SI1244643T1 - Tryptase inhibitors - Google Patents
Tryptase inhibitorsInfo
- Publication number
- SI1244643T1 SI1244643T1 SI200030477T SI200030477T SI1244643T1 SI 1244643 T1 SI1244643 T1 SI 1244643T1 SI 200030477 T SI200030477 T SI 200030477T SI 200030477 T SI200030477 T SI 200030477T SI 1244643 T1 SI1244643 T1 SI 1244643T1
- Authority
- SI
- Slovenia
- Prior art keywords
- tryptase inhibitors
- inhibitors
- tryptase
- compounds
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
- C07D295/205—Radicals derived from carbonic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Neurosurgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Neurology (AREA)
- Dermatology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Ophthalmology & Optometry (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP99125384 | 1999-12-20 | ||
EP00985174A EP1244643B1 (fr) | 1999-12-20 | 2000-12-16 | Inhibiteurs de tryptase |
PCT/EP2000/012838 WO2001046168A1 (fr) | 1999-12-20 | 2000-12-16 | Inhibiteurs de tryptase |
Publications (1)
Publication Number | Publication Date |
---|---|
SI1244643T1 true SI1244643T1 (en) | 2004-12-31 |
Family
ID=8239661
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SI200030477T SI1244643T1 (en) | 1999-12-20 | 2000-12-16 | Tryptase inhibitors |
Country Status (13)
Country | Link |
---|---|
US (1) | US7015325B2 (fr) |
EP (1) | EP1244643B1 (fr) |
JP (1) | JP2003518109A (fr) |
AT (1) | ATE269313T1 (fr) |
AU (1) | AU783217B2 (fr) |
CA (1) | CA2392121A1 (fr) |
DE (1) | DE60011677T2 (fr) |
DK (1) | DK1244643T3 (fr) |
ES (1) | ES2222259T3 (fr) |
PT (1) | PT1244643E (fr) |
SI (1) | SI1244643T1 (fr) |
TR (1) | TR200402322T4 (fr) |
WO (1) | WO2001046168A1 (fr) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2438594A1 (fr) | 2001-01-31 | 2002-08-08 | Altana Pharma Ag | Derives de diazocine et leur utilisation en tant qu'inhibiteurs de tryptase |
CA2438685A1 (fr) | 2001-02-21 | 2002-08-29 | Altana Pharma Ag | Inhibiteurs de tryptase |
WO2002066420A2 (fr) | 2001-02-21 | 2002-08-29 | Altana Pharma Ag | Inhibiteurs de la tryptase |
EP1370518A2 (fr) * | 2001-03-15 | 2003-12-17 | ALTANA Pharma AG | Inhibiteurs de la tryptase |
WO2002074732A2 (fr) * | 2001-03-15 | 2002-09-26 | Altana Pharma Ag | Inhibiteurs de la tryptase |
ATE348803T1 (de) | 2001-06-19 | 2007-01-15 | Altana Pharma Ag | Tryptase-inhibitoren |
GB0507577D0 (en) * | 2005-04-14 | 2005-05-18 | Novartis Ag | Organic compounds |
IL302144A (en) * | 2017-03-29 | 2023-06-01 | Minerva Biotechnologies Corp | Agents for stem cell differentiation and cancer treatment |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3999946A (en) * | 1976-02-23 | 1976-12-28 | Allied Chemical Corporation | Time-temperature history indicators |
US4228126A (en) * | 1977-11-25 | 1980-10-14 | Allied Chemical Corporation | Diacetylene time-temperature indicators |
JPH10501238A (ja) * | 1994-06-01 | 1998-02-03 | アリス ファーマシューティカル コーポレイション | 肥満細胞媒介症状を治療するための組成物及び方法 |
EP0782571A1 (fr) * | 1994-09-23 | 1997-07-09 | Arris Pharmaceutical Corporation | Compositions et procedes de traitement de maladies inflammatoires provoquees par les mastocytes |
KR20000029679A (ko) * | 1996-07-30 | 2000-05-25 | 헤이즈 더블유.그쉬웬드 다니엘 에이치.페트리 | 트립타아제활성관련질병을치료하기위한화합물및조성물 |
US6221914B1 (en) * | 1997-11-10 | 2001-04-24 | Array Biopharma Inc. | Sulfonamide bridging compounds that inhibit tryptase activity |
JP2002502850A (ja) | 1998-02-06 | 2002-01-29 | マックス−プランク−ゲゼルシャフト・ツア・フェルデルング・デア・ヴィッセンシャフテン・エー・ファオ | トリプターゼ阻害物質 |
AU2723099A (en) | 1998-02-06 | 1999-08-23 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Tryptase inhibitors |
WO2000014097A2 (fr) | 1998-09-04 | 2000-03-16 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Nouvelles pyranoses |
US6673786B1 (en) | 1999-08-10 | 2004-01-06 | Altana Pharma Ag | Tryptase inhibitors |
JP2003509417A (ja) | 1999-09-14 | 2003-03-11 | アルタナ ファルマ アクチエンゲゼルシャフト | トリプターゼインヒビター |
-
2000
- 2000-12-16 US US10/149,288 patent/US7015325B2/en not_active Expired - Fee Related
- 2000-12-16 JP JP2001547079A patent/JP2003518109A/ja not_active Withdrawn
- 2000-12-16 PT PT00985174T patent/PT1244643E/pt unknown
- 2000-12-16 ES ES00985174T patent/ES2222259T3/es not_active Expired - Lifetime
- 2000-12-16 EP EP00985174A patent/EP1244643B1/fr not_active Expired - Lifetime
- 2000-12-16 WO PCT/EP2000/012838 patent/WO2001046168A1/fr active IP Right Grant
- 2000-12-16 AT AT00985174T patent/ATE269313T1/de not_active IP Right Cessation
- 2000-12-16 DK DK00985174T patent/DK1244643T3/da active
- 2000-12-16 CA CA002392121A patent/CA2392121A1/fr not_active Abandoned
- 2000-12-16 DE DE60011677T patent/DE60011677T2/de not_active Expired - Fee Related
- 2000-12-16 TR TR2004/02322T patent/TR200402322T4/xx unknown
- 2000-12-16 SI SI200030477T patent/SI1244643T1/xx unknown
- 2000-12-16 AU AU21669/01A patent/AU783217B2/en not_active Ceased
Also Published As
Publication number | Publication date |
---|---|
AU2166901A (en) | 2001-07-03 |
WO2001046168A1 (fr) | 2001-06-28 |
DE60011677D1 (en) | 2004-07-22 |
AU783217B2 (en) | 2005-10-06 |
ATE269313T1 (de) | 2004-07-15 |
PT1244643E (pt) | 2004-10-29 |
DK1244643T3 (da) | 2004-10-18 |
DE60011677T2 (de) | 2005-07-14 |
US20030083344A1 (en) | 2003-05-01 |
TR200402322T4 (tr) | 2004-12-21 |
US7015325B2 (en) | 2006-03-21 |
JP2003518109A (ja) | 2003-06-03 |
ES2222259T3 (es) | 2005-02-01 |
EP1244643A1 (fr) | 2002-10-02 |
CA2392121A1 (fr) | 2001-06-28 |
EP1244643B1 (fr) | 2004-06-16 |
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