UY31921A - Combinación de derivados de amidina con depsipeptidos ciclicos - Google Patents

Combinación de derivados de amidina con depsipeptidos ciclicos

Info

Publication number
UY31921A
UY31921A UY0001031921A UY31921A UY31921A UY 31921 A UY31921 A UY 31921A UY 0001031921 A UY0001031921 A UY 0001031921A UY 31921 A UY31921 A UY 31921A UY 31921 A UY31921 A UY 31921A
Authority
UY
Uruguay
Prior art keywords
combination
derivatives
amidina
depsipeptides
cycle
Prior art date
Application number
UY0001031921A
Other languages
English (en)
Inventor
Achim Dr Harder
Dr Venkata-Rangarao Kanikanti
Dr Thomas Bach
Dr Richard Kujanek
Dr Dittmar Nerger
Original Assignee
Bayer Animal Health Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Animal Health Gmbh filed Critical Bayer Animal Health Gmbh
Publication of UY31921A publication Critical patent/UY31921A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15Depsipeptides; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se refiere a la combinación de derivados de aminofenalamida con depsipéptidos cíclicos, a productos que comprenden esta combinación y al uso de estas sustancias activas en combinación para controlar endoparásitos en seres humanos y en animales.
UY0001031921A 2008-06-28 2009-06-18 Combinación de derivados de amidina con depsipeptidos ciclicos UY31921A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102008030764A DE102008030764A1 (de) 2008-06-28 2008-06-28 Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden

Publications (1)

Publication Number Publication Date
UY31921A true UY31921A (es) 2010-01-29

Family

ID=41010493

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001031921A UY31921A (es) 2008-06-28 2009-06-18 Combinación de derivados de amidina con depsipeptidos ciclicos

Country Status (13)

Country Link
US (1) US20110201550A1 (es)
EP (1) EP2299995A1 (es)
JP (1) JP2011526262A (es)
AR (1) AR073180A1 (es)
AU (1) AU2009262581A1 (es)
BR (1) BRPI0913996A2 (es)
CA (1) CA2729420A1 (es)
DE (1) DE102008030764A1 (es)
MX (1) MX2010014442A (es)
TW (1) TW201012471A (es)
UY (1) UY31921A (es)
WO (1) WO2009156071A1 (es)
ZA (1) ZA201009064B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102344391B (zh) * 2011-07-28 2013-12-25 山东新华制药股份有限公司 N-(4-乙酰氨基苯基)-n′,n′-二甲基乙脒的合成方法
LT3298027T (lt) 2015-05-20 2021-08-10 Boehringer Ingelheim Animal Health USA Inc. Antihelmintiniai depsipeptido junginiai
AU2016380868B2 (en) 2015-12-28 2019-11-28 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
CN110167921A (zh) 2016-11-16 2019-08-23 勃林格殷格翰动物保健美国公司 驱蠕虫缩肽化合物
WO2020018888A1 (en) 2018-07-20 2020-01-23 The Board Of Regents Of The University Of Oklahoma Antimicrobial peptides and methods of use
CN114146074B (zh) * 2020-09-08 2024-03-01 中国疾病预防控制中心寄生虫病预防控制所(国家热带病研究中心) 抗寄生虫的药物组合及其应用、制备方法

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2029297A1 (de) * 1970-06-13 1971-12-30 Farbenfabriken Bayer Ag, 5090 Leverkusen Neue Aminophenyl-cycloamidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
DE2029299C3 (de) 1970-06-13 1980-08-21 Bayer Ag, 5090 Leverkusen Neue Aminophenylamidine, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel
DE2029298C3 (de) 1970-06-13 1980-04-17 Bayer Ag, 5090 Leverkusen Aminophenylamidine, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel
BE788743A (fr) * 1971-09-14 1973-03-13 Bayer Ag Nouveaux 2-(aminophenylimino)-3- aza-1-thia-cycloalcanes, leur procede de preparation et leur application comme
NO176766C (no) * 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
US5270037A (en) * 1990-07-12 1993-12-14 Boehringer Ingelheim Gmbh Use of interferon and a substance with an antimalarial activity for the treatment of malaria infections
DE69331414T2 (de) 1992-03-17 2002-08-08 Fujisawa Pharmaceutical Co., Ltd. Depsipeptide, herstellung und anwendung
DE4317458A1 (de) * 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
NZ261630A (en) 1993-02-19 1998-05-27 Meiji Seika Kaisha Heteromacrocyclic compound and use as an assthelmintie
DE4317457A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE4317432A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
AU686222B2 (en) * 1993-09-06 1998-02-05 Astellas Pharma Inc. Cyclodepsipeptide compound
DE4342907A1 (de) 1993-12-16 1995-06-22 Bayer Ag Neue cyclische Depsipeptide mit 18 Ringatomen und ihre Verwendung zur Bekämpfung von Endoparasiten
DE4401389A1 (de) 1994-01-19 1995-07-20 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 12 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 12 Ringatomen und Verfahren zu ihrer Herstellung
DE4406025A1 (de) * 1994-02-24 1995-08-31 Bayer Ag Milchsäure-haltige cyclische Depsipeptide mit 18 Ringatomen als endoparasitizide Mittel und Verfahren zu ihrer Herstellung
DE4412492A1 (de) 1994-04-12 1995-10-19 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen
DE4437198A1 (de) * 1994-10-18 1996-04-25 Bayer Ag Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden
CN1162409C (zh) * 1995-06-30 2004-08-18 藤泽药品工业株式会社 缩肽衍生物、其新型中间体以及中间体的制造方法
IL123776A (en) 1995-09-22 2002-09-12 Bayer Ag History of Cyclodepsipeptide 1022 PF
DE19545639A1 (de) 1995-12-07 1997-06-12 Bayer Ag Verfahren zur Herstellung von substituierten Arylmilchsäure-haltigen Cyclodepsipeptiden mit 24 Ringatomen
WO1998037088A1 (en) 1997-02-19 1998-08-27 Meiji Seika Kaisha Ltd. Derivatives of cyclodepsipeptide, pf1022 substance
DE19713626A1 (de) 1997-04-02 1998-10-08 Bayer Ag Neue Thiodepsipeptide zur Bekämpfung von Endoparasiten und ein einfaches Verfahren zu ihrer Herstellung
NZ501478A (en) * 1997-06-04 2001-05-25 Bayer Ag 8,20-bis-(substituted benzyl)-desoxycyclodepsipeptides and their use for combatting endoparasites
DE19811559A1 (de) 1998-03-17 1999-09-23 Bayer Ag Cyclooctadepsipeptide
DE19828047A1 (de) 1998-06-24 1999-12-30 Bayer Ag Substituierte Cyclooctadepsipeptide
DE19840320A1 (de) 1998-09-04 2000-03-09 Bayer Ag Aza-Cyclodepsipeptide
DE102007061262A1 (de) 2007-12-19 2009-06-25 Bayer Animal Health Gmbh Neue Verwendung von Tribendimidin

Also Published As

Publication number Publication date
MX2010014442A (es) 2011-01-21
DE102008030764A1 (de) 2009-12-31
JP2011526262A (ja) 2011-10-06
AU2009262581A1 (en) 2009-12-30
BRPI0913996A2 (pt) 2015-10-20
WO2009156071A1 (de) 2009-12-30
WO2009156071A8 (de) 2010-12-29
US20110201550A1 (en) 2011-08-18
TW201012471A (en) 2010-04-01
EP2299995A1 (de) 2011-03-30
ZA201009064B (en) 2012-02-29
CA2729420A1 (en) 2009-12-30
AR073180A1 (es) 2010-10-20

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20181106