UY28827A1 - Formas cristalinas de 5.11-dihidro-11-etil-5-metil-8-(2-((1-oxido-4-quinolinil)oxi)etil)-6h-dipirido(3,2-b:2`, 3`-ee) (1,4)diazepin-6-ona - Google Patents

Formas cristalinas de 5.11-dihidro-11-etil-5-metil-8-(2-((1-oxido-4-quinolinil)oxi)etil)-6h-dipirido(3,2-b:2`, 3`-ee) (1,4)diazepin-6-ona

Info

Publication number
UY28827A1
UY28827A1 UY28827A UY28827A UY28827A1 UY 28827 A1 UY28827 A1 UY 28827A1 UY 28827 A UY28827 A UY 28827A UY 28827 A UY28827 A UY 28827A UY 28827 A1 UY28827 A1 UY 28827A1
Authority
UY
Uruguay
Prior art keywords
etil
diazepin
dipirido
quinolinil
dihidro
Prior art date
Application number
UY28827A
Other languages
English (en)
Inventor
Busacca Carl Alan
Cerreta Michael Kenneth
Lorenz Jon Charles
Smoliga John Andrew
Richard J Varsolona
Vitous Jana
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34963561&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY28827(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of UY28827A1 publication Critical patent/UY28827A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Formas cristalinas dihidrato y anhidra de 5, 11-dihidro-11-etil-5-metil-8-(2-((1-óxido-4-quinolinil) oxi)etil)-6H- dipirido(3,2-b:2' , 3' -e) (1,4) diazepin-6-ona.
UY28827A 2004-04-02 2005-03-30 Formas cristalinas de 5.11-dihidro-11-etil-5-metil-8-(2-((1-oxido-4-quinolinil)oxi)etil)-6h-dipirido(3,2-b:2`, 3`-ee) (1,4)diazepin-6-ona UY28827A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US55935404P 2004-04-02 2004-04-02

Publications (1)

Publication Number Publication Date
UY28827A1 true UY28827A1 (es) 2005-10-31

Family

ID=34963561

Family Applications (1)

Application Number Title Priority Date Filing Date
UY28827A UY28827A1 (es) 2004-04-02 2005-03-30 Formas cristalinas de 5.11-dihidro-11-etil-5-metil-8-(2-((1-oxido-4-quinolinil)oxi)etil)-6h-dipirido(3,2-b:2`, 3`-ee) (1,4)diazepin-6-ona

Country Status (19)

Country Link
US (1) US7309700B2 (es)
EP (1) EP1740586A2 (es)
JP (1) JP2007530681A (es)
KR (1) KR20070014164A (es)
CN (1) CN1938306A (es)
AR (1) AR048360A1 (es)
AU (1) AU2005230922A1 (es)
BR (1) BRPI0509586A (es)
CA (1) CA2558817A1 (es)
EA (1) EA200601816A1 (es)
EC (1) ECSP066904A (es)
IL (1) IL178352A0 (es)
MX (1) MXPA06011324A (es)
NO (1) NO20064422L (es)
PE (1) PE20060164A1 (es)
TW (1) TW200602340A (es)
UY (1) UY28827A1 (es)
WO (1) WO2005097796A2 (es)
ZA (1) ZA200605930B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101541327A (zh) * 2006-01-31 2009-09-23 塔利昂制药公司 法呢基二苯并二氮杂酮的晶体形式
ES2773105T3 (es) * 2012-09-26 2020-07-09 Merck Sharp & Dohme Forma cristalina de un inhibidor de transcriptasa inversa

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI270547B (en) 2000-06-16 2007-01-11 Boehringer Ingelheim Ca Ltd Non-nucleoside reverse transcriptase inhibitors
US6759533B2 (en) 2002-06-28 2004-07-06 Boehringer Ingelheim Pharmaceuticals, Inc. Process and intermediates for making non-nucleoside HIV-1 reverse transcriptase inhibitors

Also Published As

Publication number Publication date
BRPI0509586A (pt) 2007-10-09
AU2005230922A1 (en) 2005-10-20
NO20064422L (no) 2006-09-29
ECSP066904A (es) 2006-12-20
EP1740586A2 (en) 2007-01-10
EA200601816A1 (ru) 2007-04-27
KR20070014164A (ko) 2007-01-31
US20050222134A1 (en) 2005-10-06
JP2007530681A (ja) 2007-11-01
CA2558817A1 (en) 2005-10-20
MXPA06011324A (es) 2007-03-21
PE20060164A1 (es) 2006-04-03
IL178352A0 (en) 2007-02-11
WO2005097796A2 (en) 2005-10-20
WO2005097796A3 (en) 2006-01-05
AR048360A1 (es) 2006-04-19
CN1938306A (zh) 2007-03-28
TW200602340A (en) 2006-01-16
US7309700B2 (en) 2007-12-18
ZA200605930B (en) 2007-12-27

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Legal Events

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Effective date: 20160509