UY27290A1 - NEW MODULATORS OF AMPA POSITIVE ALOSTERIC RECEPTORS (PAARM), PROCEDURES FOR THEIR PREPARATION AND EMPLOYMENT AS MEDICATIONS - Google Patents

NEW MODULATORS OF AMPA POSITIVE ALOSTERIC RECEPTORS (PAARM), PROCEDURES FOR THEIR PREPARATION AND EMPLOYMENT AS MEDICATIONS

Info

Publication number
UY27290A1
UY27290A1 UY27290A UY27290A UY27290A1 UY 27290 A1 UY27290 A1 UY 27290A1 UY 27290 A UY27290 A UY 27290A UY 27290 A UY27290 A UY 27290A UY 27290 A1 UY27290 A1 UY 27290A1
Authority
UY
Uruguay
Prior art keywords
paarm
medications
employment
receptors
procedures
Prior art date
Application number
UY27290A
Other languages
Spanish (es)
Inventor
Dr A Ceci
Dr K Klinder
Dr T Weiser
Dr K Winter
Original Assignee
Boehringer Ingelheim Pharma
Co Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma, Co Kg filed Critical Boehringer Ingelheim Pharma
Publication of UY27290A1 publication Critical patent/UY27290A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Abstract

La presente invención se refiere a nuevos moduladores de receptores AMPA alostéricos de la fórmula (I), en donde R1, R2, R3, R4 y R5 pueden tener los significados indicados en la memoria descriptiva y en las reivindicaciones, a procedimientos como medicamentosThe present invention relates to new allosteric AMPA receptor modulators of the formula (I), wherein R1, R2, R3, R4 and R5 can have the meanings indicated in the specification and in the claims, to methods such as medicaments

UY27290A 2001-05-17 2002-05-15 NEW MODULATORS OF AMPA POSITIVE ALOSTERIC RECEPTORS (PAARM), PROCEDURES FOR THEIR PREPARATION AND EMPLOYMENT AS MEDICATIONS UY27290A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10123952A DE10123952A1 (en) 2001-05-17 2001-05-17 New naphtho-1,2-thiazine compounds, useful as neuroprotectants for treating e.g. epilepsy or Alzheimer's disease, are allosteric modulators of AMPA receptors

Publications (1)

Publication Number Publication Date
UY27290A1 true UY27290A1 (en) 2002-12-31

Family

ID=7685080

Family Applications (1)

Application Number Title Priority Date Filing Date
UY27290A UY27290A1 (en) 2001-05-17 2002-05-15 NEW MODULATORS OF AMPA POSITIVE ALOSTERIC RECEPTORS (PAARM), PROCEDURES FOR THEIR PREPARATION AND EMPLOYMENT AS MEDICATIONS

Country Status (26)

Country Link
EP (1) EP1404340A1 (en)
JP (1) JP2004529980A (en)
KR (1) KR20040007572A (en)
CN (1) CN1533278A (en)
AR (1) AR036332A1 (en)
BG (1) BG108324A (en)
BR (1) BR0209796A (en)
CA (1) CA2449189A1 (en)
CO (1) CO5550460A2 (en)
CZ (1) CZ20033112A3 (en)
DE (1) DE10123952A1 (en)
EA (1) EA006608B1 (en)
EC (1) ECSP034852A (en)
EE (1) EE200300566A (en)
HR (1) HRP20030933A2 (en)
HU (1) HUP0401273A3 (en)
IL (1) IL158642A0 (en)
MX (1) MXPA03010373A (en)
NO (1) NO20035088D0 (en)
NZ (1) NZ530154A (en)
PL (1) PL364053A1 (en)
SK (1) SK14222003A3 (en)
UY (1) UY27290A1 (en)
WO (1) WO2002100411A1 (en)
YU (1) YU90403A (en)
ZA (1) ZA200308466B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8039468B2 (en) * 2006-08-31 2011-10-18 The Governors Of The University Of Alberta Method of inhibition of respiratory depression using positive allosteric AMPA receptor modulators
CN111518058B (en) * 2020-05-29 2021-03-09 四川大学华西医院 Oxathiazine compound and application thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1998012185A1 (en) * 1996-09-17 1998-03-26 The Regents Of The University Of California Benzothiadiazide derivatives and their use as allosteric up-modulators of the ampa receptor
AU4711899A (en) * 1998-06-25 2000-01-10 Merck & Co., Inc. Naphtho(1,8-de)thiasin-2-yl methyl carbapenem antibacterials
DE10004572A1 (en) * 2000-02-02 2001-08-09 Boehringer Ingelheim Pharma New positive allosteric AMPA receptor modulators (PAARM), processes for their production and their use as medicines

Also Published As

Publication number Publication date
EA200301167A1 (en) 2004-06-24
NO20035088L (en) 2003-11-14
WO2002100411A1 (en) 2002-12-19
EE200300566A (en) 2004-02-16
EP1404340A1 (en) 2004-04-07
SK14222003A3 (en) 2004-05-04
PL364053A1 (en) 2004-12-13
KR20040007572A (en) 2004-01-24
IL158642A0 (en) 2004-05-12
NZ530154A (en) 2005-09-30
CZ20033112A3 (en) 2004-03-17
DE10123952A1 (en) 2002-11-21
BG108324A (en) 2004-12-30
NO20035088D0 (en) 2003-11-14
HUP0401273A3 (en) 2006-11-28
EA006608B1 (en) 2006-02-24
YU90403A (en) 2006-05-25
CN1533278A (en) 2004-09-29
HRP20030933A2 (en) 2004-04-30
ZA200308466B (en) 2004-05-24
HUP0401273A2 (en) 2004-10-28
ECSP034852A (en) 2003-12-24
MXPA03010373A (en) 2004-03-16
BR0209796A (en) 2004-06-01
AR036332A1 (en) 2004-09-01
CA2449189A1 (en) 2002-12-19
CO5550460A2 (en) 2005-08-31
JP2004529980A (en) 2004-09-30

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20141125