SI3394051T1 - Postopek kristalizacije za pridobivanje kristalov kanagliflozin hemihidrata - Google Patents

Postopek kristalizacije za pridobivanje kristalov kanagliflozin hemihidrata

Info

Publication number
SI3394051T1
SI3394051T1 SI201630770T SI201630770T SI3394051T1 SI 3394051 T1 SI3394051 T1 SI 3394051T1 SI 201630770 T SI201630770 T SI 201630770T SI 201630770 T SI201630770 T SI 201630770T SI 3394051 T1 SI3394051 T1 SI 3394051T1
Authority
SI
Slovenia
Prior art keywords
crystallization procedure
hemihydrate crystals
canagliflozin hemihydrate
obtaining
obtaining canagliflozin
Prior art date
Application number
SI201630770T
Other languages
English (en)
Inventor
Keyser Ruben De
Stijn Laps
Thomas Joachim Landewald Rammeloo
Koen Johan Herman Weerts
Original Assignee
Janssen Pharmaceutica N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica N.V. filed Critical Janssen Pharmaceutica N.V.
Publication of SI3394051T1 publication Critical patent/SI3394051T1/sl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/10Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Crystals, And After-Treatments Of Crystals (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
SI201630770T 2015-12-21 2016-12-20 Postopek kristalizacije za pridobivanje kristalov kanagliflozin hemihidrata SI3394051T1 (sl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP15201459 2015-12-21
EP16172070 2016-05-31
EP16819899.2A EP3394051B1 (en) 2015-12-21 2016-12-20 Crystallization procedure for obtaining canagliflozin hemihydrate crystals
PCT/EP2016/081861 WO2017108752A1 (en) 2015-12-21 2016-12-20 Crystallization procedure for obtaining canagliflozin hemihydrate crystals

Publications (1)

Publication Number Publication Date
SI3394051T1 true SI3394051T1 (sl) 2020-07-31

Family

ID=57681580

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201630770T SI3394051T1 (sl) 2015-12-21 2016-12-20 Postopek kristalizacije za pridobivanje kristalov kanagliflozin hemihidrata

Country Status (18)

Country Link
US (1) US10323025B2 (sl)
EP (1) EP3394051B1 (sl)
JP (1) JP6851379B2 (sl)
KR (1) KR20180095839A (sl)
CN (1) CN108368096B (sl)
AU (1) AU2016376653B2 (sl)
CA (1) CA3006237C (sl)
CY (1) CY1124885T1 (sl)
DK (1) DK3394051T3 (sl)
EA (1) EA036793B1 (sl)
ES (1) ES2794909T3 (sl)
HR (1) HRP20200755T1 (sl)
HU (1) HUE049895T2 (sl)
LT (1) LT3394051T (sl)
PL (1) PL3394051T3 (sl)
PT (1) PT3394051T (sl)
SI (1) SI3394051T1 (sl)
WO (1) WO2017108752A1 (sl)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021012044A1 (en) 2019-07-22 2021-01-28 Canopy Growth Corporation Continuous crystallization of cannabinoids in a stirred-tank reactor

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2780403B3 (fr) * 1998-06-24 2000-07-21 Sanofi Sa Nouvelle forme de l'irbesartan, procedes pour obtenir ladite forme et compositions pharmaceutiques en contenant
GB0301259D0 (en) * 2003-01-20 2003-02-19 Novartis Ag Organic compounds
SI1651658T2 (sl) 2003-08-01 2020-12-31 Mitsubishi Tanabe Pharma Corporation Nove spojine, ki imajo inhibitorno aktivnost proti transporterju, ki je odvisen od natrija
US20080046236A1 (en) * 2006-08-15 2008-02-21 Broadcom Corporation Constrained and Controlled Decoding After Packet Loss
UY30730A1 (es) * 2006-12-04 2008-07-03 Mitsubishi Tanabe Pharma Corp Forma cristalina del hemihidrato de 1-(b (beta)-d-glucopiranosil) -4-metil-3-[5-(4-fluorofenil) -2-tienilmetil]benceno
JP5658751B2 (ja) * 2009-07-10 2015-01-28 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプJanssen Pharmaceutica Naamloze Vennootschap 1−(β−D−グルコピラノシル)−4−メチル−3−[5−(4−フルオロフェニル)−2−チエニルメチル]ベンゼンのための結晶化方法
EP2994468B1 (en) 2013-05-08 2017-07-19 LEK Pharmaceuticals d.d. Crystalline hydrates of 1-(beta-d-glucopyranosyl)-4-methyl-3-[5-(4-fluorophenyl)-2-thienylmethyl]benzene
CZ305172B6 (cs) * 2014-03-28 2015-05-27 Bochemie A.S. Diskontinuální krystalizační jednotka pro výrobu kulovitých krystalů
CN103896930B (zh) * 2014-04-02 2016-08-17 安徽联创生物医药股份有限公司 卡格列净半水合物药用晶型的制备方法

Also Published As

Publication number Publication date
US10323025B2 (en) 2019-06-18
PL3394051T3 (pl) 2020-10-19
ES2794909T3 (es) 2020-11-19
EP3394051A1 (en) 2018-10-31
EA036793B1 (ru) 2020-12-22
DK3394051T3 (da) 2020-07-20
EP3394051B1 (en) 2020-04-22
AU2016376653A1 (en) 2018-06-07
HUE049895T2 (hu) 2020-11-30
EA201891470A1 (ru) 2018-12-28
WO2017108752A1 (en) 2017-06-29
US20190002449A1 (en) 2019-01-03
CN108368096B (zh) 2021-12-10
LT3394051T (lt) 2020-08-10
HRP20200755T1 (hr) 2020-07-24
AU2016376653B2 (en) 2020-07-30
KR20180095839A (ko) 2018-08-28
CA3006237C (en) 2023-10-03
CA3006237A1 (en) 2017-06-29
CN108368096A (zh) 2018-08-03
JP2019504022A (ja) 2019-02-14
JP6851379B2 (ja) 2021-03-31
CY1124885T1 (el) 2022-07-22
PT3394051T (pt) 2020-06-08

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