UY30228A1 - Compuestos quimicos - Google Patents
Compuestos quimicosInfo
- Publication number
- UY30228A1 UY30228A1 UY30228A UY30228A UY30228A1 UY 30228 A1 UY30228 A1 UY 30228A1 UY 30228 A UY30228 A UY 30228A UY 30228 A UY30228 A UY 30228A UY 30228 A1 UY30228 A1 UY 30228A1
- Authority
- UY
- Uruguay
- Prior art keywords
- chemical compounds
- compound
- pde4
- variables
- preparing
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
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- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
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- General Health & Medical Sciences (AREA)
- Public Health (AREA)
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- Dermatology (AREA)
- Urology & Nephrology (AREA)
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Abstract
La presente invencion proporciona un compuesto de a formula (I) : donde las variables se definen en la presente, un proceso para preparar dicho compuesto; y al uso de dicho compuesto en el tratamiento de una patología mediada por PDE4.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US78485506P | 2006-03-22 | 2006-03-22 | |
US88445607P | 2007-01-11 | 2007-01-11 |
Publications (1)
Publication Number | Publication Date |
---|---|
UY30228A1 true UY30228A1 (es) | 2007-10-31 |
Family
ID=38522713
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY30228A UY30228A1 (es) | 2006-03-22 | 2007-03-21 | Compuestos quimicos |
Country Status (7)
Country | Link |
---|---|
US (1) | US20090233907A1 (es) |
EP (1) | EP1999130A4 (es) |
JP (1) | JP2009530372A (es) |
AR (1) | AR060046A1 (es) |
TW (1) | TW200800997A (es) |
UY (1) | UY30228A1 (es) |
WO (1) | WO2007108750A1 (es) |
Families Citing this family (41)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL155367A0 (en) | 2000-10-23 | 2003-12-23 | Smithkline Beecham Corp | NOVEL 2,4,8-TRISUBSTITUTED-8h-PYRIDO[2,3,-d]PYRIMIDIN-7-ONE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME, PROCESSES FOR THE PREPARATION THEREOF, AND USE THEREOF IN THE PREPARATION OF MEDICAMENTS FOR TREATING CSBP/p38 KINASE MEDIATED DISEASES |
PE20061351A1 (es) * | 2005-03-25 | 2007-01-14 | Glaxo Group Ltd | COMPUESTOS 8H-PIRIDO[2,3-d]PIRIMIDIN-7-ONA 2,4,8-TRISUSTITUIDOS COMO INHIBIDORES DE LA QUINASA CSBP/RK/p38 |
US20080096905A1 (en) * | 2005-03-25 | 2008-04-24 | Glaxo Group Limited | Process For Preparing Pyrido[2,3-D]Pyrimidin-7-One And 3,4-Dihydropyrimido{4,5-D}Pyrimidin-2(1H)-One Derivatives |
WO2008005457A2 (en) * | 2006-06-30 | 2008-01-10 | Sunesis Pharmaceuticals | Pyridinonyl pdk1 inhibitors |
TW200835497A (en) * | 2007-01-11 | 2008-09-01 | Astrazeneca Ab | Chemical compounds 636 |
SA08280783B1 (ar) * | 2007-01-11 | 2011-04-24 | استرازينيكا ايه بي | مشتقات بيريدوبيريميدين كمثبطات pde4 |
WO2008084236A1 (en) * | 2007-01-11 | 2008-07-17 | Astrazeneca Ab | Chemical compounds 635 : pyridopyrimidinediones as pde4 inhibitors |
FR2925904B1 (fr) * | 2008-01-02 | 2010-01-01 | Sanofi Aventis | DERIVES DE N-HETEROCYCLIQUE-6-HETEROCYCLIQUE-IMIDAZO°1,2-a! PYRIDINE-2-CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE |
DK2297106T3 (da) * | 2008-05-27 | 2014-10-06 | Astrazeneca Ab | Phenoxypyridinylamidderivater og deres anvendelse til behandling af pde4-medierede sygdomstilstande |
EP2348860B1 (en) | 2008-10-31 | 2015-05-27 | Genentech, Inc. | Pyrazolopyrimidine jak inhibitor compounds and methods |
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JO2985B1 (ar) * | 2006-12-20 | 2016-09-05 | Takeda Pharmaceuticals Co | مثبطات كينازmapk/erk |
TW200835497A (en) * | 2007-01-11 | 2008-09-01 | Astrazeneca Ab | Chemical compounds 636 |
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- 2007-03-09 TW TW096108179A patent/TW200800997A/zh unknown
- 2007-03-20 EP EP07747954A patent/EP1999130A4/en not_active Withdrawn
- 2007-03-20 US US12/293,480 patent/US20090233907A1/en not_active Abandoned
- 2007-03-20 WO PCT/SE2007/000269 patent/WO2007108750A1/en active Application Filing
- 2007-03-20 JP JP2009501379A patent/JP2009530372A/ja active Pending
- 2007-03-21 AR ARP070101162A patent/AR060046A1/es unknown
- 2007-03-21 UY UY30228A patent/UY30228A1/es not_active Application Discontinuation
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AR060046A1 (es) | 2008-05-21 |
EP1999130A1 (en) | 2008-12-10 |
TW200800997A (en) | 2008-01-01 |
US20090233907A1 (en) | 2009-09-17 |
EP1999130A4 (en) | 2009-11-18 |
WO2007108750A1 (en) | 2007-09-27 |
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