TW200804383A - New compounds - Google Patents
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- TW200804383A TW200804383A TW096119344A TW96119344A TW200804383A TW 200804383 A TW200804383 A TW 200804383A TW 096119344 A TW096119344 A TW 096119344A TW 96119344 A TW96119344 A TW 96119344A TW 200804383 A TW200804383 A TW 200804383A
- Authority
- TW
- Taiwan
- Prior art keywords
- disease
- compound
- pharmaceutically acceptable
- formula
- alkyl group
- Prior art date
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Classifications
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- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
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- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US20110144049A1 (en) * | 2009-10-21 | 2011-06-16 | Serebruany Victor L | Treating Cardiac Arrhythmias, Heart Failure, Peripheral Artery Disease and Stroke with Cyclopentyl-Triazolo-Pyrimidine or Derivative Thereof |
| US8765126B2 (en) * | 2011-05-05 | 2014-07-01 | Robert Sackstein | Methods of treating complications and disorders associated with G-CSF administration |
| BR112014011254A2 (pt) * | 2011-11-11 | 2017-05-16 | Pfizer | 2-tiopirimidinonas |
| US9221821B2 (en) | 2012-06-05 | 2015-12-29 | Forest Laboratories Holdings, Limited | Methods for the synthesis of 1,3-substituted aminouracils and other xanthine-related compounds |
| WO2015134210A1 (en) | 2014-03-03 | 2015-09-11 | Principia Biopharma, Inc. | BENZIMIDAZOLE DERIVATIVES AS RLK and ITK INHIBITORS |
| WO2015196245A1 (en) * | 2014-06-25 | 2015-12-30 | Adelaide Research & Innovation Pty Ltd | Modulation of osteogenesis and or angiogenesis by modulating peroxidase functionality |
| US9616063B2 (en) | 2014-12-01 | 2017-04-11 | Astrazeneca Ab | 1-[2-(aminomethyl)benzyl]-2-thioxo-1,2,3,5-tetrahydro-4H-pyrrolo[3,2-d]pyrimidin-4-ones as inhibitors of myeloperoxidase |
| CR20170498A (es) | 2015-05-05 | 2018-01-26 | Pfizer | 2-tiopirimidinonas |
| EP3298011B1 (en) | 2015-05-22 | 2021-11-17 | Principia Biopharma Inc. | Quinolone derivatives as fibroblast growth factor receptor inhibitors |
| HRP20211249T1 (hr) | 2015-06-03 | 2021-11-12 | Principia Biopharma Inc. | Inhibitori tirozin kinaze |
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| FR2665636B1 (fr) | 1990-08-10 | 1994-10-07 | Adir | Utilisation d'un derive de la trimethyl-1,3,7 xanthine pour le traitement des troubles de la memoire, des troubles intellectuels de la senescence et de la maladie d'alzheimer. |
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| ES2208063B1 (es) | 2002-04-01 | 2005-10-01 | Almirall Prodesfarma, S.A. | Nuevos derivados de la 4-(pirrolopirimidin-6-il)bencenosulfonamida. |
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| WO2006045564A1 (en) | 2004-10-22 | 2006-05-04 | Smithkline Beecham Corporation | Xanthine derivatives with hm74a receptor activity |
| SE0402591D0 (sv) | 2004-10-25 | 2004-10-25 | Astrazeneca Ab | Novel use |
| MY140748A (en) | 2004-12-06 | 2010-01-15 | Astrazeneca Ab | Novel pyrrolo [3,2-d] pyrimidin-4-one derivatives and their use in therapy |
| TW200806667A (en) * | 2006-04-13 | 2008-02-01 | Astrazeneca Ab | New compounds |
| TW200804383A (en) * | 2006-06-05 | 2008-01-16 | Astrazeneca Ab | New compounds |
| US20090054468A1 (en) * | 2007-08-23 | 2009-02-26 | Astrazeneca Ab | New Use 938 |
-
2007
- 2007-05-30 TW TW096119344A patent/TW200804383A/zh unknown
- 2007-05-31 AR ARP070102350A patent/AR061134A1/es not_active Application Discontinuation
- 2007-06-01 CL CL2007001590A patent/CL2007001590A1/es unknown
- 2007-06-01 US US11/756,967 patent/US7943625B2/en not_active Expired - Fee Related
- 2007-06-04 CA CA002653774A patent/CA2653774A1/en not_active Abandoned
- 2007-06-04 BR BRPI0712310-8A patent/BRPI0712310A2/pt not_active IP Right Cessation
- 2007-06-04 UA UAA200813045A patent/UA94606C2/ru unknown
- 2007-06-04 MX MX2008014991A patent/MX2008014991A/es active IP Right Grant
- 2007-06-04 KR KR1020087029646A patent/KR20090014189A/ko not_active Withdrawn
- 2007-06-04 RU RU2008145971/04A patent/RU2435772C2/ru not_active IP Right Cessation
- 2007-06-04 JP JP2009514228A patent/JP2009539828A/ja active Pending
- 2007-06-04 UY UY30387A patent/UY30387A1/es unknown
- 2007-06-04 WO PCT/SE2007/000537 patent/WO2007142576A1/en not_active Ceased
- 2007-06-04 US US12/300,673 patent/US20090131459A1/en not_active Abandoned
- 2007-06-04 EP EP07748200A patent/EP2029598A4/en not_active Withdrawn
- 2007-06-04 CN CNA2007800209903A patent/CN101460498A/zh active Pending
- 2007-06-04 AU AU2007256005A patent/AU2007256005B2/en not_active Ceased
-
2008
- 2008-11-13 IL IL195287A patent/IL195287A0/en unknown
- 2008-11-17 ZA ZA200809800A patent/ZA200809800B/xx unknown
- 2008-12-12 EC EC2008008965A patent/ECSP088965A/es unknown
- 2008-12-16 NO NO20085269A patent/NO20085269L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| US7943625B2 (en) | 2011-05-17 |
| UA94606C2 (ru) | 2011-05-25 |
| EP2029598A4 (en) | 2010-02-17 |
| UY30387A1 (es) | 2008-01-31 |
| MX2008014991A (es) | 2008-12-05 |
| NO20085269L (no) | 2009-03-05 |
| WO2007142576A1 (en) | 2007-12-13 |
| AR061134A1 (es) | 2008-08-06 |
| US20080221133A1 (en) | 2008-09-11 |
| CA2653774A1 (en) | 2007-12-13 |
| IL195287A0 (en) | 2009-08-03 |
| US20090131459A1 (en) | 2009-05-21 |
| AU2007256005B2 (en) | 2011-03-17 |
| RU2435772C2 (ru) | 2011-12-10 |
| JP2009539828A (ja) | 2009-11-19 |
| EP2029598A1 (en) | 2009-03-04 |
| CL2007001590A1 (es) | 2008-01-25 |
| KR20090014189A (ko) | 2009-02-06 |
| AU2007256005A1 (en) | 2007-12-13 |
| ECSP088965A (es) | 2009-01-30 |
| CN101460498A (zh) | 2009-06-17 |
| ZA200809800B (en) | 2010-04-28 |
| RU2008145971A (ru) | 2010-07-20 |
| BRPI0712310A2 (pt) | 2012-01-17 |
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