SK1895A3 - Analgetic and nootropic drugs - Google Patents

Analgetic and nootropic drugs Download PDF

Info

Publication number
SK1895A3
SK1895A3 SK18-95A SK1895A SK1895A3 SK 1895 A3 SK1895 A3 SK 1895A3 SK 1895 A SK1895 A SK 1895A SK 1895 A3 SK1895 A3 SK 1895A3
Authority
SK
Slovakia
Prior art keywords
xxx xxx
saline
maleate
compared
phenyl
Prior art date
Application number
SK18-95A
Other languages
English (en)
Slovak (sk)
Inventor
Alessandro Bartolini
Carla Ghelardini
Alberto Giotti
Fulvio Gualtieri
Serena Scapecchi
Gino Toffano
Original Assignee
Fidia Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fidia Spa filed Critical Fidia Spa
Publication of SK1895A3 publication Critical patent/SK1895A3/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SK18-95A 1992-07-08 1993-07-06 Analgetic and nootropic drugs SK1895A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ITMI921659A IT1255323B (it) 1992-07-08 1992-07-08 Composti ad attivita' analgesica e nootropa
PCT/EP1993/001743 WO1994001435A1 (en) 1992-07-08 1993-07-06 New analgesic and nootropic drugs

Publications (1)

Publication Number Publication Date
SK1895A3 true SK1895A3 (en) 1995-07-11

Family

ID=11363636

Family Applications (1)

Application Number Title Priority Date Filing Date
SK18-95A SK1895A3 (en) 1992-07-08 1993-07-06 Analgetic and nootropic drugs

Country Status (14)

Country Link
US (1) US5583142A (it)
EP (1) EP0650486A1 (it)
JP (1) JPH07508739A (it)
KR (1) KR100258336B1 (it)
AU (1) AU4564593A (it)
CA (1) CA2139739A1 (it)
CZ (1) CZ2295A3 (it)
FI (1) FI950029A (it)
HU (1) HUT73481A (it)
IT (1) IT1255323B (it)
NO (1) NO307518B1 (it)
RU (1) RU95105457A (it)
SK (1) SK1895A3 (it)
WO (1) WO1994001435A1 (it)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5794887A (en) 1995-11-17 1998-08-18 Komerath; Narayanan M. Stagnation point vortex controller
EP2206712A1 (en) * 2008-12-23 2010-07-14 CHIESI FARMACEUTICI S.p.A. "Alkaloid aminoester derivatives and medicinal composition thereof"
RU2744571C1 (ru) * 2020-04-10 2021-03-11 Общество с ограниченной ответственностью "ВладМиВа"(ООО "ВладМиВа") Дифармакофорные соединения ноотропно-анальгетического действия и способ их получения

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1289429A (fr) * 1960-03-10 1962-04-06 Lepetit Spa Procédé de préparation des nouveaux esters de la tropine
DE1670142A1 (de) * 1966-09-02 1970-07-16 Boehringer Sohn Ingelheim Verfahren zur Herstellung von Atropin,Scopolamin und deren N-substituierten Derivaten
DE4108393A1 (de) * 1991-03-15 1992-09-17 Boehringer Ingelheim Kg Neue ester bi- und tricyclischer aminoalkohole, ihre herstellung und ihre verwendung in arzneimitteln

Also Published As

Publication number Publication date
WO1994001435A1 (en) 1994-01-20
RU95105457A (ru) 1997-05-10
KR950702557A (ko) 1995-07-29
IT1255323B (it) 1995-10-31
HUT73481A (en) 1996-08-28
FI950029A0 (fi) 1995-01-03
NO307518B1 (no) 2000-04-17
HU9403797D0 (en) 1995-02-28
FI950029A (fi) 1995-03-06
ITMI921659A1 (it) 1994-01-08
CA2139739A1 (en) 1994-01-20
ITMI921659A0 (it) 1992-07-08
EP0650486A1 (en) 1995-05-03
NO950053D0 (no) 1995-01-06
JPH07508739A (ja) 1995-09-28
US5583142A (en) 1996-12-10
KR100258336B1 (ko) 2000-08-01
CZ2295A3 (en) 1996-02-14
NO950053L (no) 1995-01-06
AU4564593A (en) 1994-01-31

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