TW201518291A - 含聚乙二醇之組成物 - Google Patents

含聚乙二醇之組成物 Download PDF

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Publication number
TW201518291A
TW201518291A TW103132199A TW103132199A TW201518291A TW 201518291 A TW201518291 A TW 201518291A TW 103132199 A TW103132199 A TW 103132199A TW 103132199 A TW103132199 A TW 103132199A TW 201518291 A TW201518291 A TW 201518291A
Authority
TW
Taiwan
Prior art keywords
pharmaceutical composition
formula
polyethylene glycol
salt
acid
Prior art date
Application number
TW103132199A
Other languages
English (en)
Chinese (zh)
Inventor
村井健二
山田和人
Original Assignee
參天製藥股份有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 參天製藥股份有限公司 filed Critical 參天製藥股份有限公司
Publication of TW201518291A publication Critical patent/TW201518291A/zh

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Ophthalmology & Optometry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Dermatology (AREA)
TW103132199A 2013-09-20 2014-09-18 含聚乙二醇之組成物 TW201518291A (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2013195329 2013-09-20

Publications (1)

Publication Number Publication Date
TW201518291A true TW201518291A (zh) 2015-05-16

Family

ID=52688941

Family Applications (1)

Application Number Title Priority Date Filing Date
TW103132199A TW201518291A (zh) 2013-09-20 2014-09-18 含聚乙二醇之組成物

Country Status (17)

Country Link
US (1) US20160228420A1 (https=)
EP (1) EP3047850A4 (https=)
JP (2) JP5856264B2 (https=)
KR (1) KR20160060656A (https=)
CN (1) CN105555271A (https=)
AU (1) AU2014322111A1 (https=)
BR (1) BR112016006153A2 (https=)
CA (1) CA2924628A1 (https=)
EA (1) EA201690621A1 (https=)
HK (2) HK1221407A1 (https=)
IL (1) IL244648A0 (https=)
MX (1) MX2016003566A (https=)
MY (1) MY163236A (https=)
PH (1) PH12016500461A1 (https=)
SG (1) SG11201602020QA (https=)
TW (1) TW201518291A (https=)
WO (1) WO2015041294A1 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2979802C (en) * 2015-03-17 2023-06-27 Santen Pharmaceutical Co., Ltd. Pharmaceutical composition comprising polypeptide
TWI731853B (zh) * 2015-03-18 2021-07-01 日商參天製藥股份有限公司 徐放性醫藥組成物及其安定化方法
WO2016208742A1 (ja) * 2015-06-25 2016-12-29 参天製薬株式会社 注射剤
EP3318280A4 (en) * 2015-07-01 2018-08-22 Santen Pharmaceutical Co., Ltd Depot preparation containing citric acid ester
CN106902117A (zh) * 2015-12-23 2017-06-30 瑞阳(苏州)生物科技有限公司 一种预防或治疗脉络膜新生血管形成的药物
JP7018939B2 (ja) * 2016-09-26 2022-02-14 ルヤン (スーチョウ) バイオロジー サイエンス アンド テクノロジー カンパニー,リミテッド 眼疾患の治療のための組成物ならびに使用および調製方法

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA833692B (en) * 1982-05-28 1985-02-27 Beecham Group Plc Pharmaceutical formulations
JPS59101478A (ja) * 1982-11-29 1984-06-12 Sunstar Inc リグスチライドを安定に配合した水系組成物
JPH09110698A (ja) * 1995-10-19 1997-04-28 Taiho Yakuhin Kogyo Kk 経口用医薬組成物の製造法
ES2368153T3 (es) * 2004-02-17 2011-11-14 Santen Pharmaceutical Co., Ltd. Nuevo compuesto cíclico que presenta un grupo 4-piridilalquiltio que presenta amino (no) sustituido introducido en el mismo.
JP4626353B2 (ja) * 2004-02-17 2011-02-09 参天製薬株式会社 置換又は無置換アミノ基を導入した4−ピリジルアルキルチオ基を有する新規環式化合物
EP1717229B1 (en) * 2004-02-17 2011-06-15 Santen Pharmaceutical Co., Ltd. Novel cyclic compound having 4-pyridylalkylthio group having (un)substituted amino introduced therein
US20060153920A1 (en) * 2004-09-24 2006-07-13 Ketan Amin Lyophilized pharmaceutical compositions
JP4974903B2 (ja) 2005-02-09 2012-07-11 参天製薬株式会社 疾患または状態を処置するための液体処方物
JP2009521493A (ja) 2005-12-23 2009-06-04 アルコン,インコーポレイテッド 眼への受容体チロシンキナーゼ阻害(RTKi)化合物の送達のための医薬製剤
JP2010534201A (ja) 2007-07-20 2010-11-04 アルコン,インコーポレイテッド 受容体チロシンキナーゼ阻害(RTKi)化合物の目への送達のための医薬製剤
WO2009070687A1 (en) * 2007-11-26 2009-06-04 Merial Limited Solvent systems for pour-on formulations for combating parasites
MX2011008680A (es) 2009-03-03 2011-09-08 Alcon Res Ltd Composicion farmaceutica para el suministro de compuestos inhibidores de la tirosina cinasa receptora (rtki) para los ojos.
WO2011007870A1 (ja) * 2009-07-17 2011-01-20 参天製薬株式会社 2-[[[2-[(ヒドロキシアセチル)アミノ]-4-ピリジニル]メチル]チオ]-n-[4-(トリフルオロメトキシ)フェニル]-3-ピリジンカルボキサミドのベンゼンスルホン酸塩、その結晶、その結晶多形およびそれらの製造方法
PL3158991T3 (pl) * 2010-01-28 2021-09-27 Eagle Pharmaceuticals, Inc. Preparaty bendamustyny

Also Published As

Publication number Publication date
JP2015083565A (ja) 2015-04-30
HK1221407A1 (en) 2017-06-02
CN105555271A (zh) 2016-05-04
HK1220632A1 (zh) 2017-05-12
CA2924628A1 (en) 2015-03-26
US20160228420A1 (en) 2016-08-11
EA201690621A1 (ru) 2016-07-29
BR112016006153A2 (pt) 2017-08-01
IL244648A0 (en) 2016-04-21
KR20160060656A (ko) 2016-05-30
WO2015041294A1 (ja) 2015-03-26
EP3047850A4 (en) 2017-05-10
SG11201602020QA (en) 2016-04-28
MY163236A (en) 2017-08-30
AU2014322111A1 (en) 2016-04-07
MX2016003566A (es) 2016-06-02
EP3047850A1 (en) 2016-07-27
JP5856264B2 (ja) 2016-02-09
PH12016500461A1 (en) 2016-05-16
JP2016094442A (ja) 2016-05-26

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