UA107660C2 - Антагонисты арилсульфонамидов ccr3 - Google Patents

Антагонисты арилсульфонамидов ccr3

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Publication number
UA107660C2
UA107660C2 UAA201113726A UAA201113726A UA107660C2 UA 107660 C2 UA107660 C2 UA 107660C2 UA A201113726 A UAA201113726 A UA A201113726A UA A201113726 A UAA201113726 A UA A201113726A UA 107660 C2 UA107660 C2 UA 107660C2
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UA
Ukraine
Prior art keywords
ccr3
arylsulfonamides
antagonists
ameliorating
symptoms
Prior art date
Application number
UAA201113726A
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English (en)
Ukrainian (uk)
Inventor
Тай Вей Лай
Джаред Ендрю Форрестер
Original Assignee
Аксікін Фармасьютікалз, Інк.
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42301162&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA107660(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Аксікін Фармасьютікалз, Інк. filed Critical Аксікін Фармасьютікалз, Інк.
Publication of UA107660C2 publication Critical patent/UA107660C2/ru

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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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Abstract

Изобретение касается арилсульфонамидов, которые пригодны для модуляции активности CCR3, и их фармацевтических композиций. Также изобретение касается способов их применения для лечения, профилактики или облегчения одного или более симптомов CCR3-опосредованного нарушения, заболевания или состояния.
UAA201113726A 2009-04-22 2010-04-21 Антагонисты арилсульфонамидов ccr3 UA107660C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17178009P 2009-04-22 2009-04-22
PCT/US2010/031833 WO2010123960A2 (en) 2009-04-22 2010-04-21 Arylsulfonamide ccr3 antagonists

Publications (1)

Publication Number Publication Date
UA107660C2 true UA107660C2 (ru) 2015-02-10

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ID=42301162

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UAA201113726A UA107660C2 (ru) 2009-04-22 2010-04-21 Антагонисты арилсульфонамидов ccr3

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US (2) US8420639B2 (ru)
EP (2) EP2421838A2 (ru)
JP (1) JP2012524791A (ru)
KR (1) KR20120034627A (ru)
CN (1) CN102459210B (ru)
AR (1) AR076363A1 (ru)
AU (1) AU2010239341B2 (ru)
BR (1) BRPI1014668A2 (ru)
CA (1) CA2758729A1 (ru)
CL (1) CL2011002619A1 (ru)
CO (1) CO6470793A2 (ru)
CR (1) CR20110536A (ru)
DK (1) DK2502921T3 (ru)
EC (1) ECSP11011474A (ru)
ES (1) ES2543754T3 (ru)
HK (1) HK1176927A1 (ru)
HU (1) HUE025647T2 (ru)
IL (1) IL215843A0 (ru)
MX (1) MX2011011141A (ru)
MY (1) MY184048A (ru)
NI (1) NI201100185A (ru)
NZ (2) NZ595838A (ru)
PE (2) PE20150759A1 (ru)
RU (1) RU2539591C2 (ru)
SG (2) SG175277A1 (ru)
TW (1) TWI473793B (ru)
UA (1) UA107660C2 (ru)
WO (1) WO2010123960A2 (ru)

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Publication number Priority date Publication date Assignee Title
SG10201505313RA (en) 2009-04-22 2015-08-28 Axikin Pharmaceuticals Inc 2,5-Disubstituted Arylsulfonamide CCR3 Antagonists
CA2758985A1 (en) * 2009-04-22 2010-10-28 Axikin Pharmaceuticals, Inc. 2,5-disubstituted arylsulfonamide ccr3 antagonists
HUE025699T2 (en) * 2010-03-02 2016-04-28 Axikin Pharmaceuticals Inc Isotopically enriched arylsulfonamide derivatives as CCR3 antagonists
CA2814011A1 (en) * 2010-10-11 2012-04-19 Axikin Pharmaceuticals, Inc. Salts of arylsulfonamide ccr3 antagonists
KR20150053906A (ko) 2012-09-07 2015-05-19 액시킨 파마수티컬스 인코포레이티드 동위원소 농축 아릴설폰아미드 ccr3 길항제
GB2560713A (en) * 2017-03-20 2018-09-26 Eternygen Gmbh Inhibitor of citrate transporter

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