SK5552002A3 - Pituitary adenylate cyclase activating peptide (PACAP) receptor 3 (R3) agonists and their pharmacological methods of use - Google Patents
Pituitary adenylate cyclase activating peptide (PACAP) receptor 3 (R3) agonists and their pharmacological methods of use Download PDFInfo
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- SK5552002A3 SK5552002A3 SK555-2002A SK5552002A SK5552002A3 SK 5552002 A3 SK5552002 A3 SK 5552002A3 SK 5552002 A SK5552002 A SK 5552002A SK 5552002 A3 SK5552002 A3 SK 5552002A3
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/57563—Vasoactive intestinal peptide [VIP]; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- General Health & Medical Sciences (AREA)
- Endocrinology (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Toxicology (AREA)
- General Chemical & Material Sciences (AREA)
- Obesity (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Hematology (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Emergency Medicine (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Vascular Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Zoology (AREA)
- Gastroenterology & Hepatology (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Micro-Organisms Or Cultivation Processes Thereof (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US40783299A | 1999-09-28 | 1999-09-28 | |
| US59528000A | 2000-06-15 | 2000-06-15 | |
| PCT/US2000/026638 WO2001023420A2 (fr) | 1999-09-28 | 2000-09-27 | Recepteurs 3 agonistes (r3) pituitaire adenyl cyclase activateur de peptide (pacap) et leurs procedes pharmacologiques d'utilisation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SK5552002A3 true SK5552002A3 (en) | 2003-05-02 |
Family
ID=27020026
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK555-2002A SK5552002A3 (en) | 1999-09-28 | 2000-09-27 | Pituitary adenylate cyclase activating peptide (PACAP) receptor 3 (R3) agonists and their pharmacological methods of use |
Country Status (19)
| Country | Link |
|---|---|
| EP (1) | EP1192182B1 (fr) |
| AT (1) | ATE397625T1 (fr) |
| AU (1) | AU7726600A (fr) |
| CA (1) | CA2379604A1 (fr) |
| CO (1) | CO5280048A1 (fr) |
| CZ (1) | CZ296858B6 (fr) |
| DE (1) | DE60039111D1 (fr) |
| DO (1) | DOP2000000071A (fr) |
| ES (1) | ES2307534T3 (fr) |
| GT (1) | GT200000162A (fr) |
| HU (1) | HUP0202175A3 (fr) |
| MY (1) | MY131983A (fr) |
| PE (1) | PE20010612A1 (fr) |
| RU (1) | RU2269354C2 (fr) |
| SK (1) | SK5552002A3 (fr) |
| SV (1) | SV2002000184A (fr) |
| TW (1) | TWI264438B (fr) |
| UY (1) | UY26360A1 (fr) |
| WO (1) | WO2001023420A2 (fr) |
Families Citing this family (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA74912C2 (en) | 2001-07-06 | 2006-02-15 | Merck & Co Inc | Beta-aminotetrahydroimidazo-(1,2-a)-pyrazines and tetratriazolo-(4,3-a)-pyrazines as inhibitors of dipeptylpeptidase for the treatment or prevention of diabetes |
| EP1476178A4 (fr) * | 2002-02-14 | 2009-08-26 | Bayer Pharmaceuticals Corp | Strategies de formulation dans la stabilisation de peptides dans des solvants organiques et a l'etat seche |
| WO2004062684A2 (fr) * | 2003-01-16 | 2004-07-29 | D. Collen Research Foundation Vzw Onderwijs En Navorsing Campus Gasthuisberg K.U. Leuven | Inhibition de la signalisation pacap dans la prevention et le traitement de la thrombocytopenie |
| US7947261B2 (en) | 2003-05-23 | 2011-05-24 | Nektar Therapeutics | Conjugates formed from polymer derivatives having particular atom arrangements |
| ES2725808T3 (es) | 2003-05-23 | 2019-09-27 | Nektar Therapeutics | Derivados de PEG que contienen dos cadenas de PEG |
| RU2006130691A (ru) * | 2004-01-27 | 2008-03-10 | Байер Фармасьютикалс Корпорейшн (US) | Агонисты рецептора (vpac2), активирующего аденилатциклазу гипофиза пептида (расар), и фармакологические способы их применения |
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| EP3035950A4 (fr) * | 2013-08-14 | 2017-05-03 | The Arizona Board Of Regents On Behalf Of The University Of Arizona | Analogues de pacap/vip glycosylés avec pénétration du snc augmentée pour le traitement de maladies neurodégénératives |
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|---|---|---|---|---|
| JP3107225B2 (ja) * | 1990-03-17 | 2000-11-06 | 武田薬品工業株式会社 | Ｐａｃａｐに対する抗体およびその用途 |
| AU656230B2 (en) * | 1991-10-11 | 1995-01-27 | F. Hoffmann-La Roche Ag | Cyclic vasoactive peptides |
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| WO1998002453A2 (fr) * | 1996-07-15 | 1998-01-22 | Universite Libre De Bruxelles | Ligands peptidiques possedant une selectivite plus elevee pour le recepteur vip1 que pour le recepteur vip¿2? |
| FR2775902B1 (fr) * | 1998-03-13 | 2001-05-11 | Assist Publ Hopitaux De Paris | Utilisation d'analogues du vip dans la prevention et le traitement des lesions cerebrales du nouveau-ne humain |
| WO2000005260A1 (fr) * | 1998-07-20 | 2000-02-03 | Societe De Conseils De Recherches Et D'applications Scientifiques Sas | Analogues peptidiques des pacap |
-
2000
- 2000-09-27 EP EP00967002A patent/EP1192182B1/fr not_active Expired - Lifetime
- 2000-09-27 CZ CZ20021085A patent/CZ296858B6/cs not_active IP Right Cessation
- 2000-09-27 DE DE60039111T patent/DE60039111D1/de not_active Expired - Lifetime
- 2000-09-27 WO PCT/US2000/026638 patent/WO2001023420A2/fr active IP Right Grant
- 2000-09-27 ES ES00967002T patent/ES2307534T3/es not_active Expired - Lifetime
- 2000-09-27 RU RU2001136014/15A patent/RU2269354C2/ru active
- 2000-09-27 AU AU77266/00A patent/AU7726600A/en not_active Abandoned
- 2000-09-27 AT AT00967002T patent/ATE397625T1/de not_active IP Right Cessation
- 2000-09-27 PE PE2000001015A patent/PE20010612A1/es not_active Application Discontinuation
- 2000-09-27 CA CA002379604A patent/CA2379604A1/fr not_active Abandoned
- 2000-09-27 HU HU0202175A patent/HUP0202175A3/hu unknown
- 2000-09-27 SK SK555-2002A patent/SK5552002A3/sk unknown
- 2000-09-28 DO DO2000000071A patent/DOP2000000071A/es unknown
- 2000-09-28 TW TW089120330A patent/TWI264438B/zh not_active IP Right Cessation
- 2000-09-28 MY MYPI20004551A patent/MY131983A/en unknown
- 2000-09-28 GT GT200000162A patent/GT200000162A/es unknown
- 2000-09-28 UY UY26360A patent/UY26360A1/es unknown
- 2000-09-28 CO CO00073865A patent/CO5280048A1/es active IP Right Grant
- 2000-09-28 SV SV2000000184A patent/SV2002000184A/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CZ296858B6 (cs) | 2006-07-12 |
| AU7726600A (en) | 2001-04-30 |
| EP1192182B1 (fr) | 2008-06-04 |
| SV2002000184A (es) | 2002-06-07 |
| MY131983A (en) | 2007-09-28 |
| HUP0202175A3 (en) | 2005-01-28 |
| GT200000162A (es) | 2002-03-22 |
| ATE397625T1 (de) | 2008-06-15 |
| CZ20021085A3 (cs) | 2003-01-15 |
| DOP2000000071A (es) | 2002-02-28 |
| PE20010612A1 (es) | 2001-07-12 |
| RU2269354C2 (ru) | 2006-02-10 |
| HUP0202175A2 (en) | 2002-10-28 |
| TWI264438B (en) | 2006-10-21 |
| DE60039111D1 (de) | 2008-07-17 |
| WO2001023420A2 (fr) | 2001-04-05 |
| CO5280048A1 (es) | 2003-05-30 |
| WO2001023420A3 (fr) | 2001-08-30 |
| ES2307534T3 (es) | 2008-12-01 |
| CA2379604A1 (fr) | 2001-04-05 |
| EP1192182A2 (fr) | 2002-04-03 |
| UY26360A1 (es) | 2001-04-30 |
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