UA74767C2 - Method and composition for oral use of taxanes in patients - Google Patents
Method and composition for oral use of taxanes in patients Download PDFInfo
- Publication number
- UA74767C2 UA74767C2 UA99116450A UA99116450A UA74767C2 UA 74767 C2 UA74767 C2 UA 74767C2 UA 99116450 A UA99116450 A UA 99116450A UA 99116450 A UA99116450 A UA 99116450A UA 74767 C2 UA74767 C2 UA 74767C2
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- UA
- Ukraine
- Prior art keywords
- paclitaxel
- taxane
- administration
- agents
- cyclosporin
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
- A61K38/13—Cyclosporins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Urology & Nephrology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Gastroenterology & Hepatology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US86351397A | 1997-05-27 | 1997-05-27 | |
| PCT/US1998/007776 WO1998053811A1 (en) | 1997-05-27 | 1998-04-22 | Method and compositions for administering taxanes orally to human patients |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA74767C2 true UA74767C2 (en) | 2006-02-15 |
Family
ID=25341241
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UA99116450A UA74767C2 (en) | 1997-05-27 | 1998-04-22 | Method and composition for oral use of taxanes in patients |
Country Status (23)
| Country | Link |
|---|---|
| EP (1) | EP0994706B1 (hu) |
| JP (1) | JP2002500667A (hu) |
| KR (1) | KR100615783B1 (hu) |
| CN (2) | CN1550231A (hu) |
| AR (1) | AR012731A1 (hu) |
| AT (1) | ATE308365T1 (hu) |
| AU (1) | AU7130098A (hu) |
| BR (1) | BR9809694A (hu) |
| CA (1) | CA2290446C (hu) |
| CZ (1) | CZ9904244A3 (hu) |
| DE (1) | DE69832173T2 (hu) |
| DK (1) | DK0994706T3 (hu) |
| ES (1) | ES2247690T3 (hu) |
| HK (1) | HK1026637A1 (hu) |
| HU (1) | HUP0003546A3 (hu) |
| IL (2) | IL132992A0 (hu) |
| NO (1) | NO995812L (hu) |
| PL (1) | PL337064A1 (hu) |
| RU (1) | RU2205005C2 (hu) |
| SK (1) | SK157599A3 (hu) |
| UA (1) | UA74767C2 (hu) |
| WO (1) | WO1998053811A1 (hu) |
| ZA (1) | ZA984268B (hu) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6964946B1 (en) * | 1995-10-26 | 2005-11-15 | Baker Norton Pharmaceuticals, Inc. | Oral pharmaceutical compositions containing taxanes and methods of treatment employing the same |
| ATE219363T1 (de) * | 1997-06-20 | 2002-07-15 | Baker Norton Pharma | Lösliche prodrugs von paclitaxel |
| GB9718903D0 (en) | 1997-09-05 | 1997-11-12 | Glaxo Group Ltd | Method,compositions and kits for increasing the oral bioavailability of pharmaceutical agents |
| EP1749540B1 (en) | 1999-05-17 | 2010-10-13 | Cancer Research Ventures Limited | Compositions for improving bioavailability of orally administered drugs |
| IL149360A0 (en) * | 1999-10-27 | 2002-11-10 | Baker Norton Pharma | Method and compositions for administering taxanes orally to human patients |
| KR20020013174A (ko) * | 2000-08-11 | 2002-02-20 | 민경윤 | 경구 흡수율이 낮은 약물의 흡수율을 증가시키기 위한경구용 조성물 |
| US7115565B2 (en) | 2001-01-18 | 2006-10-03 | Pharmacia & Upjohn Company | Chemotherapeutic microemulsion compositions of paclitaxel with improved oral bioavailability |
| NZ539046A (en) * | 2001-01-18 | 2006-11-30 | Pharmacia & Upjohn Co Llc | Chemotherapeutic self-emulsifying microemulsion compositions of paclitaxel with improved oral bioavailability |
| UY27185A1 (es) * | 2001-02-28 | 2002-09-30 | Bristol Myers Squibb Co | Dosificación metronómica de taxanos |
| SI1372636T1 (sl) * | 2001-02-28 | 2006-12-31 | Bristol Myers Squibb Co | Metronomsko odmerjanje taksanov za inhibiranje tumorske rasti |
| US7063977B2 (en) | 2001-08-21 | 2006-06-20 | Bristol-Myers Squibb Company | Enzymatic resolution of t-butyl taxane derivatives |
| GB0523659D0 (en) * | 2005-11-21 | 2005-12-28 | Novartis Ag | Organic compounds |
| CN102803234A (zh) * | 2009-06-02 | 2012-11-28 | 霓坎制药有限责任公司 | 用于治疗疾病的人甲酰基肽受体的拮抗作用 |
| EP4059497A1 (en) * | 2021-03-17 | 2022-09-21 | Dompé farmaceutici S.p.a. | C5ar1 inhibitors for treating hypersensitivity reactions to taxanes |
| BR112023018826A2 (pt) * | 2021-03-17 | 2024-03-12 | Dompe Farm Spa | Inibidores de c5ar1 para tratamento de reações de hipersensibilidade a taxanos |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US5411947A (en) * | 1989-06-28 | 1995-05-02 | Vestar, Inc. | Method of converting a drug to an orally available form by covalently bonding a lipid to the drug |
| EP0563134B1 (en) * | 1990-12-18 | 1996-06-19 | The Wellcome Foundation Limited | Agents for potentiating the effects of antitumor agents and combating multiple drug resistance |
| CZ283038B6 (cs) * | 1991-01-11 | 1997-12-17 | Laboratoires Glaxo Sa | Akridinové deriváty, způsob výroby a farmaceutické prostředky s jejich obsahem |
| US5567592A (en) * | 1994-02-02 | 1996-10-22 | Regents Of The University Of California | Screening method for the identification of bioenhancers through the inhibition of P-glycoprotein transport in the gut of a mammal |
| DK0773938T3 (da) * | 1994-07-26 | 1999-09-20 | Indena Spa | Semi-syntetiske taxaner med anti-tumoraktivitet |
| TW354293B (en) * | 1995-06-06 | 1999-03-11 | Bristol Myers Squibb Co | Prodrugs of paclitaxel derivatives |
| CA2224227A1 (en) * | 1995-06-07 | 1996-12-19 | Avmax, Inc. | Use of essential oils to increase bioavailability of oral pharmaceutical compounds |
| US6245805B1 (en) * | 1995-10-26 | 2001-06-12 | Baker Norton Pharmaceuticals, Inc. | Method, compositions and kits for increasing the oral bioavailability of pharmaceutical agents |
| EP0822815A4 (en) * | 1996-01-31 | 1998-04-01 | Bristol Myers Squibb Co | PROCESS FOR MAKING ORAL-LIKE TAXANES ACTIVE FROM THE PHARMACEUTICAL VIEW |
| US6025359A (en) * | 1996-06-17 | 2000-02-15 | Eli Lilly And Company | Drug resistance and multidrug resistance modulators |
| GB9718903D0 (en) * | 1997-09-05 | 1997-11-12 | Glaxo Group Ltd | Method,compositions and kits for increasing the oral bioavailability of pharmaceutical agents |
| CA2326485C (en) * | 1998-04-01 | 2008-12-09 | Rtp Pharma Inc. | Anticancer compositions |
-
1998
- 1998-04-22 BR BR9809694-0A patent/BR9809694A/pt not_active IP Right Cessation
- 1998-04-22 RU RU99128033/14A patent/RU2205005C2/ru not_active IP Right Cessation
- 1998-04-22 CN CNA2004100304785A patent/CN1550231A/zh active Pending
- 1998-04-22 PL PL98337064A patent/PL337064A1/xx unknown
- 1998-04-22 ES ES98918361T patent/ES2247690T3/es not_active Expired - Lifetime
- 1998-04-22 KR KR1019997011000A patent/KR100615783B1/ko not_active IP Right Cessation
- 1998-04-22 CZ CZ19994244A patent/CZ9904244A3/cs unknown
- 1998-04-22 AT AT98918361T patent/ATE308365T1/de not_active IP Right Cessation
- 1998-04-22 AU AU71300/98A patent/AU7130098A/en not_active Abandoned
- 1998-04-22 DK DK98918361T patent/DK0994706T3/da active
- 1998-04-22 DE DE69832173T patent/DE69832173T2/de not_active Expired - Fee Related
- 1998-04-22 JP JP50066399A patent/JP2002500667A/ja active Pending
- 1998-04-22 CN CN98806440A patent/CN1261275A/zh active Pending
- 1998-04-22 UA UA99116450A patent/UA74767C2/uk unknown
- 1998-04-22 SK SK1575-99A patent/SK157599A3/sk unknown
- 1998-04-22 WO PCT/US1998/007776 patent/WO1998053811A1/en active IP Right Grant
- 1998-04-22 CA CA002290446A patent/CA2290446C/en not_active Expired - Fee Related
- 1998-04-22 IL IL13299298A patent/IL132992A0/xx active IP Right Grant
- 1998-04-22 EP EP98918361A patent/EP0994706B1/en not_active Expired - Lifetime
- 1998-04-22 HU HU0003546A patent/HUP0003546A3/hu unknown
- 1998-05-20 ZA ZA984268A patent/ZA984268B/xx unknown
- 1998-05-21 AR ARP980102356A patent/AR012731A1/es unknown
-
1999
- 1999-11-17 IL IL132992A patent/IL132992A/en not_active IP Right Cessation
- 1999-11-26 NO NO995812A patent/NO995812L/no not_active Application Discontinuation
-
2000
- 2000-09-20 HK HK00105943A patent/HK1026637A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| IL132992A0 (en) | 2001-03-19 |
| CA2290446A1 (en) | 1998-12-03 |
| HK1026637A1 (en) | 2000-12-22 |
| CN1550231A (zh) | 2004-12-01 |
| DE69832173T2 (de) | 2006-08-03 |
| NO995812D0 (no) | 1999-11-26 |
| CN1261275A (zh) | 2000-07-26 |
| AR012731A1 (es) | 2000-11-08 |
| CA2290446C (en) | 2008-01-29 |
| CZ9904244A3 (cs) | 2001-10-17 |
| HUP0003546A2 (hu) | 2002-11-28 |
| DE69832173D1 (de) | 2005-12-08 |
| WO1998053811A1 (en) | 1998-12-03 |
| RU2205005C2 (ru) | 2003-05-27 |
| HUP0003546A3 (en) | 2002-12-28 |
| IL132992A (en) | 2006-08-20 |
| NO995812L (no) | 2000-01-25 |
| ZA984268B (en) | 1999-06-23 |
| KR20010013025A (ko) | 2001-02-26 |
| ATE308365T1 (de) | 2005-11-15 |
| BR9809694A (pt) | 2000-10-03 |
| EP0994706A1 (en) | 2000-04-26 |
| AU7130098A (en) | 1998-12-30 |
| SK157599A3 (en) | 2002-10-08 |
| PL337064A1 (en) | 2000-07-31 |
| ES2247690T3 (es) | 2006-03-01 |
| KR100615783B1 (ko) | 2006-08-25 |
| JP2002500667A (ja) | 2002-01-08 |
| DK0994706T3 (da) | 2006-03-06 |
| EP0994706B1 (en) | 2005-11-02 |
| EP0994706A4 (en) | 2001-05-16 |
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