SK60394A3 - 2-hydroxy-3-£1-(1h-imidazol-4-yl)alkyl|-benzenecarboxamidines, method of their preparation and ophthalmologic compositions with their contents - Google Patents

2-hydroxy-3-£1-(1h-imidazol-4-yl)alkyl|-benzenecarboxamidines, method of their preparation and ophthalmologic compositions with their contents Download PDF

Info

Publication number
SK60394A3
SK60394A3 SK603-94A SK60394A SK60394A3 SK 60394 A3 SK60394 A3 SK 60394A3 SK 60394 A SK60394 A SK 60394A SK 60394 A3 SK60394 A3 SK 60394A3
Authority
SK
Slovakia
Prior art keywords
imidazol
hydroxy
alkyl
formula
toxic
Prior art date
Application number
SK603-94A
Other languages
English (en)
Slovak (sk)
Inventor
Philippe Michel
Eric Cossement
Jean Gobert
Ernst Wulfert
Original Assignee
Ucb Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ucb Sa filed Critical Ucb Sa
Publication of SK60394A3 publication Critical patent/SK60394A3/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Treatments For Attaching Organic Compounds To Fibrous Goods (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SK603-94A 1993-05-27 1994-05-23 2-hydroxy-3-£1-(1h-imidazol-4-yl)alkyl|-benzenecarboxamidines, method of their preparation and ophthalmologic compositions with their contents SK60394A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB939310965A GB9310965D0 (en) 1993-05-27 1993-05-27 2-hydroxy-3-(1h-imidazol-4-yl)alkyl)benzenecarboximidamides

Publications (1)

Publication Number Publication Date
SK60394A3 true SK60394A3 (en) 1995-07-11

Family

ID=10736226

Family Applications (1)

Application Number Title Priority Date Filing Date
SK603-94A SK60394A3 (en) 1993-05-27 1994-05-23 2-hydroxy-3-£1-(1h-imidazol-4-yl)alkyl|-benzenecarboxamidines, method of their preparation and ophthalmologic compositions with their contents

Country Status (21)

Country Link
US (1) US5385927A (ru)
EP (1) EP0626372B1 (ru)
JP (1) JPH0770082A (ru)
AT (1) ATE198196T1 (ru)
AU (1) AU673422B2 (ru)
CA (1) CA2124289A1 (ru)
CZ (1) CZ287136B6 (ru)
DE (1) DE69426433D1 (ru)
FI (1) FI942390A (ru)
GB (1) GB9310965D0 (ru)
HU (1) HUT67813A (ru)
IL (1) IL109750A (ru)
MY (1) MY111216A (ru)
NO (1) NO303824B1 (ru)
NZ (1) NZ260588A (ru)
PL (1) PL175970B1 (ru)
RU (1) RU2125557C1 (ru)
SG (1) SG42791A1 (ru)
SK (1) SK60394A3 (ru)
TW (1) TW263500B (ru)
ZA (1) ZA943651B (ru)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9521680D0 (en) * 1995-10-23 1996-01-03 Orion Yhtymo Oy New use of imidazole derivatives
US6200967B1 (en) 1996-06-25 2001-03-13 Eli Lilly And Company Anticoagulant agents
WO1997049404A1 (en) 1996-06-25 1997-12-31 Eli Lilly And Company Anticoagulant agents
US7902247B2 (en) * 2008-01-09 2011-03-08 Allergan, Inc. Substituted-aryl-2-phenylethyl-1H-imidazole compounds as subtype selective modulators of alpha 2B and/or alpha 2C adrenergic receptors
EP2196461A1 (de) 2008-12-15 2010-06-16 Bayer CropScience AG 4-Amino-1,2,3-benzoxathiazin-Derivate als Pestizide

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8626287D0 (en) * 1986-11-04 1986-12-03 Ucb Sa Substituted 1h-imidazoles
GB8810067D0 (en) * 1988-04-28 1988-06-02 Ucb Sa Substituted 1-(1h-imidazol-4-yl)alkyl-benzamides
FI98815C (fi) * 1990-11-30 1997-08-25 Santen Oy Menetelmä uusien, farmakologisesti käyttökelpoisten bispilokarpiinihapon esterijohdannaisten valmistamiseksi

Also Published As

Publication number Publication date
AU6330394A (en) 1994-12-01
NO303824B1 (no) 1998-09-07
PL175970B1 (pl) 1999-03-31
NO941932D0 (no) 1994-05-25
JPH0770082A (ja) 1995-03-14
IL109750A0 (en) 1994-08-26
IL109750A (en) 1998-06-15
FI942390A0 (fi) 1994-05-24
EP0626372B1 (fr) 2000-12-20
US5385927A (en) 1995-01-31
RU2125557C1 (ru) 1999-01-27
AU673422B2 (en) 1996-11-07
CZ287136B6 (en) 2000-09-13
FI942390A (fi) 1994-11-28
ATE198196T1 (de) 2001-01-15
NZ260588A (en) 1995-09-26
HUT67813A (en) 1995-05-29
HU9401574D0 (en) 1994-08-29
ZA943651B (en) 1995-01-26
CA2124289A1 (en) 1994-11-28
CZ124794A3 (en) 1994-12-15
MY111216A (en) 1999-09-30
EP0626372A1 (fr) 1994-11-30
NO941932L (no) 1994-11-28
SG42791A1 (en) 1997-10-17
TW263500B (ru) 1995-11-21
DE69426433D1 (de) 2001-01-25
GB9310965D0 (en) 1993-07-14

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