TW201444821A - 經取代之哌啶化合物及其作為食慾素受體調節劑之用途 - Google Patents

經取代之哌啶化合物及其作為食慾素受體調節劑之用途 Download PDF

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TW201444821A
TW201444821A TW103108298A TW103108298A TW201444821A TW 201444821 A TW201444821 A TW 201444821A TW 103108298 A TW103108298 A TW 103108298A TW 103108298 A TW103108298 A TW 103108298A TW 201444821 A TW201444821 A TW 201444821A
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alkyl
compound
methyl
phenyl
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TW103108298A
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Chinese (zh)
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Heather R Coate
Curt A Dvorak
Cathy Preville
Brock T Shireman
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Janssen Pharmaceutica Nv
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07—ORGANIC CHEMISTRY
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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07—ORGANIC CHEMISTRY
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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • Chemical Kinetics & Catalysis (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • Neurology (AREA)
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  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Addiction (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Endocrinology (AREA)
  • Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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  • Child & Adolescent Psychology (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Otolaryngology (AREA)
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TW103108298A 2013-03-13 2014-03-11 經取代之哌啶化合物及其作為食慾素受體調節劑之用途 TW201444821A (zh)

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US201361780302P 2013-03-13 2013-03-13

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US (2) US9115117B2 (enExample)
EP (1) EP2970207B1 (enExample)
JP (1) JP6275814B2 (enExample)
CN (1) CN105228995B (enExample)
AR (1) AR095422A1 (enExample)
AU (2) AU2014248763B2 (enExample)
TW (1) TW201444821A (enExample)
UY (1) UY35410A (enExample)
WO (1) WO2014165065A1 (enExample)

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UY35410A (es) 2014-09-30
JP6275814B2 (ja) 2018-02-07
EP2970207B1 (en) 2018-05-16
CN105228995B (zh) 2018-12-25
CN105228995A (zh) 2016-01-06
WO2014165065A1 (en) 2014-10-09
AU2018229449A1 (en) 2018-10-04
US9611251B2 (en) 2017-04-04
EP2970207A1 (en) 2016-01-20
AR095422A1 (es) 2015-10-14
US20160046599A1 (en) 2016-02-18
JP2016512534A (ja) 2016-04-28
AU2014248763B2 (en) 2018-08-30
AU2014248763A1 (en) 2015-08-27
US9115117B2 (en) 2015-08-25

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