SK5322002A3 - Hygromycin A prodrugs - Google Patents

Hygromycin A prodrugs Download PDF

Info

Publication number
SK5322002A3
SK5322002A3 SK532-2002A SK5322002A SK5322002A3 SK 5322002 A3 SK5322002 A3 SK 5322002A3 SK 5322002 A SK5322002 A SK 5322002A SK 5322002 A3 SK5322002 A3 SK 5322002A3
Authority
SK
Slovakia
Prior art keywords
hydrogen
formula
compound
alkyl
acyl
Prior art date
Application number
SK532-2002A
Other languages
English (en)
Slovak (sk)
Inventor
Takushi Kaneko
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of SK5322002A3 publication Critical patent/SK5322002A3/sk

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/203Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26Acyclic or carbocyclic radicals, substituted by hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
SK532-2002A 1999-10-29 2000-09-28 Hygromycin A prodrugs SK5322002A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US16272299P 1999-10-29 1999-10-29
PCT/IB2000/001390 WO2001030793A1 (en) 1999-10-29 2000-09-28 Hygromycin a prodrugs

Publications (1)

Publication Number Publication Date
SK5322002A3 true SK5322002A3 (en) 2003-01-09

Family

ID=22586880

Family Applications (1)

Application Number Title Priority Date Filing Date
SK532-2002A SK5322002A3 (en) 1999-10-29 2000-09-28 Hygromycin A prodrugs

Country Status (32)

Country Link
US (1) US6492342B1 (zh)
EP (1) EP1224194A1 (zh)
JP (1) JP2003512472A (zh)
KR (1) KR20020043255A (zh)
CN (1) CN1382149A (zh)
AP (1) AP2002002492A0 (zh)
AR (1) AR026285A1 (zh)
AU (1) AU7307900A (zh)
BG (1) BG106635A (zh)
BR (1) BR0015156A (zh)
CA (1) CA2389019A1 (zh)
CO (1) CO5261547A1 (zh)
CZ (1) CZ20021347A3 (zh)
EA (1) EA200200413A1 (zh)
EC (1) ECSP003743A (zh)
EE (1) EE200200226A (zh)
GT (1) GT200000178A (zh)
HK (1) HK1049844A1 (zh)
HU (1) HUP0203223A2 (zh)
IL (1) IL148580A0 (zh)
IS (1) IS6312A (zh)
MA (1) MA26839A1 (zh)
MX (1) MXPA02004359A (zh)
NO (1) NO20021822L (zh)
OA (1) OA12079A (zh)
PE (1) PE20010757A1 (zh)
PL (1) PL357080A1 (zh)
SK (1) SK5322002A3 (zh)
SV (1) SV2002000210A (zh)
TN (1) TNSN00209A1 (zh)
TR (1) TR200201143T2 (zh)
WO (1) WO2001030793A1 (zh)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20210275559A1 (en) * 2018-08-20 2021-09-09 Kim Lewis Hygromycin a compounds and methods of treating spirochete diseases

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2352332C (en) * 1998-12-02 2004-12-07 Pfizer Products Inc. Hygromycin a derivatives

Also Published As

Publication number Publication date
AU7307900A (en) 2001-05-08
EP1224194A1 (en) 2002-07-24
CO5261547A1 (es) 2003-03-31
KR20020043255A (ko) 2002-06-08
US6492342B1 (en) 2002-12-10
TNSN00209A1 (fr) 2005-11-10
NO20021822D0 (no) 2002-04-18
HUP0203223A2 (en) 2003-02-28
BR0015156A (pt) 2002-07-16
EE200200226A (et) 2003-06-16
WO2001030793A1 (en) 2001-05-03
HK1049844A1 (zh) 2003-05-30
TR200201143T2 (tr) 2002-08-21
MXPA02004359A (es) 2002-11-07
AR026285A1 (es) 2003-02-05
ECSP003743A (es) 2002-05-23
AP2002002492A0 (en) 2002-06-30
IL148580A0 (en) 2002-09-12
CZ20021347A3 (cs) 2002-11-13
SV2002000210A (es) 2002-06-07
JP2003512472A (ja) 2003-04-02
CN1382149A (zh) 2002-11-27
IS6312A (is) 2002-03-19
MA26839A1 (fr) 2004-12-20
PL357080A1 (en) 2004-07-12
NO20021822L (no) 2002-04-18
CA2389019A1 (en) 2001-05-03
GT200000178A (es) 2002-04-09
PE20010757A1 (es) 2001-07-25
EA200200413A1 (ru) 2002-10-31
OA12079A (en) 2006-05-04
BG106635A (en) 2002-12-29

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