UY31252A1 - Derivados de macrolidos utiles en el tratamiento de la malaria - Google Patents
Derivados de macrolidos utiles en el tratamiento de la malariaInfo
- Publication number
- UY31252A1 UY31252A1 UY31252A UY31252A UY31252A1 UY 31252 A1 UY31252 A1 UY 31252A1 UY 31252 A UY31252 A UY 31252A UY 31252 A UY31252 A UY 31252A UY 31252 A1 UY31252 A1 UY 31252A1
- Authority
- UY
- Uruguay
- Prior art keywords
- derivatives
- malaria
- macrolides
- useful
- treatment
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
La presente invencion se refiere a nuevos derivados de 9-desoxo-9a-metil-9a-aza-9a-homoeritromicina A 2??-0-sustituida que tienen actividad contra la malaria. Más particularmente, la invencion se refiere a derivados de 9-desoxo-9a-metil-9a-aza-9a-homoeritromicina A 2??-0-sustituida y a 3-0-decladinosil-9-desoxo-9a-metil-9a-aza-9a-homoeritromicina A2??-0-sustituida que tienen actividad contra la malaria, a los intermedios para su preparacion, a los métodos para su preparacion, a su uso como agentes terapéuticos y a las sales de las mismas que tienen actividad contra la malaria.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US95264907P | 2007-07-30 | 2007-07-30 |
Publications (1)
Publication Number | Publication Date |
---|---|
UY31252A1 true UY31252A1 (es) | 2009-03-02 |
Family
ID=39874927
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY31252A UY31252A1 (es) | 2007-07-30 | 2008-07-29 | Derivados de macrolidos utiles en el tratamiento de la malaria |
Country Status (10)
Country | Link |
---|---|
US (1) | US20090036388A1 (es) |
EP (1) | EP2183265A1 (es) |
JP (1) | JP2010534709A (es) |
CN (1) | CN101809026A (es) |
AR (1) | AR067718A1 (es) |
CL (1) | CL2008002223A1 (es) |
PE (1) | PE20090879A1 (es) |
TW (1) | TW200922943A (es) |
UY (1) | UY31252A1 (es) |
WO (1) | WO2009016142A1 (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2012516305A (ja) | 2009-01-30 | 2012-07-19 | グラクソ グループ リミテッド | 好中球優位の炎症性疾患の治療のための9−デオキソ−9a−メチル−9a−アザ−9a−ホモエリスロマイシンa誘導体 |
WO2010086351A1 (en) * | 2009-01-30 | 2010-08-05 | Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. | 3'-n-substituted 9-deoxo-9a-methyl-9a-aza-homoerythromycin having antimalarial activity |
WO2011131749A1 (en) | 2010-04-23 | 2011-10-27 | Glaxo Group Limited | New 14 and 15 membered macrolides for the treatment of neutrophil dominated inflammatory diseases |
WO2021204423A1 (en) | 2020-04-05 | 2021-10-14 | University of Zagreb School of Medicine | Use of 15-membered azalides as active agents in the treatment of viral infections |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6407074B1 (en) * | 1997-06-11 | 2002-06-18 | Pfizer Inc | C-4″-substituted macrolide derivatives |
WO2006085228A2 (en) * | 2005-01-14 | 2006-08-17 | Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. | 9a-carbamoyl-y-aminopropyl and 9a-thiocarbamoyl-y-aminopropyl-azalides with antimalarial activity |
ATE429921T1 (de) * | 2005-01-14 | 2009-05-15 | Glaxosmithkline Zagreb | 9a-carbamoyl- und thiocarbamoylazalide mit antimalariawirkung |
-
2008
- 2008-07-25 PE PE2008001268A patent/PE20090879A1/es not_active Application Discontinuation
- 2008-07-28 AR ARP080103267A patent/AR067718A1/es not_active Application Discontinuation
- 2008-07-28 EP EP08775365A patent/EP2183265A1/en not_active Withdrawn
- 2008-07-28 US US12/180,675 patent/US20090036388A1/en not_active Abandoned
- 2008-07-28 WO PCT/EP2008/059848 patent/WO2009016142A1/en active Application Filing
- 2008-07-28 CN CN200880109593A patent/CN101809026A/zh active Pending
- 2008-07-28 JP JP2010518640A patent/JP2010534709A/ja active Pending
- 2008-07-29 TW TW097128544A patent/TW200922943A/zh unknown
- 2008-07-29 UY UY31252A patent/UY31252A1/es unknown
- 2008-07-29 CL CL2008002223A patent/CL2008002223A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
CN101809026A (zh) | 2010-08-18 |
JP2010534709A (ja) | 2010-11-11 |
PE20090879A1 (es) | 2009-07-25 |
CL2008002223A1 (es) | 2009-08-07 |
EP2183265A1 (en) | 2010-05-12 |
US20090036388A1 (en) | 2009-02-05 |
AR067718A1 (es) | 2009-10-21 |
TW200922943A (en) | 2009-06-01 |
WO2009016142A1 (en) | 2009-02-05 |
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