UY29211A1 - Azabenzoxazoles para el tratamiento de los trastornos del snc - Google Patents

Azabenzoxazoles para el tratamiento de los trastornos del snc

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Publication number
UY29211A1
UY29211A1 UY29211A UY29211A UY29211A1 UY 29211 A1 UY29211 A1 UY 29211A1 UY 29211 A UY29211 A UY 29211A UY 29211 A UY29211 A UY 29211A UY 29211 A1 UY29211 A1 UY 29211A1
Authority
UY
Uruguay
Prior art keywords
formula
azabenzoxazoles
treatment
nicotinic receptor
cns disorders
Prior art date
Application number
UY29211A
Other languages
English (en)
Inventor
Bruce Nelsen Rogers
Allen Jacob Duplantier
Christopher John O Donnell
Lei Zhang
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35588927&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY29211(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of UY29211A1 publication Critical patent/UY29211A1/es

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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Abstract

La presente invención se refiere a agonistas del receptor nicotínico a(alfa)7 de fórmula I como se describen en el presente documento y a un procedimiento para tratar trastornos del Sistema Nervioso Central (SNC) y otros trastornos en un mamífero, incluyendo un humano, administrando al mamífero un agonista del receptor nicotínico a(alfa)7 de fórmula I como se muestra en el presente documento. Se refiere también a composiciones farmacéuticas que contienen un vehículo farmacéuticamente aceptable y un agonista del receptor nicotínico a(alfa)7 penetrante del SNC de fórmula I.
UY29211A 2004-11-15 2005-11-14 Azabenzoxazoles para el tratamiento de los trastornos del snc UY29211A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US65146304P 2004-11-15 2004-11-15

Publications (1)

Publication Number Publication Date
UY29211A1 true UY29211A1 (es) 2006-06-30

Family

ID=35588927

Family Applications (1)

Application Number Title Priority Date Filing Date
UY29211A UY29211A1 (es) 2004-11-15 2005-11-14 Azabenzoxazoles para el tratamiento de los trastornos del snc

Country Status (13)

Country Link
US (1) US20060166974A1 (es)
EP (1) EP1814887A1 (es)
JP (1) JP2008519820A (es)
AR (1) AR052236A1 (es)
CA (1) CA2587826A1 (es)
GT (1) GT200500333A (es)
NL (1) NL1030417C2 (es)
PA (1) PA8653001A1 (es)
PE (1) PE20061053A1 (es)
SV (1) SV2006002304A (es)
TW (1) TW200628476A (es)
UY (1) UY29211A1 (es)
WO (1) WO2006051407A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3250B1 (ar) 2009-09-22 2018-09-16 Novartis Ag إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7
JP6440625B2 (ja) 2012-11-14 2018-12-19 ザ・ジョンズ・ホプキンス・ユニバーシティー 精神分裂病を処置するための方法および組成物
CN107188900B (zh) * 2017-05-27 2019-09-06 北京师范大学 α7烟碱型乙酰胆碱受体的配体化合物及其应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2809730B1 (fr) * 2000-05-31 2002-07-19 Sanofi Synthelabo Derives de 1,4-diazabicyclo[3.2.2] nonanebenzoxazole, -benzothiazole et -benzimidazole, leur preparation et leur application therapeutique
US20020086871A1 (en) * 2000-12-29 2002-07-04 O'neill Brian Thomas Pharmaceutical composition for the treatment of CNS and other disorders
FR2832714B1 (fr) * 2001-11-23 2004-07-16 Sanofi Synthelabo Derives de 4-(oxazolopyridin-2-yl)-1,4-diazabicyclo[3.2.2] nonane, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
JP2008519820A (ja) 2008-06-12
TW200628476A (en) 2006-08-16
CA2587826A1 (en) 2006-05-18
US20060166974A1 (en) 2006-07-27
GT200500333A (es) 2006-06-13
SV2006002304A (es) 2006-09-14
NL1030417C2 (nl) 2006-11-23
PA8653001A1 (es) 2006-09-22
PE20061053A1 (es) 2006-10-20
EP1814887A1 (en) 2007-08-08
WO2006051407A1 (en) 2006-05-18
AR052236A1 (es) 2007-03-07
NL1030417A1 (nl) 2006-05-16

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