SV2002000418A - INHIBITOR OF THE PARTNER-HYDROGEN EXCHANGER OF TYPE 1 REF. PC1086AADO / BB - Google Patents

INHIBITOR OF THE PARTNER-HYDROGEN EXCHANGER OF TYPE 1 REF. PC1086AADO / BB

Info

Publication number
SV2002000418A
SV2002000418A SV2001000418A SV2001000418A SV2002000418A SV 2002000418 A SV2002000418 A SV 2002000418A SV 2001000418 A SV2001000418 A SV 2001000418A SV 2001000418 A SV2001000418 A SV 2001000418A SV 2002000418 A SV2002000418 A SV 2002000418A
Authority
SV
El Salvador
Prior art keywords
inhibitor
pc1086aado
ref
partner
type
Prior art date
Application number
SV2001000418A
Other languages
Spanish (es)
Inventor
Weichao George Chen
Eric David Cox
Perez Angel Guzman
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of SV2002000418A publication Critical patent/SV2002000418A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Abstract

UN INHIBIDOR DE NHE-1, METODOS PARA UTILIZAR EL INHIBIDOR DE NHE-1 Y COMPOSICIONES FARMACEUTICAS QUE CONTIENEN EL INHIBIDOR DE NHE-1. EL INHIBIDOR DE NHE-1 ES UTIL PARA LA REDUCCION DE LAS LESIONES TISULARES RESULTANTES DE LA ISQUEMIA DE LOS TEJIDOS.AN NHE-1 INHIBITOR, METHODS FOR USING THE NHE-1 INHIBITOR AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE NHE-1 INHIBITOR. THE NHE-1 INHIBITOR IS USEFUL FOR THE REDUCTION OF THE TISSULAR INJURIES RESULTING FROM THE TISSUE ISCHEMIA.

SV2001000418A 2000-04-28 2001-04-27 INHIBITOR OF THE PARTNER-HYDROGEN EXCHANGER OF TYPE 1 REF. PC1086AADO / BB SV2002000418A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US20043200P 2000-04-28 2000-04-28

Publications (1)

Publication Number Publication Date
SV2002000418A true SV2002000418A (en) 2002-07-03

Family

ID=22741697

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2001000418A SV2002000418A (en) 2000-04-28 2001-04-27 INHIBITOR OF THE PARTNER-HYDROGEN EXCHANGER OF TYPE 1 REF. PC1086AADO / BB

Country Status (40)

Country Link
EP (1) EP1276737A1 (en)
JP (1) JP2003531900A (en)
KR (1) KR20020093079A (en)
CN (1) CN1225466C (en)
AP (1) AP2002002651A0 (en)
AR (1) AR028375A1 (en)
AU (1) AU2001235896A1 (en)
BG (1) BG107139A (en)
BR (1) BR0110268A (en)
CA (1) CA2407535A1 (en)
CO (1) CO5221125A1 (en)
CR (1) CR6797A (en)
CZ (1) CZ20023408A3 (en)
DZ (1) DZ3310A1 (en)
EA (1) EA004882B1 (en)
EE (1) EE200200615A (en)
GT (1) GT200100064A (en)
HN (1) HN2001000042A (en)
HR (1) HRP20020851A2 (en)
HU (1) HUP0300651A2 (en)
IL (1) IL152075A0 (en)
IS (2) IS6567A (en)
MA (1) MA26897A1 (en)
MX (1) MXPA02010600A (en)
MY (1) MY133842A (en)
NO (1) NO20025132L (en)
NZ (1) NZ521348A (en)
OA (1) OA12256A (en)
PA (1) PA8513301A1 (en)
PE (1) PE20011270A1 (en)
PL (1) PL357765A1 (en)
SK (1) SK14872002A3 (en)
SV (1) SV2002000418A (en)
TN (1) TNSN01065A1 (en)
TR (1) TR200202439T2 (en)
UA (1) UA73348C2 (en)
UY (1) UY26680A1 (en)
WO (1) WO2001083470A1 (en)
YU (1) YU79602A (en)
ZA (1) ZA200208605B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002060892A1 (en) * 2001-01-31 2002-08-08 Pfizer Products Inc. Ethanolates of sodium-hydrogen exchanger type-1 inhibitor
CA2469305A1 (en) * 2001-12-19 2003-06-26 Frank Robert Busch Methods for preparing sodium-hydrogen exchanger type-1 inhibitors
CA2483927A1 (en) * 2002-05-02 2003-11-13 Pfizer Products Inc. Treatment of diabetes and diabetic complications with nhe-1 inhibitors
FR2840302B1 (en) * 2002-06-03 2004-07-16 Aventis Pharma Sa ISOINDOLONE DERIVATIVES, PREPARATION METHOD AND INTERMEDIARY THEREOF AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME
ES2220185B1 (en) * 2002-07-16 2006-04-01 Consejo Sup. De Investig. Cientificas NEW INHIBITOR PEPTIDE OF THE NA + / H + EXCHANGER (PINHE), AND ITS APPLICATIONS.
EP1596860A4 (en) * 2003-02-14 2009-05-27 Smithkline Beecham Corp Novel compounds
RU2518741C1 (en) * 2013-03-22 2014-06-10 Федеральное государственное автономное образовательное учреждение высшего профессионального образования "ЮЖНЫЙ ФЕДЕРАЛЬНЫЙ УНИВЕРСИТЕТ" MEDICATION, INHIBITING Na+/H+-EXCHANGE, AND HALOGENIDES OF 1-DIALKYLAMINOETHYL-3-[SUBSTITUTED(DISUBSTITUTED)PHENACYL]-2-AMINOBENZIMIDAZOLIUM

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU739403B2 (en) * 1998-02-27 2001-10-11 Pfizer Products Inc. N-((substituted five-membered di- or triaza diunsaturated ring)carbonyl) guanidine derivatives for the treatment of ischemia

Also Published As

Publication number Publication date
UY26680A1 (en) 2001-12-28
OA12256A (en) 2003-11-06
CR6797A (en) 2004-05-17
MXPA02010600A (en) 2003-03-10
IS6588A (en) 2002-10-21
TNSN01065A1 (en) 2005-11-10
DZ3310A1 (en) 2001-11-07
IS6567A (en) 2002-09-24
JP2003531900A (en) 2003-10-28
CO5221125A1 (en) 2002-11-28
PL357765A1 (en) 2004-07-26
IL152075A0 (en) 2003-05-29
TR200202439T2 (en) 2003-02-21
EP1276737A1 (en) 2003-01-22
NO20025132D0 (en) 2002-10-25
PE20011270A1 (en) 2001-12-12
MA26897A1 (en) 2004-12-20
YU79602A (en) 2006-05-25
NZ521348A (en) 2004-09-24
UA73348C2 (en) 2005-07-15
NO20025132L (en) 2002-12-12
CN1426404A (en) 2003-06-25
KR20020093079A (en) 2002-12-12
AU2001235896A1 (en) 2001-11-12
AP2002002651A0 (en) 2002-12-31
GT200100064A (en) 2002-03-22
HN2001000042A (en) 2001-07-09
EE200200615A (en) 2004-04-15
HUP0300651A2 (en) 2003-07-28
CA2407535A1 (en) 2001-11-08
HRP20020851A2 (en) 2005-02-28
BG107139A (en) 2003-07-31
ZA200208605B (en) 2003-10-24
EA200201023A1 (en) 2003-02-27
WO2001083470A1 (en) 2001-11-08
CN1225466C (en) 2005-11-02
BR0110268A (en) 2003-12-30
SK14872002A3 (en) 2004-03-02
PA8513301A1 (en) 2003-09-05
EA004882B1 (en) 2004-08-26
AR028375A1 (en) 2003-05-07
MY133842A (en) 2007-11-30
CZ20023408A3 (en) 2004-01-14

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