TW201326134A - 以被取代吡唑基甲醯胺及被以一含氮基團取代之含有一苯基基元之尿素衍生物做為類香草素受體之配位體 - Google Patents
以被取代吡唑基甲醯胺及被以一含氮基團取代之含有一苯基基元之尿素衍生物做為類香草素受體之配位體 Download PDFInfo
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- TW201326134A TW201326134A TW101141482A TW101141482A TW201326134A TW 201326134 A TW201326134 A TW 201326134A TW 101141482 A TW101141482 A TW 101141482A TW 101141482 A TW101141482 A TW 101141482A TW 201326134 A TW201326134 A TW 201326134A
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- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
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- Pain & Pain Management (AREA)
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- Rheumatology (AREA)
- Pulmonology (AREA)
- Hematology (AREA)
- Psychiatry (AREA)
- Virology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Psychology (AREA)
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- Dermatology (AREA)
- Endocrinology (AREA)
- Molecular Biology (AREA)
- Addiction (AREA)
- Communicable Diseases (AREA)
- Hospice & Palliative Care (AREA)
- Biotechnology (AREA)
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- Oncology (AREA)
- Emergency Medicine (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP11008913 | 2011-11-09 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW201326134A true TW201326134A (zh) | 2013-07-01 |
Family
ID=47143123
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW101141482A TW201326134A (zh) | 2011-11-09 | 2012-11-08 | 以被取代吡唑基甲醯胺及被以一含氮基團取代之含有一苯基基元之尿素衍生物做為類香草素受體之配位體 |
Country Status (13)
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3224252B1 (en) * | 2014-11-24 | 2019-01-09 | Medifron Dbt Inc. | Substituted oxazole- and thiazole-based carboxamide and urea derivatives as vanilloid receptor ligands ii |
| CN114920697A (zh) * | 2022-05-16 | 2022-08-19 | 河南应用技术职业学院 | 杂环基取代的茚满丙酰胺类化合物及其应用 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999012910A1 (fr) * | 1997-09-11 | 1999-03-18 | Nissan Chemical Industries, Ltd. | Composes a base de pyrazole et agent de lutte contre les maladies vegetales |
| AR056875A1 (es) * | 2005-10-19 | 2007-10-31 | Gruenenthal Gmbh | Ligandos del receptor vaniloide y su aplicacion para la fabricacion de medicamentos |
| WO2008073825A1 (en) * | 2006-12-08 | 2008-06-19 | Exelixis, Inc. | Lxr and fxr modulators |
| BRPI0810035A2 (pt) * | 2007-04-16 | 2016-07-26 | Gruenenthal Gmbh | ligantes de receptor de vaniloide e seu uso para produção de medicamento |
| DE102007018151A1 (de) * | 2007-04-16 | 2008-10-23 | Günenthal GmbH | Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln |
| MX2011011797A (es) | 2009-05-07 | 2011-11-29 | Gruenenthal Gmbh | Fenilureas y fenilamidas sustituidas como ligandos del receptor de vanilloides. |
| PT2427436E (pt) | 2009-05-07 | 2013-03-04 | Gruenenthal Gmbh | Derivados aromáticos substituídos de carboxamida e ureia como ligantes de receptor de vanilóide |
| EP2776424A1 (en) * | 2011-11-09 | 2014-09-17 | Grünenthal GmbH | Substituted pyrazolyl-based carboxamide and urea derivatives bearing a phenyl moiety substituted with an n-cyclic group as vanilloid receptor ligands |
-
2012
- 2012-11-08 HK HK15102577.0A patent/HK1202116A1/xx unknown
- 2012-11-08 BR BR112014010957A patent/BR112014010957A2/pt not_active IP Right Cessation
- 2012-11-08 WO PCT/EP2012/072141 patent/WO2013068462A1/en active Application Filing
- 2012-11-08 TW TW101141482A patent/TW201326134A/zh unknown
- 2012-11-08 IN IN847KON2014 patent/IN2014KN00847A/en unknown
- 2012-11-08 CA CA2854935A patent/CA2854935A1/en not_active Abandoned
- 2012-11-08 AR ARP120104203A patent/AR088701A1/es unknown
- 2012-11-08 CN CN201280055195.9A patent/CN103906736A/zh active Pending
- 2012-11-08 MX MX2014005611A patent/MX2014005611A/es not_active Application Discontinuation
- 2012-11-08 AU AU2012334066A patent/AU2012334066A1/en not_active Abandoned
- 2012-11-08 EP EP12781341.8A patent/EP2776399A1/en not_active Withdrawn
- 2012-11-08 JP JP2014540454A patent/JP2014532742A/ja active Pending
- 2012-11-08 KR KR1020147015425A patent/KR20140096351A/ko not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| MX2014005611A (es) | 2014-07-30 |
| AU2012334066A1 (en) | 2014-05-22 |
| IN2014KN00847A (enrdf_load_html_response) | 2015-10-02 |
| EP2776399A1 (en) | 2014-09-17 |
| BR112014010957A2 (pt) | 2017-06-06 |
| WO2013068462A1 (en) | 2013-05-16 |
| CA2854935A1 (en) | 2013-05-16 |
| AR088701A1 (es) | 2014-06-25 |
| CN103906736A (zh) | 2014-07-02 |
| HK1202116A1 (en) | 2015-09-18 |
| JP2014532742A (ja) | 2014-12-08 |
| KR20140096351A (ko) | 2014-08-05 |
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