AR073180A1 - Productos que contienen derivados de amidina con depsipeptidos ciclicos - Google Patents
Productos que contienen derivados de amidina con depsipeptidos ciclicosInfo
- Publication number
- AR073180A1 AR073180A1 ARP090102325A ARP090102325A AR073180A1 AR 073180 A1 AR073180 A1 AR 073180A1 AR P090102325 A ARP090102325 A AR P090102325A AR P090102325 A ARP090102325 A AR P090102325A AR 073180 A1 AR073180 A1 AR 073180A1
- Authority
- AR
- Argentina
- Prior art keywords
- amidina
- depsipeptides
- cycle
- products containing
- containing derivatives
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/15—Depsipeptides; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Tropical Medicine & Parasitology (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Combinacion de derivados de aminofenilamidina con depsipéptidos cíclicos, productos que comprenden esta combinacion y uso de estas sustancias activas en combinacion para controlar endoparásitos en seres humanos y en animales.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE102008030764A DE102008030764A1 (de) | 2008-06-28 | 2008-06-28 | Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden |
Publications (1)
Publication Number | Publication Date |
---|---|
AR073180A1 true AR073180A1 (es) | 2010-10-20 |
Family
ID=41010493
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP090102325A AR073180A1 (es) | 2008-06-28 | 2009-06-24 | Productos que contienen derivados de amidina con depsipeptidos ciclicos |
Country Status (13)
Country | Link |
---|---|
US (1) | US20110201550A1 (es) |
EP (1) | EP2299995A1 (es) |
JP (1) | JP2011526262A (es) |
AR (1) | AR073180A1 (es) |
AU (1) | AU2009262581A1 (es) |
BR (1) | BRPI0913996A2 (es) |
CA (1) | CA2729420A1 (es) |
DE (1) | DE102008030764A1 (es) |
MX (1) | MX2010014442A (es) |
TW (1) | TW201012471A (es) |
UY (1) | UY31921A (es) |
WO (1) | WO2009156071A1 (es) |
ZA (1) | ZA201009064B (es) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102344391B (zh) * | 2011-07-28 | 2013-12-25 | 山东新华制药股份有限公司 | N-(4-乙酰氨基苯基)-n′,n′-二甲基乙脒的合成方法 |
SG10202103403SA (en) | 2015-05-20 | 2021-05-28 | Boehringer Ingelheim Animal Health Usa Inc | Anthelmintic depsipeptide compounds |
SG11201805368YA (en) | 2015-12-28 | 2018-07-30 | Merial Inc | Anthelmintic depsipeptide compounds |
EP3541789A1 (en) | 2016-11-16 | 2019-09-25 | Boehringer Ingelheim Animal Health USA Inc. | Anthelmintic depsipeptide compounds |
WO2020018888A1 (en) | 2018-07-20 | 2020-01-23 | The Board Of Regents Of The University Of Oklahoma | Antimicrobial peptides and methods of use |
CN114146074B (zh) * | 2020-09-08 | 2024-03-01 | 中国疾病预防控制中心寄生虫病预防控制所(国家热带病研究中心) | 抗寄生虫的药物组合及其应用、制备方法 |
Family Cites Families (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2029297A1 (de) * | 1970-06-13 | 1971-12-30 | Farbenfabriken Bayer Ag, 5090 Leverkusen | Neue Aminophenyl-cycloamidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
DE2029299C3 (de) * | 1970-06-13 | 1980-08-21 | Bayer Ag, 5090 Leverkusen | Neue Aminophenylamidine, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel |
DE2029298C3 (de) | 1970-06-13 | 1980-04-17 | Bayer Ag, 5090 Leverkusen | Aminophenylamidine, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel |
BE788743A (fr) | 1971-09-14 | 1973-03-13 | Bayer Ag | Nouveaux 2-(aminophenylimino)-3- aza-1-thia-cycloalcanes, leur procede de preparation et leur application comme |
NO176766C (no) | 1989-02-07 | 1995-05-24 | Meiji Seika Kaisha | Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet |
US5270037A (en) * | 1990-07-12 | 1993-12-14 | Boehringer Ingelheim Gmbh | Use of interferon and a substance with an antimalarial activity for the treatment of malaria infections |
DK0634408T3 (da) | 1992-03-17 | 2002-04-22 | Fujisawa Pharmaceutical Co | Depsipeptidderivater, fremstilling og anvendelse deraf |
DE4317458A1 (de) * | 1992-06-11 | 1993-12-16 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung |
WO1994019334A1 (en) * | 1993-02-19 | 1994-09-01 | Meiji Seika Kaisha, Ltd. | Pf1022 derivative, cyclic depsipeptide |
DE4317457A1 (de) | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
DE4317432A1 (de) | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
WO1995007272A1 (en) * | 1993-09-06 | 1995-03-16 | Fujisawa Pharmaceutical Co., Ltd. | Cyclodepsipeptide compound |
DE4342907A1 (de) | 1993-12-16 | 1995-06-22 | Bayer Ag | Neue cyclische Depsipeptide mit 18 Ringatomen und ihre Verwendung zur Bekämpfung von Endoparasiten |
DE4401389A1 (de) | 1994-01-19 | 1995-07-20 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 12 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 12 Ringatomen und Verfahren zu ihrer Herstellung |
DE4406025A1 (de) * | 1994-02-24 | 1995-08-31 | Bayer Ag | Milchsäure-haltige cyclische Depsipeptide mit 18 Ringatomen als endoparasitizide Mittel und Verfahren zu ihrer Herstellung |
DE4412492A1 (de) | 1994-04-12 | 1995-10-19 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen |
DE4437198A1 (de) | 1994-10-18 | 1996-04-25 | Bayer Ag | Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden |
DE69637876D1 (de) | 1995-06-30 | 2009-04-30 | Astellas Pharma Inc | Ng und zwischenprodukt dafür |
WO1997011064A1 (fr) * | 1995-09-22 | 1997-03-27 | Meiji Seika Kaisha, Ltd. | Nouveaux derives depsipeptides cycliques de pf1022 |
DE19545639A1 (de) | 1995-12-07 | 1997-06-12 | Bayer Ag | Verfahren zur Herstellung von substituierten Arylmilchsäure-haltigen Cyclodepsipeptiden mit 24 Ringatomen |
WO1998037088A1 (en) | 1997-02-19 | 1998-08-27 | Meiji Seika Kaisha Ltd. | Derivatives of cyclodepsipeptide, pf1022 substance |
DE19713626A1 (de) * | 1997-04-02 | 1998-10-08 | Bayer Ag | Neue Thiodepsipeptide zur Bekämpfung von Endoparasiten und ein einfaches Verfahren zu ihrer Herstellung |
NZ501478A (en) * | 1997-06-04 | 2001-05-25 | Bayer Ag | 8,20-bis-(substituted benzyl)-desoxycyclodepsipeptides and their use for combatting endoparasites |
DE19811559A1 (de) | 1998-03-17 | 1999-09-23 | Bayer Ag | Cyclooctadepsipeptide |
DE19828047A1 (de) | 1998-06-24 | 1999-12-30 | Bayer Ag | Substituierte Cyclooctadepsipeptide |
DE19840320A1 (de) | 1998-09-04 | 2000-03-09 | Bayer Ag | Aza-Cyclodepsipeptide |
DE102007061262A1 (de) | 2007-12-19 | 2009-06-25 | Bayer Animal Health Gmbh | Neue Verwendung von Tribendimidin |
-
2008
- 2008-06-28 DE DE102008030764A patent/DE102008030764A1/de not_active Withdrawn
-
2009
- 2009-06-16 EP EP09768920A patent/EP2299995A1/de not_active Withdrawn
- 2009-06-16 MX MX2010014442A patent/MX2010014442A/es not_active Application Discontinuation
- 2009-06-16 CA CA2729420A patent/CA2729420A1/en not_active Abandoned
- 2009-06-16 AU AU2009262581A patent/AU2009262581A1/en not_active Abandoned
- 2009-06-16 WO PCT/EP2009/004304 patent/WO2009156071A1/de active Application Filing
- 2009-06-16 US US13/000,510 patent/US20110201550A1/en not_active Abandoned
- 2009-06-16 BR BRPI0913996A patent/BRPI0913996A2/pt not_active IP Right Cessation
- 2009-06-16 JP JP2011515161A patent/JP2011526262A/ja active Pending
- 2009-06-18 UY UY0001031921A patent/UY31921A/es not_active Application Discontinuation
- 2009-06-24 AR ARP090102325A patent/AR073180A1/es unknown
- 2009-06-26 TW TW098121497A patent/TW201012471A/zh unknown
-
2010
- 2010-12-17 ZA ZA2010/09064A patent/ZA201009064B/en unknown
Also Published As
Publication number | Publication date |
---|---|
WO2009156071A1 (de) | 2009-12-30 |
ZA201009064B (en) | 2012-02-29 |
EP2299995A1 (de) | 2011-03-30 |
CA2729420A1 (en) | 2009-12-30 |
MX2010014442A (es) | 2011-01-21 |
BRPI0913996A2 (pt) | 2015-10-20 |
WO2009156071A8 (de) | 2010-12-29 |
JP2011526262A (ja) | 2011-10-06 |
TW201012471A (en) | 2010-04-01 |
US20110201550A1 (en) | 2011-08-18 |
UY31921A (es) | 2010-01-29 |
AU2009262581A1 (en) | 2009-12-30 |
DE102008030764A1 (de) | 2009-12-31 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CY1120407T1 (el) | Φαρμακοτεχνικες μορφες ινσουλινων μακρας-δρασεως | |
CL2011001232A1 (es) | Combinacion farmaceutica que comprende un anticuerpo que reconoce especificamente la cd38 y al menos citarabina; y su uso para el tratamiento de cancer | |
CL2012003657A1 (es) | Formulacion estable que comprende la proteina iduronato -2- sulfatasa y un tensoactivo de polisorbato; contenedor que comprende dicha formulacion; uso de dicha formulacion para tratar sindrome de hunters. | |
CL2012001950A1 (es) | Uso de una cepa bacteriana probiotico en la fabricacion de un medicamento o composicion nutricional en humanos o animales para alterar los patrones del sueño | |
CL2014002348A1 (es) | Compuestos derivados de fenicol; composicion farmaceutica que los comprende; y su uso para controlar o tratar infecciones bacterianas en ganado. | |
BRPI0919193A2 (pt) | Uso de lipídeo, e, composição nutricional | |
CL2013003577A1 (es) | Uso de una composicion farmaceutica que comprende panobinostat y ruxolitinib en la prevencion y/o tratamiento de neoplasias mieloproliferativas. | |
BRPI0914678A8 (pt) | Dispositivo dispensador para vaso sanitário e processo para distribuir uma composição de tratamento a um dispositivo sanitário | |
BR112015015898A8 (pt) | composição farmacêutica de solução sólida, e, uso de uma composição farmacêutica | |
CL2012003516A1 (es) | Compuesto derivado de 5-fenil-5-trifluorometil-4,5-dihidroisoxazol; composicion que lo comprende; y su uso para controlar piojos de mar en peces. | |
ECSP109852A (es) | Uso de homo y copolímeros para la estabilización de formulaciones de principios activos | |
CL2008002381A1 (es) | Oligonucleotido inmunoestimulador; composicion farmaceutica que lo comprende; y su uso para tratar un trastorno o afeccion en un sujeto, incluyendo cancer. | |
BR112015015870A8 (pt) | composição farmacêutica, e, uso de uma composição farmacêutica | |
BRPI0923164A2 (pt) | formulações de imiquimod com concentração de dosagem menos e regimes de dosagem curtos para o tratamento de ceratose actínica. | |
SV2009003366A (es) | Estabilizacion de vitamina b12 | |
AR073180A1 (es) | Productos que contienen derivados de amidina con depsipeptidos ciclicos | |
EA201200484A1 (ru) | Фармацевтическая композиция с действующими веществами - метформином и ситаглиптином или вилдаглиптином | |
NI201000189A (es) | Formulación de medicamento sólido con liberación retardadas. | |
GT201200304A (es) | Composiciones farmacéuticas que comprenden hidromorfona y naloxona | |
CL2011001058A1 (es) | Combinaciones plagicidas que comprenden cetoenoles ciclicos y spinetoram; uso de dichas combinaciones y metodos que emplean la misma para combatir plagas animales. | |
BRPI0812331A2 (pt) | Umidificador descartável para uso com produtos de tabaco e embalagem para produtos de tabaco | |
CL2012003265A1 (es) | Polisacarido de semillas de tamarindo para usarse en el tratamiento de enfermedades infecciosas; composicion farmacéutica y/o dermocosmética antiinflamatoria que contiene dicho polisacárido; uso de un polisacárido de semilla de tamarindo. | |
CR20140293A (es) | Preparaciones que comprenden emodepsido amorfo | |
BRPI0923642A2 (pt) | dispositivo de dosagem para gerar um fluxo de gás com uma substância ativa finamente dispersada no último. | |
CL2009000665A1 (es) | Compuestos derivados de pirrolidinilo; composicion farmaceutica que comprende a dichos compuestos; y su uso en el tratamiento de la ansiedad, depresion o ambas. |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB | Suspension of granting procedure |