AU2014248763B2 - Substituted piperidine compounds and their use as orexin receptor modulators - Google Patents

Substituted piperidine compounds and their use as orexin receptor modulators Download PDF

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AU2014248763B2
AU2014248763B2 AU2014248763A AU2014248763A AU2014248763B2 AU 2014248763 B2 AU2014248763 B2 AU 2014248763B2 AU 2014248763 A AU2014248763 A AU 2014248763A AU 2014248763 A AU2014248763 A AU 2014248763A AU 2014248763 B2 AU2014248763 B2 AU 2014248763B2
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methanone
methyl
pyridin
trifluoromethyl
piperidin
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AU2014248763A1 (en
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Heather R. COATE
Curt A. Dvorak
Cathy PREVILLE
Brock T. Shireman
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Janssen Pharmaceutica NV
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Janssen Pharmaceutica NV
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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AU2014248763A 2013-03-13 2014-03-12 Substituted piperidine compounds and their use as orexin receptor modulators Active AU2014248763B2 (en)

Priority Applications (1)

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AU2018229449A AU2018229449A1 (en) 2013-03-13 2018-09-12 Substituted piperidine compounds and their use as orexin receptor modulators

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US201361780302P 2013-03-13 2013-03-13
US61/780,302 2013-03-13
PCT/US2014/024284 WO2014165065A1 (en) 2013-03-13 2014-03-12 Substituted piperidine compounds and their use as orexin receptor modulators

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AU2014248763B2 true AU2014248763B2 (en) 2018-08-30

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EP (1) EP2970207B1 (enExample)
JP (1) JP6275814B2 (enExample)
CN (1) CN105228995B (enExample)
AR (1) AR095422A1 (enExample)
AU (2) AU2014248763B2 (enExample)
TW (1) TW201444821A (enExample)
UY (1) UY35410A (enExample)
WO (1) WO2014165065A1 (enExample)

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US20090163485A1 (en) * 2007-12-21 2009-06-25 Henner Knust Heteroaryl derivatives as orexin receptor antagonists
WO2009133522A1 (en) * 2008-04-30 2009-11-05 Actelion Pharmaceuticals Ltd Piperidine and pyrrolidine compounds

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AU2014248763A1 (en) 2015-08-27
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US9115117B2 (en) 2015-08-25
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UY35410A (es) 2014-09-30

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