SV2002000210A - Profarmacos de higromicina a ref. pc10548ajnm/bb - Google Patents

Profarmacos de higromicina a ref. pc10548ajnm/bb

Info

Publication number
SV2002000210A
SV2002000210A SV2000000210A SV2000000210A SV2002000210A SV 2002000210 A SV2002000210 A SV 2002000210A SV 2000000210 A SV2000000210 A SV 2000000210A SV 2000000210 A SV2000000210 A SV 2000000210A SV 2002000210 A SV2002000210 A SV 2002000210A
Authority
SV
El Salvador
Prior art keywords
compounds
infections
propharms
hygromycin
ref
Prior art date
Application number
SV2000000210A
Other languages
English (en)
Inventor
Takushi Kaneko
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of SV2002000210A publication Critical patent/SV2002000210A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/203Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26Acyclic or carbocyclic radicals, substituted by hetero rings

Abstract

ESTA INVENCION SE REFIERE A COMPUESTOS DE FORMULAY A SALES Y SOLVATOS FARMACEUTICAMENTE ACEPTABLES DE ESTOS,SIENDO a, b, X, Y, Z,R1,R2, Y R3 COMO SE HAN DEFINIDO EN LA DESCRIPCION ADJUNTA. LOS COMPUESTOS DE FORMULA I SON AGENTES ANTIBACTERIANOS Y ANTIPROTOZOOARIOS QUE PUEDEN UTILIZARSE PARA TRATAR INFECCIONES BACTERIANAS Y PROTOZOOARIAS Y ENFERMEDADES RELACIONADAS CON DICHAS INFECCIONES. LA INVENCION SE REFIERE TAMBIEN A COMPOSICIONES FARMACEUTICAS QUE CONTIENEN LOS COMPUESTOS DEFORMULA I Y A PROCEDIMIENTOS PARA TRATAR INFECCIONES BACTERIANAS Y PROTOZOOARIAS MEDIANTE LAADMINISTRACIÓN DELOS COMPUESTOS DE FORMULA I.
SV2000000210A 1999-10-29 2000-10-27 Profarmacos de higromicina a ref. pc10548ajnm/bb SV2002000210A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US16272299P 1999-10-29 1999-10-29

Publications (1)

Publication Number Publication Date
SV2002000210A true SV2002000210A (es) 2002-06-07

Family

ID=22586880

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2000000210A SV2002000210A (es) 1999-10-29 2000-10-27 Profarmacos de higromicina a ref. pc10548ajnm/bb

Country Status (32)

Country Link
US (1) US6492342B1 (es)
EP (1) EP1224194A1 (es)
JP (1) JP2003512472A (es)
KR (1) KR20020043255A (es)
CN (1) CN1382149A (es)
AP (1) AP2002002492A0 (es)
AR (1) AR026285A1 (es)
AU (1) AU7307900A (es)
BG (1) BG106635A (es)
BR (1) BR0015156A (es)
CA (1) CA2389019A1 (es)
CO (1) CO5261547A1 (es)
CZ (1) CZ20021347A3 (es)
EA (1) EA200200413A1 (es)
EC (1) ECSP003743A (es)
EE (1) EE200200226A (es)
GT (1) GT200000178A (es)
HK (1) HK1049844A1 (es)
HU (1) HUP0203223A2 (es)
IL (1) IL148580A0 (es)
IS (1) IS6312A (es)
MA (1) MA26839A1 (es)
MX (1) MXPA02004359A (es)
NO (1) NO20021822D0 (es)
OA (1) OA12079A (es)
PE (1) PE20010757A1 (es)
PL (1) PL357080A1 (es)
SK (1) SK5322002A3 (es)
SV (1) SV2002000210A (es)
TN (1) TNSN00209A1 (es)
TR (1) TR200201143T2 (es)
WO (1) WO2001030793A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020041179A1 (en) * 2018-08-20 2020-02-27 Northeastern University Hygromycin a compounds and methods of treating spirochete diseases

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ID28848A (id) * 1998-12-02 2001-07-05 Pfizer Prod Inc Turunan-turunan higromisin a

Also Published As

Publication number Publication date
OA12079A (en) 2006-05-04
EP1224194A1 (en) 2002-07-24
BR0015156A (pt) 2002-07-16
GT200000178A (es) 2002-04-09
HUP0203223A2 (en) 2003-02-28
MXPA02004359A (es) 2002-11-07
IL148580A0 (en) 2002-09-12
EA200200413A1 (ru) 2002-10-31
TR200201143T2 (tr) 2002-08-21
EE200200226A (et) 2003-06-16
AR026285A1 (es) 2003-02-05
NO20021822L (no) 2002-04-18
IS6312A (is) 2002-03-19
BG106635A (en) 2002-12-29
HK1049844A1 (zh) 2003-05-30
NO20021822D0 (no) 2002-04-18
MA26839A1 (fr) 2004-12-20
PE20010757A1 (es) 2001-07-25
TNSN00209A1 (fr) 2005-11-10
CN1382149A (zh) 2002-11-27
AU7307900A (en) 2001-05-08
PL357080A1 (en) 2004-07-12
AP2002002492A0 (en) 2002-06-30
JP2003512472A (ja) 2003-04-02
SK5322002A3 (en) 2003-01-09
CA2389019A1 (en) 2001-05-03
CZ20021347A3 (cs) 2002-11-13
WO2001030793A1 (en) 2001-05-03
CO5261547A1 (es) 2003-03-31
US6492342B1 (en) 2002-12-10
ECSP003743A (es) 2002-05-23
KR20020043255A (ko) 2002-06-08

Similar Documents

Publication Publication Date Title
PA8486001A1 (es) Composiciones de celecoxib
TR200201505T2 (tr) Terapötik maddeler olarak pirazolopirimidinler
CO4930259A1 (es) Derivados 6,6-heterobiciclicos sustituidos y composiciones farmaceuticas que los contienen
PA8489501A1 (es) Antibioticos cetolidos
PA8591701A1 (es) Derivados de pirrolopirimidina
HN2000000115A (es) Formulacion de sal comun y moxifloxacina
BG108268A (en) Pyrazolopyrimidines as therapeutic agents
BR9911482A (pt) Composto, composição farmacêutica, uso do composto, e, processos para o tratamento ou profilaxia de doenças inflamatórias, e para a preparação de um composto
BG108269A (en) Pyrazolopyrimidines as therapeutic agents
DE60038183D1 (de) Verbindungen und zusammensetzungen zur abgabe aktiver wirkstoffe
CO4810375A1 (es) Derivados de 9-amino-3-ceto eritromicina
PA8432901A1 (es) Compuestos de piridilpirrol
PA8495101A1 (es) Derivados de 13-metileritromicina
PA8451801A1 (es) Derivados de la 9-oxima eritromicina
PA8465901A1 (es) Nuevos derivados de la eritromicina
PA8485601A1 (es) Azalidas de 13 miembros y su uso como agentes antibioticos.
SE0101932D0 (sv) Pharmaceutical combinations
SE9901077D0 (sv) Novel use
AR021843A1 (es) Derivados de propanolamina sustituidos con heterociclos, procedimiento para su preparacion, y su utilizacion.
SE9801494D0 (sv) Novel use
AR020563A1 (es) Compuestos (poli)tia-alquinoicos y sus derivados, composiciones que los incluyen y su utilizacion
CO4810376A1 (es) Derivados de eritromicina triciclicos
PA8471801A1 (es) Derivados de higromicina a
AR025379A1 (es) 9a-azalidas con actividad antibacteriana.
SV2002000210A (es) Profarmacos de higromicina a ref. pc10548ajnm/bb