GT200500333A - Azabenzoxazoles para el tratamiento de los trastornos del snc - Google Patents

Azabenzoxazoles para el tratamiento de los trastornos del snc

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Publication number
GT200500333A
GT200500333A GT200500333A GT200500333A GT200500333A GT 200500333 A GT200500333 A GT 200500333A GT 200500333 A GT200500333 A GT 200500333A GT 200500333 A GT200500333 A GT 200500333A GT 200500333 A GT200500333 A GT 200500333A
Authority
GT
Guatemala
Prior art keywords
azabenzoxazoles
treatment
disorders
cns disorders
alfa7
Prior art date
Application number
GT200500333A
Other languages
English (en)
Inventor
Bruce Nelsen Rogers
Allen Jacob Duplantier
Christopher John O'donnell
Lei Zhang
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Application filed filed Critical
Publication of GT200500333A publication Critical patent/GT200500333A/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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    • A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
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  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Biomedical Technology (AREA)
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  • Pulmonology (AREA)
  • Virology (AREA)
  • Rheumatology (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Psychiatry (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
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  • Tropical Medicine & Parasitology (AREA)
  • Ophthalmology & Optometry (AREA)
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  • Child & Adolescent Psychology (AREA)
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Abstract

LA PRESENTE INVENCIÓN SE REFIERE A AGONISTAS DEL RECEPTOR NICOTÍNICO ALFA7 DE FÓRMULA I, Y A UN PROCEDIMIENTO PARA TRATAR TRASTORNOS DEL SISTEMA NERVIOSO CENTRAL (SNC) Y OTROS TRASTORNOS EN UN MAMIFERO, INCLUYENDO UN HUMANO, ADMINISTRANDO AL MAMIFERO UN AGONISTA DEL RECEPTOR NICOTINICO ALFA7 DE FORMULA I. SE REFIERE TAMBIÉN A COMPOSICIONES FARMACÉUTICAS QUE CONTIENEN UN VEHICULO FARMACÉUTICO ACEPTABLE Y UN AGONISTA DEL RECEPTOR NICOTÍNICO ALFA7 PENETRANTE AL SNC DE FÓRMULA I
GT200500333A 2004-11-15 2005-11-15 Azabenzoxazoles para el tratamiento de los trastornos del snc GT200500333A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US65146304P 2004-11-15 2004-11-15

Publications (1)

Publication Number Publication Date
GT200500333A true GT200500333A (es) 2006-06-13

Family

ID=35588927

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200500333A GT200500333A (es) 2004-11-15 2005-11-15 Azabenzoxazoles para el tratamiento de los trastornos del snc

Country Status (13)

Country Link
US (1) US20060166974A1 (es)
EP (1) EP1814887A1 (es)
JP (1) JP2008519820A (es)
AR (1) AR052236A1 (es)
CA (1) CA2587826A1 (es)
GT (1) GT200500333A (es)
NL (1) NL1030417C2 (es)
PA (1) PA8653001A1 (es)
PE (1) PE20061053A1 (es)
SV (1) SV2006002304A (es)
TW (1) TW200628476A (es)
UY (1) UY29211A1 (es)
WO (1) WO2006051407A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3250B1 (ar) 2009-09-22 2018-09-16 Novartis Ag إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7
US10154988B2 (en) 2012-11-14 2018-12-18 The Johns Hopkins University Methods and compositions for treating schizophrenia
CN107188900B (zh) * 2017-05-27 2019-09-06 北京师范大学 α7烟碱型乙酰胆碱受体的配体化合物及其应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2809730B1 (fr) * 2000-05-31 2002-07-19 Sanofi Synthelabo Derives de 1,4-diazabicyclo[3.2.2] nonanebenzoxazole, -benzothiazole et -benzimidazole, leur preparation et leur application therapeutique
US20020086871A1 (en) * 2000-12-29 2002-07-04 O'neill Brian Thomas Pharmaceutical composition for the treatment of CNS and other disorders
FR2832714B1 (fr) * 2001-11-23 2004-07-16 Sanofi Synthelabo Derives de 4-(oxazolopyridin-2-yl)-1,4-diazabicyclo[3.2.2] nonane, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
TW200628476A (en) 2006-08-16
WO2006051407A1 (en) 2006-05-18
CA2587826A1 (en) 2006-05-18
NL1030417A1 (nl) 2006-05-16
JP2008519820A (ja) 2008-06-12
NL1030417C2 (nl) 2006-11-23
SV2006002304A (es) 2006-09-14
EP1814887A1 (en) 2007-08-08
UY29211A1 (es) 2006-06-30
PA8653001A1 (es) 2006-09-22
US20060166974A1 (en) 2006-07-27
PE20061053A1 (es) 2006-10-20
AR052236A1 (es) 2007-03-07

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