TW229208B - - Google Patents

Info

Publication number
TW229208B
TW229208B TW080107102A TW80107102A TW229208B TW 229208 B TW229208 B TW 229208B TW 080107102 A TW080107102 A TW 080107102A TW 80107102 A TW80107102 A TW 80107102A TW 229208 B TW229208 B TW 229208B
Authority
TW
Taiwan
Prior art keywords
compound
preparation
pharmaceutical compositions
compositions containing
relates
Prior art date
Application number
TW080107102A
Other languages
English (en)
Chinese (zh)
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24320279&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TW229208(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corp filed Critical Schering Corp
Application granted granted Critical
Publication of TW229208B publication Critical patent/TW229208B/zh

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J17/00Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0043Nose

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
TW080107102A 1990-09-10 1991-09-09 TW229208B (forum.php)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US58023990A 1990-09-10 1990-09-10

Publications (1)

Publication Number Publication Date
TW229208B true TW229208B (forum.php) 1994-09-01

Family

ID=24320279

Family Applications (2)

Application Number Title Priority Date Filing Date
TW080107102A TW229208B (forum.php) 1990-09-10 1991-09-09
TW083106101A TW272195B (forum.php) 1990-09-10 1991-09-09

Family Applications After (1)

Application Number Title Priority Date Filing Date
TW083106101A TW272195B (forum.php) 1990-09-10 1991-09-09

Country Status (35)

Country Link
US (1) US6180781B1 (forum.php)
EP (1) EP0548114B1 (forum.php)
JP (1) JPH0725789B2 (forum.php)
KR (1) KR960013445B1 (forum.php)
CN (1) CN1030920C (forum.php)
AT (1) ATE113604T1 (forum.php)
AU (1) AU663471B2 (forum.php)
BG (1) BG60755B2 (forum.php)
CA (1) CA2091360C (forum.php)
CZ (1) CZ281318B6 (forum.php)
DE (2) DE69104991T2 (forum.php)
DK (1) DK0548114T5 (forum.php)
EE (1) EE02962B1 (forum.php)
ES (1) ES2065701T3 (forum.php)
FI (1) FI111078B (forum.php)
HK (1) HK185996A (forum.php)
HR (1) HRP920383B1 (forum.php)
HU (1) HU213401B (forum.php)
IE (1) IE67056B1 (forum.php)
IL (1) IL99437A (forum.php)
LU (1) LU90366I2 (forum.php)
MX (2) MX9203396A (forum.php)
MY (1) MY106644A (forum.php)
NL (1) NL980012I2 (forum.php)
NO (1) NO300548B1 (forum.php)
NZ (1) NZ239711A (forum.php)
OA (1) OA09772A (forum.php)
PH (1) PH30443A (forum.php)
PL (1) PL165803B1 (forum.php)
PT (1) PT98905B (forum.php)
SI (1) SI9111497A (forum.php)
TW (2) TW229208B (forum.php)
WO (1) WO1992004365A1 (forum.php)
YU (1) YU48666B (forum.php)
ZA (1) ZA917148B (forum.php)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CZ281318B6 (cs) * 1990-09-10 1996-08-14 Schering Corporation Monohydrát mometasonfuroátu, způsob přípravy této látky a přípravy lékových kompozic z ní
PE44995A1 (es) * 1994-01-27 1995-12-18 Schering Corp Furoato de mometasona para el tratamiento de las enfermedades pulmonares y de las vias respiratorias
US5837699A (en) 1994-01-27 1998-11-17 Schering Corporation Use of mometasone furoate for treating upper airway passage diseases
US5886200A (en) * 1996-07-01 1999-03-23 Schering Corporation Process for the preparation of 17-esters of 9 α, 21-dihalo-pregnane-11 β, 17 α-diol-20-ones
US5976573A (en) 1996-07-03 1999-11-02 Rorer Pharmaceutical Products Inc. Aqueous-based pharmaceutical composition
CN1059476C (zh) * 1996-08-21 2000-12-13 邓维鹏 金黄色铝合金硒盐电解着色方法
DE69804998T2 (de) * 1997-10-09 2002-12-12 Schering Corp., Kenilworth Mometasonfuroat-suspensionen zum zerstäuben
US6187765B1 (en) * 1997-10-09 2001-02-13 Schering Corporation Mometasone furoate suspensions for nebulization
MY133181A (en) * 1998-09-10 2007-10-31 Schering Corp Methods and compositions for treating sinusitis, otitis media and other related disorders using antihistamines
HUP0200871A3 (en) 1999-05-04 2004-04-28 Strakan Int Ltd Androgen glycosides and androgenic activity thereof
GB0207906D0 (en) * 2002-04-05 2002-05-15 3M Innovative Properties Co Formoterol and mometasone aerosol formulations
US9808471B2 (en) 2003-04-16 2017-11-07 Mylan Specialty Lp Nasal pharmaceutical formulations and methods of using the same
US8912174B2 (en) 2003-04-16 2014-12-16 Mylan Pharmaceuticals Inc. Formulations and methods for treating rhinosinusitis
US7811606B2 (en) 2003-04-16 2010-10-12 Dey, L.P. Nasal pharmaceutical formulations and methods of using the same
NZ545748A (en) * 2003-08-29 2010-03-26 Ranbaxy Lab Ltd Isoxazoline derivatives as inhibitors of phosphodiesterase type-IV
EP1694655A2 (en) * 2003-11-26 2006-08-30 Ranbaxy Laboratories Limited Phosphodiesterase inhibitors
US7491725B2 (en) 2004-02-06 2009-02-17 Bristol-Myers Squibb Company Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
WO2007031838A1 (en) 2005-09-16 2007-03-22 Ranbaxy Laboratories Limited Substituted pyrazolo [3,4-b] pyridines as phosphodiesterase inhibitors
US20070099883A1 (en) * 2005-10-07 2007-05-03 Cheryl Lynn Calis Anhydrous mometasone furoate formulation
EP1948167A1 (en) * 2005-10-19 2008-07-30 Ranbaxy Laboratories, Ltd. Compositions of phosphodiesterase type iv inhibitors
EP1948164A1 (en) 2005-10-19 2008-07-30 Ranbaxy Laboratories, Ltd. Pharmaceutical compositions of muscarinic receptor antagonists
CN100436473C (zh) * 2005-12-09 2008-11-26 天津药业集团有限公司 糠酸莫美他松中间体21-酯及制法
CN100389121C (zh) * 2005-12-09 2008-05-21 天津药业集团有限公司 糠酸莫美他松中间体21-羟的制备方法
DE102006034883A1 (de) * 2006-07-25 2008-01-31 Hermal Kurt Herrmann Gmbh & Co. Ohg Pharmazeutische Zusammensetzung enthaltend Mometasonfuroat
US20110021473A1 (en) * 2006-09-22 2011-01-27 Ranbaxy Laboratories Limited Inhibitors of phosphodiesterase type-iv
US20100029728A1 (en) * 2006-09-22 2010-02-04 Ranbaxy Laboratories Limited Phosphodiesterase inhibitors
US20080207659A1 (en) * 2007-02-15 2008-08-28 Asit Kumar Chakraborti Inhibitors of phosphodiesterase type 4
ATE545417T1 (de) * 2007-03-14 2012-03-15 Ranbaxy Lab Ltd Pyrazoloä3,4-büpyridin-derivate als phosphodiesterasehemmer
US20110130403A1 (en) * 2007-03-14 2011-06-02 Ranbaxy Laboratories Limited Pyrazolo [3, 4-b] pyridine derivatives as phosphodiesterase inhibitors
EP2111861A1 (en) 2008-04-21 2009-10-28 Ranbaxy Laboratories Limited Compositions of phosphodiesterase type IV inhibitors
PT3111927T (pt) 2009-05-29 2020-03-03 Pearl Therapeutics Inc Composições para administração respiratória de agentes ativos e métodos e sistemas associados
US8815258B2 (en) * 2009-05-29 2014-08-26 Pearl Therapeutics, Inc. Compositions, methods and systems for respiratory delivery of two or more active agents
PT105058B (pt) 2010-04-21 2013-04-17 Hovione Farmaciencia S A Processo para processamento de partículas de ingredientes activos farmacêuticos
EP2968152B2 (en) 2013-03-15 2022-06-22 Pearl Therapeutics, Inc. Methods and systems for conditioning of particulate crystalline materials
CN107260671B (zh) * 2016-04-08 2021-03-26 天津金耀集团有限公司 一种糠酸莫米松混悬鼻喷剂组合物
CN107266518B (zh) * 2016-04-08 2021-03-30 天津金耀集团有限公司 一种糠酸莫米松晶型及其制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3260474D1 (en) * 1981-02-02 1984-09-06 Schering Corp Aromatic heterocyclic esters of steroids, their preparation and pharmaceutical compositions containing them
US4783444A (en) 1984-09-17 1988-11-08 Schering Corporation Antiglaucoma compositions and methods
US4808610A (en) * 1986-10-02 1989-02-28 Schering Corporation Mometasone furoate anti-inflammatory cream composition using hexylene glycol
US4775529A (en) * 1987-05-21 1988-10-04 Schering Corporation Steroid lotion
CZ281318B6 (cs) * 1990-09-10 1996-08-14 Schering Corporation Monohydrát mometasonfuroátu, způsob přípravy této látky a přípravy lékových kompozic z ní

Also Published As

Publication number Publication date
AU8497491A (en) 1992-03-30
NO930693D0 (no) 1993-02-26
PL165803B1 (pl) 1995-02-28
US6180781B1 (en) 2001-01-30
CA2091360C (en) 1997-04-08
DE19875032I2 (de) 2007-04-19
OA09772A (en) 1993-11-30
NO930693L (no) 1993-02-26
CZ281318B6 (cs) 1996-08-14
WO1992004365A1 (en) 1992-03-19
HK185996A (en) 1996-10-11
NZ239711A (en) 1992-09-25
DE69104991T2 (de) 1995-04-20
MX9203396A (es) 1992-07-31
EP0548114A1 (en) 1993-06-30
ZA917148B (en) 1992-08-26
HRP920383A2 (en) 1998-06-30
TW272195B (forum.php) 1996-03-11
IL99437A0 (en) 1992-08-18
EE02962B1 (et) 1997-02-17
JPH05506667A (ja) 1993-09-30
SI9111497A (sl) 1998-04-30
YU48666B (sh) 1999-06-15
HU9300685D0 (en) 1993-06-28
FI931031A0 (fi) 1993-03-09
NO300548B1 (no) 1997-06-16
PT98905B (pt) 1998-08-31
BG60755B2 (bg) 1996-02-29
IE67056B1 (en) 1996-02-21
HU213401B (en) 1997-06-30
IL99437A (en) 1995-05-29
FI931031L (fi) 1993-03-09
DK0548114T5 (da) 1995-01-30
IE913155A1 (en) 1992-03-11
CN1030920C (zh) 1996-02-07
AU663471B2 (en) 1995-10-12
HUT64361A (en) 1993-12-28
MX9100990A (es) 1992-05-04
DE69104991D1 (de) 1994-12-08
KR960013445B1 (ko) 1996-10-05
CN1059911A (zh) 1992-04-01
ATE113604T1 (de) 1994-11-15
JPH0725789B2 (ja) 1995-03-22
PH30443A (en) 1997-05-09
NL980012I1 (nl) 1998-05-06
MY106644A (en) 1995-07-31
NL980012I2 (nl) 2004-11-01
HRP920383B1 (en) 2000-04-30
CA2091360A1 (en) 1992-03-11
YU149791A (sh) 1994-01-20
LU90366I2 (fr) 1999-05-05
CZ38393A3 (en) 1994-01-19
PT98905A (pt) 1992-09-30
FI111078B (fi) 2003-05-30
ES2065701T3 (es) 1995-02-16
EP0548114B1 (en) 1994-11-02

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Legal Events

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