TR200401815T4 - Evcil hayvanlarda pirimidin endotelin antagonistlerinin kullanımı. - Google Patents
Evcil hayvanlarda pirimidin endotelin antagonistlerinin kullanımı.Info
- Publication number
- TR200401815T4 TR200401815T4 TR2004/01815T TR200401815T TR200401815T4 TR 200401815 T4 TR200401815 T4 TR 200401815T4 TR 2004/01815 T TR2004/01815 T TR 2004/01815T TR 200401815 T TR200401815 T TR 200401815T TR 200401815 T4 TR200401815 T4 TR 200401815T4
- Authority
- TR
- Turkey
- Prior art keywords
- domestic animals
- pyrimidine
- endothelin antagonists
- endothelin
- antagonists
- Prior art date
Links
- 102000002045 Endothelin Human genes 0.000 title abstract 2
- 108050009340 Endothelin Proteins 0.000 title abstract 2
- 241001465754 Metazoa Species 0.000 title abstract 2
- ZUBDGKVDJUIMQQ-UBFCDGJISA-N endothelin-1 Chemical compound C([C@@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CC=1C2=CC=CC=C2NC=1)C(O)=O)NC(=O)[C@H]1NC(=O)[C@H](CC=2C=CC=CC=2)NC(=O)[C@@H](CC=2C=CC(O)=CC=2)NC(=O)[C@H](C(C)C)NC(=O)[C@H]2CSSC[C@@H](C(N[C@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](CCSC)C(=O)N[C@H](CC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N2)=O)NC(=O)[C@@H](CO)NC(=O)[C@H](N)CSSC1)C1=CNC=N1 ZUBDGKVDJUIMQQ-UBFCDGJISA-N 0.000 title abstract 2
- CZPWVGJYEJSRLH-UHFFFAOYSA-N Pyrimidine Chemical compound C1=CN=CN=C1 CZPWVGJYEJSRLH-UHFFFAOYSA-N 0.000 title 1
- 239000005557 antagonist Substances 0.000 title 1
- 241000282472 Canis lupus familiaris Species 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Epidemiology (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Chemical Treatment Of Metals (AREA)
Abstract
Ikame maddelerinin burada tarif edilen degerlere sahip oldugu formül I'in bilesikleri, evcil hayvanlarda özellikle köpekler, kendiler ve atlarda endotelin'in aracilik ettigi bozukluklarin iyilestirilmesinde faydalidir.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0003234.2A GB0003234D0 (en) | 2000-02-11 | 2000-02-11 | Method of treatment |
| PCT/IB2001/000142 WO2001058882A1 (en) | 2000-02-11 | 2001-02-06 | Use of pyrimidine endothelin antagonists in companion animals |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR200401815T4 true TR200401815T4 (tr) | 2004-08-23 |
Family
ID=9885465
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2004/01815T TR200401815T4 (tr) | 2000-02-11 | 2001-02-06 | Evcil hayvanlarda pirimidin endotelin antagonistlerinin kullanımı. |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP1254120B1 (tr) |
| JP (1) | JP2003528050A (tr) |
| KR (1) | KR20020075791A (tr) |
| AT (1) | ATE271042T1 (tr) |
| AU (1) | AU3043601A (tr) |
| CA (1) | CA2398007A1 (tr) |
| DE (1) | DE60104283T2 (tr) |
| DK (1) | DK1254120T3 (tr) |
| ES (1) | ES2222975T3 (tr) |
| GB (1) | GB0003234D0 (tr) |
| HU (1) | HUP0204370A3 (tr) |
| IL (1) | IL150488A0 (tr) |
| NZ (1) | NZ519002A (tr) |
| PT (1) | PT1254120E (tr) |
| TR (1) | TR200401815T4 (tr) |
| WO (1) | WO2001058882A1 (tr) |
| ZA (1) | ZA200206343B (tr) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8647660B2 (en) | 2004-12-29 | 2014-02-11 | Hill's Pet Nutrition, Inc. | Combination of limited nutrients and enhanced dietary antioxidants to impart improved kidney health |
| WO2006113752A1 (en) | 2005-04-19 | 2006-10-26 | Hill's Pet Nutrition, Inc. | Methods and compositions for the prevention and treatment of kidney disease |
| JP5637608B2 (ja) * | 2010-02-25 | 2014-12-10 | エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ | 高親和性化合物の結合定数を求めるための方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP3087968B2 (ja) * | 1995-12-20 | 2000-09-18 | 山之内製薬株式会社 | アリールエテンスルホンアミド誘導体及びその医薬組成物 |
| WO1998057938A1 (fr) * | 1997-06-19 | 1998-12-23 | Yamanouchi Pharmaceutical Co., Ltd. | Derives d'alcanesulfonamide inferieur substitue et composition pharmaceutique les contenant |
-
2000
- 2000-02-11 GB GBGB0003234.2A patent/GB0003234D0/en not_active Ceased
-
2001
- 2001-02-06 ES ES01902578T patent/ES2222975T3/es not_active Expired - Lifetime
- 2001-02-06 NZ NZ519002A patent/NZ519002A/en unknown
- 2001-02-06 KR KR1020027010354A patent/KR20020075791A/ko not_active Application Discontinuation
- 2001-02-06 EP EP01902578A patent/EP1254120B1/en not_active Expired - Lifetime
- 2001-02-06 JP JP2001558433A patent/JP2003528050A/ja not_active Withdrawn
- 2001-02-06 TR TR2004/01815T patent/TR200401815T4/tr unknown
- 2001-02-06 DE DE2001604283 patent/DE60104283T2/de not_active Expired - Fee Related
- 2001-02-06 DK DK01902578T patent/DK1254120T3/da active
- 2001-02-06 HU HU0204370A patent/HUP0204370A3/hu unknown
- 2001-02-06 CA CA002398007A patent/CA2398007A1/en not_active Abandoned
- 2001-02-06 PT PT01902578T patent/PT1254120E/pt unknown
- 2001-02-06 WO PCT/IB2001/000142 patent/WO2001058882A1/en not_active Application Discontinuation
- 2001-02-06 AU AU30436/01A patent/AU3043601A/en not_active Abandoned
- 2001-02-06 IL IL15048801A patent/IL150488A0/xx unknown
- 2001-02-06 AT AT01902578T patent/ATE271042T1/de not_active IP Right Cessation
-
2002
- 2002-08-08 ZA ZA200206343A patent/ZA200206343B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2003528050A (ja) | 2003-09-24 |
| PT1254120E (pt) | 2004-10-29 |
| ATE271042T1 (de) | 2004-07-15 |
| WO2001058882A1 (en) | 2001-08-16 |
| HUP0204370A3 (en) | 2003-07-28 |
| KR20020075791A (ko) | 2002-10-05 |
| CA2398007A1 (en) | 2001-08-16 |
| DK1254120T3 (da) | 2004-10-04 |
| DE60104283D1 (de) | 2004-08-19 |
| DE60104283T2 (de) | 2004-11-18 |
| EP1254120B1 (en) | 2004-07-14 |
| NZ519002A (en) | 2004-06-25 |
| GB0003234D0 (en) | 2000-04-05 |
| IL150488A0 (en) | 2002-12-01 |
| HUP0204370A2 (en) | 2003-05-28 |
| AU3043601A (en) | 2001-08-20 |
| ES2222975T3 (es) | 2005-02-16 |
| EP1254120A1 (en) | 2002-11-06 |
| ZA200206343B (en) | 2003-08-08 |
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