AR073180A1 - Productos que contienen derivados de amidina con depsipeptidos ciclicos - Google Patents

Productos que contienen derivados de amidina con depsipeptidos ciclicos

Info

Publication number
AR073180A1
AR073180A1 ARP090102325A ARP090102325A AR073180A1 AR 073180 A1 AR073180 A1 AR 073180A1 AR P090102325 A ARP090102325 A AR P090102325A AR P090102325 A ARP090102325 A AR P090102325A AR 073180 A1 AR073180 A1 AR 073180A1
Authority
AR
Argentina
Prior art keywords
amidina
depsipeptides
cycle
products containing
containing derivatives
Prior art date
Application number
ARP090102325A
Other languages
English (en)
Original Assignee
Bayer Animal Health Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Animal Health Gmbh filed Critical Bayer Animal Health Gmbh
Publication of AR073180A1 publication Critical patent/AR073180A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15Depsipeptides; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Combinacion de derivados de aminofenilamidina con depsipéptidos cíclicos, productos que comprenden esta combinacion y uso de estas sustancias activas en combinacion para controlar endoparásitos en seres humanos y en animales.
ARP090102325A 2008-06-28 2009-06-24 Productos que contienen derivados de amidina con depsipeptidos ciclicos AR073180A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102008030764A DE102008030764A1 (de) 2008-06-28 2008-06-28 Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden

Publications (1)

Publication Number Publication Date
AR073180A1 true AR073180A1 (es) 2010-10-20

Family

ID=41010493

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP090102325A AR073180A1 (es) 2008-06-28 2009-06-24 Productos que contienen derivados de amidina con depsipeptidos ciclicos

Country Status (13)

Country Link
US (1) US20110201550A1 (es)
EP (1) EP2299995A1 (es)
JP (1) JP2011526262A (es)
AR (1) AR073180A1 (es)
AU (1) AU2009262581A1 (es)
BR (1) BRPI0913996A2 (es)
CA (1) CA2729420A1 (es)
DE (1) DE102008030764A1 (es)
MX (1) MX2010014442A (es)
TW (1) TW201012471A (es)
UY (1) UY31921A (es)
WO (1) WO2009156071A1 (es)
ZA (1) ZA201009064B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102344391B (zh) * 2011-07-28 2013-12-25 山东新华制药股份有限公司 N-(4-乙酰氨基苯基)-n′,n′-二甲基乙脒的合成方法
SG10202103403SA (en) 2015-05-20 2021-05-28 Boehringer Ingelheim Animal Health Usa Inc Anthelmintic depsipeptide compounds
SG11201805368YA (en) 2015-12-28 2018-07-30 Merial Inc Anthelmintic depsipeptide compounds
EP3541789A1 (en) 2016-11-16 2019-09-25 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
WO2020018888A1 (en) 2018-07-20 2020-01-23 The Board Of Regents Of The University Of Oklahoma Antimicrobial peptides and methods of use
CN114146074B (zh) * 2020-09-08 2024-03-01 中国疾病预防控制中心寄生虫病预防控制所(国家热带病研究中心) 抗寄生虫的药物组合及其应用、制备方法

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2029297A1 (de) * 1970-06-13 1971-12-30 Farbenfabriken Bayer Ag, 5090 Leverkusen Neue Aminophenyl-cycloamidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
DE2029299C3 (de) * 1970-06-13 1980-08-21 Bayer Ag, 5090 Leverkusen Neue Aminophenylamidine, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel
DE2029298C3 (de) 1970-06-13 1980-04-17 Bayer Ag, 5090 Leverkusen Aminophenylamidine, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel
BE788743A (fr) 1971-09-14 1973-03-13 Bayer Ag Nouveaux 2-(aminophenylimino)-3- aza-1-thia-cycloalcanes, leur procede de preparation et leur application comme
NO176766C (no) 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
US5270037A (en) * 1990-07-12 1993-12-14 Boehringer Ingelheim Gmbh Use of interferon and a substance with an antimalarial activity for the treatment of malaria infections
DK0634408T3 (da) 1992-03-17 2002-04-22 Fujisawa Pharmaceutical Co Depsipeptidderivater, fremstilling og anvendelse deraf
DE4317458A1 (de) * 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
WO1994019334A1 (en) * 1993-02-19 1994-09-01 Meiji Seika Kaisha, Ltd. Pf1022 derivative, cyclic depsipeptide
DE4317457A1 (de) 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE4317432A1 (de) 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
WO1995007272A1 (en) * 1993-09-06 1995-03-16 Fujisawa Pharmaceutical Co., Ltd. Cyclodepsipeptide compound
DE4342907A1 (de) 1993-12-16 1995-06-22 Bayer Ag Neue cyclische Depsipeptide mit 18 Ringatomen und ihre Verwendung zur Bekämpfung von Endoparasiten
DE4401389A1 (de) 1994-01-19 1995-07-20 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 12 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 12 Ringatomen und Verfahren zu ihrer Herstellung
DE4406025A1 (de) * 1994-02-24 1995-08-31 Bayer Ag Milchsäure-haltige cyclische Depsipeptide mit 18 Ringatomen als endoparasitizide Mittel und Verfahren zu ihrer Herstellung
DE4412492A1 (de) 1994-04-12 1995-10-19 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen
DE4437198A1 (de) 1994-10-18 1996-04-25 Bayer Ag Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden
DE69637876D1 (de) 1995-06-30 2009-04-30 Astellas Pharma Inc Ng und zwischenprodukt dafür
WO1997011064A1 (fr) * 1995-09-22 1997-03-27 Meiji Seika Kaisha, Ltd. Nouveaux derives depsipeptides cycliques de pf1022
DE19545639A1 (de) 1995-12-07 1997-06-12 Bayer Ag Verfahren zur Herstellung von substituierten Arylmilchsäure-haltigen Cyclodepsipeptiden mit 24 Ringatomen
WO1998037088A1 (en) 1997-02-19 1998-08-27 Meiji Seika Kaisha Ltd. Derivatives of cyclodepsipeptide, pf1022 substance
DE19713626A1 (de) * 1997-04-02 1998-10-08 Bayer Ag Neue Thiodepsipeptide zur Bekämpfung von Endoparasiten und ein einfaches Verfahren zu ihrer Herstellung
NZ501478A (en) * 1997-06-04 2001-05-25 Bayer Ag 8,20-bis-(substituted benzyl)-desoxycyclodepsipeptides and their use for combatting endoparasites
DE19811559A1 (de) 1998-03-17 1999-09-23 Bayer Ag Cyclooctadepsipeptide
DE19828047A1 (de) 1998-06-24 1999-12-30 Bayer Ag Substituierte Cyclooctadepsipeptide
DE19840320A1 (de) 1998-09-04 2000-03-09 Bayer Ag Aza-Cyclodepsipeptide
DE102007061262A1 (de) 2007-12-19 2009-06-25 Bayer Animal Health Gmbh Neue Verwendung von Tribendimidin

Also Published As

Publication number Publication date
WO2009156071A1 (de) 2009-12-30
ZA201009064B (en) 2012-02-29
EP2299995A1 (de) 2011-03-30
CA2729420A1 (en) 2009-12-30
MX2010014442A (es) 2011-01-21
BRPI0913996A2 (pt) 2015-10-20
WO2009156071A8 (de) 2010-12-29
JP2011526262A (ja) 2011-10-06
TW201012471A (en) 2010-04-01
US20110201550A1 (en) 2011-08-18
UY31921A (es) 2010-01-29
AU2009262581A1 (en) 2009-12-30
DE102008030764A1 (de) 2009-12-31

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