UY31853A - Derivados sustituidos de2,3-oxo-n-(4-(trifluorometoxi)bencil)isoindolina-1-carboxamidas, composiciones conteniéndolos y aplicaciones - Google Patents

Derivados sustituidos de2,3-oxo-n-(4-(trifluorometoxi)bencil)isoindolina-1-carboxamidas, composiciones conteniéndolos y aplicaciones

Info

Publication number
UY31853A
UY31853A UY0001031853A UY31853A UY31853A UY 31853 A UY31853 A UY 31853A UY 0001031853 A UY0001031853 A UY 0001031853A UY 31853 A UY31853 A UY 31853A UY 31853 A UY31853 A UY 31853A
Authority
UY
Uruguay
Prior art keywords
isoindolina
trifluorometoxi
bencil
carboxamides
oxo
Prior art date
Application number
UY0001031853A
Other languages
English (en)
Inventor
Per I Arvidsson
Besidski Yevgenu
Linda I Nilsson
Ahlin Kristofer
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY31853A publication Critical patent/UY31853A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44Iso-indoles; Hydrogenated iso-indoles
    • C07D209/46Iso-indoles; Hydrogenated iso-indoles with an oxygen atom in position 1
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Se reivindica un compuesto de la Fórmula I en donde R1, R2, R3, m, L1 y L2 son como se definieron en la Memoria y Reivindicaciones.
UY0001031853A 2008-05-30 2009-05-29 Derivados sustituidos de2,3-oxo-n-(4-(trifluorometoxi)bencil)isoindolina-1-carboxamidas, composiciones conteniéndolos y aplicaciones UY31853A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US5731908P 2008-05-30 2008-05-30

Publications (1)

Publication Number Publication Date
UY31853A true UY31853A (es) 2010-01-05

Family

ID=41377344

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001031853A UY31853A (es) 2008-05-30 2009-05-29 Derivados sustituidos de2,3-oxo-n-(4-(trifluorometoxi)bencil)isoindolina-1-carboxamidas, composiciones conteniéndolos y aplicaciones

Country Status (6)

Country Link
AR (1) AR071956A1 (es)
CL (1) CL2009001330A1 (es)
PE (1) PE20091947A1 (es)
TW (1) TW201000447A (es)
UY (1) UY31853A (es)
WO (1) WO2009145719A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013007768A1 (en) 2011-07-13 2013-01-17 F. Hoffmann-La Roche Ag Tricyclic heterocyclic compounds, compositions and methods of use thereof as jak inhibitors
WO2015102929A1 (en) * 2013-12-30 2015-07-09 Novartis Ag Tricyclic sulfonamide derivatives
WO2018110669A1 (en) 2016-12-15 2018-06-21 Ono Pharmaceutical Co., Ltd. Activator of trek (twik related k+ channels) channels
CA3147397A1 (en) 2019-07-22 2021-01-28 Lupin Limited Macrocyclic compounds as sting agonists and methods and uses thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200613272A (en) * 2004-08-13 2006-05-01 Astrazeneca Ab Isoindolone compounds and their use as metabotropic glutamate receptor potentiators
TW200804281A (en) * 2006-02-16 2008-01-16 Astrazeneca Ab New metabotropic glutamate receptor-potentiating isoindolones
TW200812962A (en) * 2006-07-12 2008-03-16 Astrazeneca Ab New compounds I/418
WO2008008020A1 (en) * 2006-07-12 2008-01-17 Astrazeneca Ab 3-oxoisoindoline-1-carboxamide derivatives as analgesic agents
GB0705882D0 (en) * 2007-03-27 2007-05-02 Glaxo Group Ltd Novel compounds

Also Published As

Publication number Publication date
CL2009001330A1 (es) 2010-01-15
PE20091947A1 (es) 2010-01-28
TW201000447A (en) 2010-01-01
WO2009145719A1 (en) 2009-12-03
AR071956A1 (es) 2010-07-28

Similar Documents

Publication Publication Date Title
CY1119515T1 (el) Οξαζολο υποκατεστημενα ινδαζολια ως αναστολεις ρι3-κινασης
EA201001359A1 (ru) Гетероциклические соединения в качестве ингибиторов cxcr2
ECSP10010334A (es) Derivados de quinolina y su uso como fungicidas
CY1118104T1 (el) Νεα κυτταροστατικα νουκλεοζιδια 7-αποαζαπουρινης
EA201070519A1 (ru) Соединения тропана
UY36907A (es) Nuevas carboxamidas de acción microbiocida
CO6321282A2 (es) Derivados de piperidinilindol como inhibidores de aldosterona sintasa
CO6491116A2 (es) Derivados de 5-fluoropirimidinona
ATE554066T1 (de) Entzündungshemmende substituierte cyclobutendionverbindungen
CL2011002825A1 (es) Compuestos derivados de bencimidazol heteroarilo sustituido; composición farmacéutica que los comprende; y su uso en el tratamiento de la hepatitis c.
UY30670A1 (es) Nuevos compuestos de pirazolina, composiciones conteniéndolos y aplicaciones.
NI201000054A (es) Compuestos químicos.
DK2134691T3 (da) Quinolinonderivativer som parp- og tank-inhibitorer
EA201390877A1 (ru) Замещенные 6,6-конденсированные азотсодержащие гетероциклические соединения и их применение
GEP20156266B (en) Spiroheterocyclic n-oxypiperidines as pesticides
UY32292A (es) Agonistas de s1p1 y métodos de preparación y uso
UA106880C2 (uk) Нові гербіциди
CO6551705A2 (es) Derivados de 3.4.4a.10b- tetrahidro-1h-tiopirano-[4.3-c]- isoquinolina
TR201908180T4 (tr) N1-asil- 5-floropirimidinon deriveleri.
UY32667A (es) Nuevos derivados de furano espiroheterocíclico y tiofuranodiona
EA201270256A1 (ru) Производные т1-замещенного 5-фтор-2-оксопиримидинон-1 (2h) -карбоксамида
BRPI0909333A2 (pt) derivado de espiroindolinona
CR10637A (es) Fungicidas
UY30545A1 (es) Derivados sustituidos del acido acilamino-benzoico, composiciones que los contienen y aplicaciones
UY31853A (es) Derivados sustituidos de2,3-oxo-n-(4-(trifluorometoxi)bencil)isoindolina-1-carboxamidas, composiciones conteniéndolos y aplicaciones

Legal Events

Date Code Title Description
DESI Application deemed to be withdrawn

Effective date: 20130122