (1) MX2011005586A (es)
RU (1) RU2011130552A (es)
TW (1) TW201028176A (es)
UY (1) UY32353A (es)
WO (1) WO2010074961A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103664905B (zh) * 2013-12-25 2015-10-14 四川科瑞德制药有限公司 盐酸坦度螺酮晶型ii及其制备方法
CN108619100B (zh) * 2017-03-16 2022-05-13 四川科瑞德制药股份有限公司 一种氮杂螺酮类药物注射剂及其制备方法和用途

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4407791A (en) * 1981-09-28 1983-10-04 Alcon Laboratories, Inc. Ophthalmic solutions
US5648348A (en) * 1991-10-28 1997-07-15 Mona Industries, Inc. Phospholipid antimicrobial compositions
US5286719A (en) * 1991-10-28 1994-02-15 Mona Industries, Inc. Phospholipid virucidal compositions
CA2166722A1 (en) * 1994-05-06 1995-11-16 Manoj L. Maniar Use of vitamin e tocopheryl derivatives in ophthalmic compositions
US5874469A (en) * 1996-01-05 1999-02-23 Alcon Laboratories, Inc. Fluoroalkyl hydrocarbons for administering water insoluble or unstable drugs
PT877600E (pt) * 1996-08-09 2004-02-27 Alcon Mfg Ltd Sistemas conservantes para composicoes farmaceuticas contendo ciclodextrinas
US6120758A (en) * 1998-07-16 2000-09-19 Shaklee Corporation Preservative system for topically applied products
US20030207890A1 (en) * 2001-02-23 2003-11-06 Collier Robert J Compounds with 5-ht1a activity useful for treating disorders of the outer retina
PE20020578A1 (es) * 2000-10-10 2002-08-14 Upjohn Co Una composicion de antibiotico topico para el tratamiento de infecciones oculares
JP2004262812A (ja) * 2003-02-28 2004-09-24 Rohto Pharmaceut Co Ltd 眼圧低下剤
US6969706B1 (en) * 2004-05-12 2005-11-29 Allergan, Inc. Preserved pharmaceutical compositions comprising cyclodextrins
MX2009000885A (es) * 2006-07-25 2009-02-05 Osmotica Corp Soluciones oftalmicas.
TWI394564B (zh) * 2006-09-21 2013-05-01 Alcon Res Ltd 自行保存型水性藥學組成物
TW200904485A (en) * 2007-05-18 2009-02-01 Alcon Res Ltd Phospholipid compositions for contact lens care and preservation of pharmaceutical compositions
AU2009223649B2 (en) * 2008-03-11 2013-08-29 Novartis Ag Low viscosity, highly flocculated triamcinolone acetonide suspensions for intravitreal injection
TW201010727A (en) * 2008-09-03 2010-03-16 Alcon Res Ltd Pharmaceutical composition having relatively low ionic strength

Also Published As

Publication number Publication date
WO2010074961A1 (en) 2010-07-01
CN102264344A (zh) 2011-11-30
AU2009330517A1 (en) 2010-07-01
TW201028176A (en) 2010-08-01
EP2367528A1 (en) 2011-09-28
JP2012513393A (ja) 2012-06-14
RU2011130552A (ru) 2013-01-27
CA2747917A1 (en) 2010-07-01
AR074828A1 (es) 2011-02-16
US20100160342A1 (en) 2010-06-24
BRPI0923502A2 (pt) 2019-09-24
CL2009002197A1 (es) 2011-02-11
KR20110099044A (ko) 2011-09-05
MX2011005586A (es) 2011-06-20

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Legal Events

Date Code Title Description
RDES Application refused

Effective date: 20201223