SK17682002A3 - Liečivá na prevenciu a liečbu neurodegeneratívnych ochorení - Google Patents

Liečivá na prevenciu a liečbu neurodegeneratívnych ochorení Download PDF

Info

Publication number
SK17682002A3
SK17682002A3 SK1768-2002A SK17682002A SK17682002A3 SK 17682002 A3 SK17682002 A3 SK 17682002A3 SK 17682002 A SK17682002 A SK 17682002A SK 17682002 A3 SK17682002 A3 SK 17682002A3
Authority
SK
Slovakia
Prior art keywords
naphthyridin
oxadiazol
treatment
substituted
prevention
Prior art date
Application number
SK1768-2002A
Other languages
English (en)
Slovak (sk)
Inventor
Kiyoshi Furukawa
Satoshi Kurumiya
Kazuo Okimoto
Kazunori Ohno
Original Assignee
Dainippon Pharmaceutical Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dainippon Pharmaceutical Co., Ltd. filed Critical Dainippon Pharmaceutical Co., Ltd.
Publication of SK17682002A3 publication Critical patent/SK17682002A3/sk

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines having two or more nitrogen atoms in the same ring, e.g. oxadiazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SK1768-2002A 2000-06-21 2001-06-12 Liečivá na prevenciu a liečbu neurodegeneratívnych ochorení SK17682002A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2000185814 2000-06-21
PCT/JP2001/004934 WO2001098300A1 (fr) 2000-06-21 2001-06-12 Medicaments utilises dans la prevention et le traitement de maladies neurodegeneratives

Publications (1)

Publication Number Publication Date
SK17682002A3 true SK17682002A3 (sk) 2003-08-05

Family

ID=18686074

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1768-2002A SK17682002A3 (sk) 2000-06-21 2001-06-12 Liečivá na prevenciu a liečbu neurodegeneratívnych ochorení

Country Status (19)

Country Link
US (1) US6743803B2 (hu)
EP (1) EP1295883A4 (hu)
KR (1) KR20030010740A (hu)
CN (1) CN100354274C (hu)
AU (2) AU6274101A (hu)
BR (1) BR0111799A (hu)
CA (1) CA2412199A1 (hu)
CZ (1) CZ20024153A3 (hu)
EE (1) EE04941B1 (hu)
HU (1) HUP0301319A3 (hu)
IL (2) IL153439A0 (hu)
MX (1) MXPA02012599A (hu)
NO (1) NO20026148L (hu)
NZ (1) NZ523189A (hu)
PL (1) PL200537B1 (hu)
RU (1) RU2258506C2 (hu)
SK (1) SK17682002A3 (hu)
TW (1) TWI298068B (hu)
WO (1) WO2001098300A1 (hu)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6822097B1 (en) * 2002-02-07 2004-11-23 Amgen, Inc. Compounds and methods of uses
TW200533371A (en) * 2004-04-15 2005-10-16 Dainippon Pharmaceutical Co Medicament comprising a combination of an acetylcholinesterase inhibitor and a 5-substituted-3-oxadiazolyl-1,6-naphthyridin-2(1h)-one derivative
EP1595881A1 (en) * 2004-05-12 2005-11-16 Pfizer Limited Tetrahydronaphthyridine derivates useful as histamine H3 receptor ligands
WO2010002451A1 (en) * 2008-07-01 2010-01-07 Concert Pharmaceuticals, Inc. Naphthyridin derivatives
JP6551671B2 (ja) * 2015-08-11 2019-07-31 国立大学法人 熊本大学 アルツハイマー治療薬
BR112022000811A2 (pt) * 2019-07-18 2022-03-29 Abaxys Therapeutics Formulação sólida de um derivado de 1,2,4-oxadiazol

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2683818B1 (fr) 1991-11-14 1993-12-31 Adir Cie Nouveaux derives de 3-sulfonylamino-2-(1h)-quinoleinone, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
JPH09291034A (ja) * 1996-02-27 1997-11-11 Yoshitomi Pharmaceut Ind Ltd 縮合ピリジン化合物およびその医薬としての用途
ZA985870B (en) * 1997-07-15 1999-01-27 Dainippon Pharmaceutical Co 5-substituted-3-oxadiazolyl-1, 6-naphthyridin-2(1H)-one derivatives
AR013184A1 (es) * 1997-07-18 2000-12-13 Astrazeneca Ab Aminas heterociclicas espiroazobiciclicas, composicion farmaceutica, uso de dichas aminas para preparar medicamentos y metodo de tratamiento o profilaxis
WO2000073283A1 (en) 1999-06-02 2000-12-07 Nps Pharmaceuticals, Inc. Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases

Also Published As

Publication number Publication date
IL153439A (en) 2007-07-24
EP1295883A1 (en) 2003-03-26
EE200200698A (et) 2004-08-16
PL200537B1 (pl) 2009-01-30
NZ523189A (en) 2004-08-27
TWI298068B (en) 2008-06-21
US20030166673A1 (en) 2003-09-04
AU2001262741B2 (en) 2005-07-07
PL363869A1 (en) 2004-11-29
WO2001098300A1 (fr) 2001-12-27
IL153439A0 (en) 2003-07-06
CN1447809A (zh) 2003-10-08
NO20026148D0 (no) 2002-12-20
KR20030010740A (ko) 2003-02-05
CN100354274C (zh) 2007-12-12
BR0111799A (pt) 2003-05-27
EP1295883A4 (en) 2003-06-11
MXPA02012599A (es) 2003-05-14
EE04941B1 (et) 2007-12-17
AU6274101A (en) 2002-01-02
CA2412199A1 (en) 2001-12-27
HUP0301319A3 (en) 2008-06-30
US6743803B2 (en) 2004-06-01
HUP0301319A2 (hu) 2003-09-29
RU2258506C2 (ru) 2005-08-20
NO20026148L (no) 2003-02-20
CZ20024153A3 (cs) 2003-06-18

Similar Documents

Publication Publication Date Title
US5945416A (en) Method for treating pain
KR20170003527A (ko) 경구 투여용 펜토산 폴리설페이트 염의 조성물
US6262081B1 (en) Composition for and method of treating neurological disorders
EP1063995B1 (en) Combination for the treatment of alcohol dependence containing an opioid antagonist and a nmda receptor complex modulator
JP2000507544A (ja) 痛みの治療方法
CN109475539B (zh) 帕金森氏病的治疗
SK7542003A3 (en) Medicinal compositions containing aspirin
CA2167004C (en) Agent for treating mental disorders associated with cerebrovascular disorders
JPH01100118A (ja) ホスホジエステラーゼ阻害剤及びトロンボキサンa↓2拮抗剤を含む新規な医薬組成物、その使用及びその製造法
SK17682002A3 (sk) Liečivá na prevenciu a liečbu neurodegeneratívnych ochorení
EA015483B1 (ru) ПРИМЕНЕНИЕ ИНГИБИТОРА p38 КИНАЗЫ ДЛЯ ЛЕЧЕНИЯ ПСИХИАТРИЧЕСКИХ РАССТРОЙСТВ
US20080275075A1 (en) Medicine Comprising a Combination of an Acetylcholinesterase Inhibitor and a 5-Substituted-3-Oxadiazolyl-1,6-Naphthyridin-2(1H)-One Derivative
AU2021349680B2 (en) Use of sphingosine-1-phosphate receptor agonist
JP2004508272A (ja) アセチルコリンエンハンサー
RU2761219C2 (ru) Терапевтическое средство от расстройств, связанных с употреблением алкоголя
JP2002249432A (ja) 併用剤
MXPA04012706A (es) Tratamiento de combinacion para depresion y ansiedad.
JP2009510158A (ja) 毒物依存症の治療におけるネボグラミンの使用
CA2423364A1 (en) Preventives/remedies for emotional disorders

Legal Events

Date Code Title Description
FB9A Suspension of patent application procedure