SI1861404T1 - Polimorfna oblika 6- 4-klorofenil)-2 2-dimetil-7-fenil-2 3-dihidro- 1H-pirolizin-5-ilocetne kisline - Google Patents

Polimorfna oblika 6- 4-klorofenil)-2 2-dimetil-7-fenil-2 3-dihidro- 1H-pirolizin-5-ilocetne kisline

Info

Publication number
SI1861404T1
SI1861404T1 SI200631089T SI200631089T SI1861404T1 SI 1861404 T1 SI1861404 T1 SI 1861404T1 SI 200631089 T SI200631089 T SI 200631089T SI 200631089 T SI200631089 T SI 200631089T SI 1861404 T1 SI1861404 T1 SI 1861404T1
Authority
SI
Slovenia
Prior art keywords
pyrrolizin
chlorophenyl
dihydro
dimethyl
phenyl
Prior art date
Application number
SI200631089T
Other languages
English (en)
Inventor
Wolfgang Albrecht
Thomas Kammermeier
Hans-Gunter Striegel
Philipp Merckle
Stefan Laufer
Original Assignee
Merckle Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merckle Gmbh filed Critical Merckle Gmbh
Publication of SI1861404T1 publication Critical patent/SI1861404T1/sl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SI200631089T 2005-03-21 2006-03-20 Polimorfna oblika 6- 4-klorofenil)-2 2-dimetil-7-fenil-2 3-dihidro- 1H-pirolizin-5-ilocetne kisline SI1861404T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102005012971A DE102005012971A1 (de) 2005-03-21 2005-03-21 Polymorphe Form von 6-(4-Chlorphenyl)-2,2-dimethyl-7-phenyl-2,3-dihydro-1H-pyrrolizin-5-yl-essigsäure
PCT/EP2006/002539 WO2006100019A1 (en) 2005-03-21 2006-03-20 Polymorphic form of 6- (4-chlorophenyl) -2, 2-dimethyl-7-phenyl-2, 3-dihydro-lh-pyrrolizin-5-ylacetic acid
EP06723557A EP1861404B1 (en) 2005-03-21 2006-03-20 Polymorphic form of 6- (4-chlorophenyl) -2, 2-dimethyl-7-phenyl-2, 3-dihydro-lh-pyrrolizin-5-ylacetic acid

Publications (1)

Publication Number Publication Date
SI1861404T1 true SI1861404T1 (sl) 2011-11-30

Family

ID=36568591

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200631089T SI1861404T1 (sl) 2005-03-21 2006-03-20 Polimorfna oblika 6- 4-klorofenil)-2 2-dimetil-7-fenil-2 3-dihidro- 1H-pirolizin-5-ilocetne kisline

Country Status (15)

Country Link
US (1) US8034837B2 (sl)
EP (1) EP1861404B1 (sl)
JP (1) JP5009280B2 (sl)
CN (1) CN101160311B (sl)
AT (1) ATE509932T1 (sl)
AU (1) AU2006226625B2 (sl)
CA (1) CA2602224A1 (sl)
DE (1) DE102005012971A1 (sl)
ES (1) ES2367274T3 (sl)
MX (1) MX2007011455A (sl)
PL (1) PL1861404T3 (sl)
PT (1) PT1861404E (sl)
RU (1) RU2007138924A (sl)
SI (1) SI1861404T1 (sl)
WO (1) WO2006100019A1 (sl)

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3915450A1 (de) 1989-05-11 1990-11-15 Gerd Prof Dr Dannhardt Substituierte pyrrolverbindungen und deren anwendung in der pharmazie
US5260451A (en) * 1989-05-11 1993-11-09 Merckle Gmbh Substituted pyrrole compounds and use thereof in pharmaceutical compositions
DE4419247A1 (de) * 1994-06-01 1995-12-07 Merckle Gmbh Sulfonylierte Pyrrolizincarbonsäureamide und deren Anwendung in der Pharmazie
DE4419315A1 (de) 1994-06-01 1995-12-07 Merckle Gmbh Heteropyrrolizinverbindungen und deren Anwendung in der Pharmazie
DE4419246A1 (de) 1994-06-01 1995-12-07 Merckle Gmbh Heteroarylsubstituierte Pyrrolizinverbindungen und deren Anwendung in der Pharmazie
ATE210461T1 (de) * 1996-02-13 2001-12-15 Searle & Co Zusammensetzungen mit immunosuppressiven wirkungen, welche 5-lipoxygenase-inhibitoren und cyclooxygenase-2-inhibitoren enthalten
EA004938B1 (ru) * 2000-01-28 2004-10-28 Меркле Гмбх Способ получения 6-(4-хлорфенил)-2,2-диметил-7-фенил-2,3-дигидро-1h-пирролизин-5-илуксусной кислоты
DE10141285A1 (de) * 2001-08-23 2003-03-27 Merckle Gmbh Verfahren zur Herstellung von 6-(4-Chlorphenyl)-2,2-dimethyl-7-phnyl-2,3-dihydro-1H-pyrrolizin-5-yl-essigsäure
ES2275218T3 (es) * 2003-05-07 2007-06-01 Osteologix A/S Sales de estroncio hidrosolubles para el tratamiento de afecciones de cartilagos y/o huesos.

Also Published As

Publication number Publication date
AU2006226625A1 (en) 2006-09-28
JP2008535809A (ja) 2008-09-04
CN101160311A (zh) 2008-04-09
CA2602224A1 (en) 2006-09-28
MX2007011455A (es) 2007-12-06
US20090209610A1 (en) 2009-08-20
RU2007138924A (ru) 2009-04-27
JP5009280B2 (ja) 2012-08-22
ES2367274T3 (es) 2011-11-02
PT1861404E (pt) 2011-09-01
EP1861404A1 (en) 2007-12-05
AU2006226625B2 (en) 2011-04-21
EP1861404B1 (en) 2011-05-18
CN101160311B (zh) 2010-11-24
PL1861404T3 (pl) 2011-12-30
US8034837B2 (en) 2011-10-11
ATE509932T1 (de) 2011-06-15
WO2006100019A1 (en) 2006-09-28
DE102005012971A1 (de) 2006-09-28

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