EA200601816A1 - КРИСТАЛЛИЧЕСКИЕ ФОРМЫ 5,11-ДИГИДРО-11-ЭТИЛ-5-МЕТИЛ-8-{2-{(1-ОКСИДО-4-ХИНОЛИНИЛ)ОКСИ}ЭТИЛ}-6Н-ДИПИРИДО[3,2-b:2',3'-e][1,4]ДИАЗЕПИН-6-ОНА - Google Patents
КРИСТАЛЛИЧЕСКИЕ ФОРМЫ 5,11-ДИГИДРО-11-ЭТИЛ-5-МЕТИЛ-8-{2-{(1-ОКСИДО-4-ХИНОЛИНИЛ)ОКСИ}ЭТИЛ}-6Н-ДИПИРИДО[3,2-b:2',3'-e][1,4]ДИАЗЕПИН-6-ОНАInfo
- Publication number
- EA200601816A1 EA200601816A1 EA200601816A EA200601816A EA200601816A1 EA 200601816 A1 EA200601816 A1 EA 200601816A1 EA 200601816 A EA200601816 A EA 200601816A EA 200601816 A EA200601816 A EA 200601816A EA 200601816 A1 EA200601816 A1 EA 200601816A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- ethyl
- dipyrido
- diazepin
- dihydro
- oxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Virology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- AIDS & HIV (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
В заявке описаны дигидратная и безводная кристаллические формы 5,11-дигидро-11-этил-5-метил-8-{2-{(1-оксидо-4-хинолинил)окси}этил}-6Н-дипиридо[3,2-b:2',3'-е][1,4]диазепин-6-она.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US55935404P | 2004-04-02 | 2004-04-02 | |
PCT/US2005/009655 WO2005097796A2 (en) | 2004-04-02 | 2005-03-23 | Crystalline forms of 5,11-dihydro-11-ethyl-5-methyl-8-{2-{(1-oxido-4-quinolinyl)oxy}ethyl}-6h-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6-one |
Publications (1)
Publication Number | Publication Date |
---|---|
EA200601816A1 true EA200601816A1 (ru) | 2007-04-27 |
Family
ID=34963561
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200601816A EA200601816A1 (ru) | 2004-04-02 | 2005-03-23 | КРИСТАЛЛИЧЕСКИЕ ФОРМЫ 5,11-ДИГИДРО-11-ЭТИЛ-5-МЕТИЛ-8-{2-{(1-ОКСИДО-4-ХИНОЛИНИЛ)ОКСИ}ЭТИЛ}-6Н-ДИПИРИДО[3,2-b:2',3'-e][1,4]ДИАЗЕПИН-6-ОНА |
Country Status (19)
Country | Link |
---|---|
US (1) | US7309700B2 (ru) |
EP (1) | EP1740586A2 (ru) |
JP (1) | JP2007530681A (ru) |
KR (1) | KR20070014164A (ru) |
CN (1) | CN1938306A (ru) |
AR (1) | AR048360A1 (ru) |
AU (1) | AU2005230922A1 (ru) |
BR (1) | BRPI0509586A (ru) |
CA (1) | CA2558817A1 (ru) |
EA (1) | EA200601816A1 (ru) |
EC (1) | ECSP066904A (ru) |
IL (1) | IL178352A0 (ru) |
MX (1) | MXPA06011324A (ru) |
NO (1) | NO20064422L (ru) |
PE (1) | PE20060164A1 (ru) |
TW (1) | TW200602340A (ru) |
UY (1) | UY28827A1 (ru) |
WO (1) | WO2005097796A2 (ru) |
ZA (1) | ZA200605930B (ru) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2009527466A (ja) * | 2006-01-31 | 2009-07-30 | タリオン ファーマシューティカルズ インク. | ファルネシルジベンゾジアゼピノンの結晶形 |
EP2900240B1 (en) | 2012-09-26 | 2020-01-08 | Merck Sharp & Dohme Corp. | Crystalline form of a reverse transcriptase inhibitor |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI270547B (en) * | 2000-06-16 | 2007-01-11 | Boehringer Ingelheim Ca Ltd | Non-nucleoside reverse transcriptase inhibitors |
US6759533B2 (en) | 2002-06-28 | 2004-07-06 | Boehringer Ingelheim Pharmaceuticals, Inc. | Process and intermediates for making non-nucleoside HIV-1 reverse transcriptase inhibitors |
-
2005
- 2005-03-18 US US11/083,401 patent/US7309700B2/en active Active
- 2005-03-23 BR BRPI0509586-7A patent/BRPI0509586A/pt not_active Application Discontinuation
- 2005-03-23 MX MXPA06011324A patent/MXPA06011324A/es unknown
- 2005-03-23 KR KR1020067023046A patent/KR20070014164A/ko not_active Application Discontinuation
- 2005-03-23 AU AU2005230922A patent/AU2005230922A1/en not_active Abandoned
- 2005-03-23 CA CA002558817A patent/CA2558817A1/en not_active Abandoned
- 2005-03-23 EA EA200601816A patent/EA200601816A1/ru unknown
- 2005-03-23 EP EP05729416A patent/EP1740586A2/en not_active Withdrawn
- 2005-03-23 JP JP2007506248A patent/JP2007530681A/ja active Pending
- 2005-03-23 CN CNA2005800104438A patent/CN1938306A/zh active Pending
- 2005-03-23 WO PCT/US2005/009655 patent/WO2005097796A2/en active Application Filing
- 2005-03-30 UY UY28827A patent/UY28827A1/es not_active Application Discontinuation
- 2005-03-31 PE PE2005000373A patent/PE20060164A1/es not_active Application Discontinuation
- 2005-04-01 TW TW094110415A patent/TW200602340A/zh unknown
- 2005-04-01 AR ARP050101292A patent/AR048360A1/es unknown
-
2006
- 2006-07-18 ZA ZA200605930A patent/ZA200605930B/xx unknown
- 2006-09-28 IL IL178352A patent/IL178352A0/en unknown
- 2006-09-29 NO NO20064422A patent/NO20064422L/no not_active Application Discontinuation
- 2006-10-02 EC EC2006006904A patent/ECSP066904A/es unknown
Also Published As
Publication number | Publication date |
---|---|
JP2007530681A (ja) | 2007-11-01 |
US20050222134A1 (en) | 2005-10-06 |
WO2005097796A3 (en) | 2006-01-05 |
US7309700B2 (en) | 2007-12-18 |
WO2005097796A2 (en) | 2005-10-20 |
PE20060164A1 (es) | 2006-04-03 |
IL178352A0 (en) | 2007-02-11 |
ZA200605930B (en) | 2007-12-27 |
CN1938306A (zh) | 2007-03-28 |
MXPA06011324A (es) | 2007-03-21 |
EP1740586A2 (en) | 2007-01-10 |
ECSP066904A (es) | 2006-12-20 |
NO20064422L (no) | 2006-09-29 |
TW200602340A (en) | 2006-01-16 |
KR20070014164A (ko) | 2007-01-31 |
AR048360A1 (es) | 2006-04-19 |
UY28827A1 (es) | 2005-10-31 |
AU2005230922A1 (en) | 2005-10-20 |
BRPI0509586A (pt) | 2007-10-09 |
CA2558817A1 (en) | 2005-10-20 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA200801663A1 (ru) | КРИСТАЛЛИЧЕСКАЯ ФОРМА 1'-(1-МЕТИЛЭТИЛ)-4'-[(2-ФТОР-4-МЕТОКСИФЕНИЛ)МЕТИЛ]-5'-МЕТИЛ-1H-ПИРАЗОЛ-3'-O-β-D-ГЛЮКОПИРАНОЗИДА, СПОСОБ ЕГО ПОЛУЧЕНИЯ И ЕГО ПРИМЕНЕНИЕ ДЛЯ ПРИГОТОВЛЕНИЯ ЛЕКАРСТВЕННЫХ СРЕДСТВ | |
EA200601747A1 (ru) | Три(цикло)замещённые амидные соединения | |
EA200802213A1 (ru) | Способы лечения заболеваний крови | |
NO20070782L (no) | Tetrapeptidanaloger. | |
IS7215A (is) | Aðferðir til að meðhöndla nýæðarsjúkdóma í augum | |
WO2007061737A3 (en) | FUSED BICYCLIC mTOR INHIBITORS | |
DK1633726T3 (da) | Pyrimidinderivater, der er egnede til behandling af CRTH2-formidlede sygdomme | |
ATE516291T1 (de) | Thenopyrimidin-verbindungen mit fungizider aktivität | |
DK1781296T3 (da) | Quinazolinderivater og deres anvendelse ved behandlingen af thrombocytæmi | |
DK1411926T3 (da) | Integrininhibitorer til behandling af öjensygdomme | |
NO20045554L (no) | Fremgangsmate for behandling av diabetes | |
AT500499A3 (de) | Mittelpunktbestimmung von justiermarken | |
DK1482936T3 (da) | Öjenpræparat omfattende ascomycin | |
DK2185561T3 (da) | Derivater af 1,2,3,4-tetrahydropyrrolo(1,2-a)pyrazin-6-carboxamid og 2,3,4,5-tetrahydroprrolo(1,2-a)-diazepin-7-carboxamid, fremstilling deraf og terapeutisk anvendelse deraf | |
WO2004019879A3 (en) | Motilide compounds | |
GB0526486D0 (en) | Stockings of no wearing mark | |
CY2011018I1 (el) | Νεα κρυσταλλικη μορφη toy 8-kyan-1-kykλoπpoπyλ-7-(1s,6s-2,8-διαζαδικυκλο[4.3.0]εννεαν-8-υλ)-6-φθορο-1,4-διυδρο-4-οξο-3-κινολινο-καρβοξυλικου οξεος | |
MY140538A (en) | Substituted n-acyl-2-aminothiazoles | |
ZA200900165B (en) | 4-amino-3-arylamino-6-arylpyrazolo[3,4-D]pyrimidine derivatives, methods for their preparation and their use as antiviral agents | |
EA200601816A1 (ru) | КРИСТАЛЛИЧЕСКИЕ ФОРМЫ 5,11-ДИГИДРО-11-ЭТИЛ-5-МЕТИЛ-8-{2-{(1-ОКСИДО-4-ХИНОЛИНИЛ)ОКСИ}ЭТИЛ}-6Н-ДИПИРИДО[3,2-b:2',3'-e][1,4]ДИАЗЕПИН-6-ОНА | |
EA200601366A1 (ru) | Кристаллическая форма мононатрия ризедроната | |
DK1188815T3 (da) | Transparent, elastisk og fritstående forbindelse til fremstillingen af lys og fritstående lys opnået med denne forbindelse | |
DE60200268D1 (de) | Einkristallzüchtungsverfahren | |
DE60121542D1 (de) | Zweiachsiger Kreisel mit offener Regelschleife | |
DE602004020337D1 (de) | Anticholinergika enthaltende Arzneimittel zur Behandlung von Krankheiten der ableitenden Harnwege |