SG52464A1 - A novel compound form - Google Patents

A novel compound form

Info

Publication number
SG52464A1
SG52464A1 SG1996004887A SG1996004887A SG52464A1 SG 52464 A1 SG52464 A1 SG 52464A1 SG 1996004887 A SG1996004887 A SG 1996004887A SG 1996004887 A SG1996004887 A SG 1996004887A SG 52464 A1 SG52464 A1 SG 52464A1
Authority
SG
Singapore
Prior art keywords
novel compound
compound form
crystallinity
manufacture
useful
Prior art date
Application number
SG1996004887A
Other languages
English (en)
Inventor
Lars Ake Kallstrom
Monica Annelie Nygren
Original Assignee
Astra Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20390588&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG52464(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astra Ab filed Critical Astra Ab
Publication of SG52464A1 publication Critical patent/SG52464A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Conductive Materials (AREA)
  • Contacts (AREA)
  • Electroplating Methods And Accessories (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Fats And Perfumes (AREA)
  • Medicinal Preparation (AREA)
  • Glass Compositions (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Powder Metallurgy (AREA)
SG1996004887A 1993-07-09 1994-07-08 A novel compound form SG52464A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE19939302396A SE9302396D0 (sv) 1993-07-09 1993-07-09 A novel compound form

Publications (1)

Publication Number Publication Date
SG52464A1 true SG52464A1 (en) 1998-09-28

Family

ID=20390588

Family Applications (1)

Application Number Title Priority Date Filing Date
SG1996004887A SG52464A1 (en) 1993-07-09 1994-07-08 A novel compound form

Country Status (42)

Country Link
US (1) US5900424A (xx)
EP (2) EP0707580B1 (xx)
JP (2) JP3635432B2 (xx)
KR (1) KR100353783B1 (xx)
CN (1) CN1064680C (xx)
AT (1) ATE212628T1 (xx)
AU (1) AU679766B2 (xx)
BR (1) BR9406940A (xx)
CA (1) CA2166794C (xx)
CZ (1) CZ288933B6 (xx)
DE (2) DE707580T1 (xx)
DK (1) DK0707580T3 (xx)
DZ (1) DZ1792A1 (xx)
EE (1) EE03127B1 (xx)
EG (1) EG21437A (xx)
ES (1) ES2100136T3 (xx)
FI (1) FI114154B (xx)
GR (1) GR970300015T1 (xx)
HK (1) HK1008329A1 (xx)
HR (1) HRP940385B1 (xx)
HU (1) HU226861B1 (xx)
IL (1) IL110190A (xx)
IS (1) IS2075B (xx)
MA (1) MA23257A1 (xx)
MX (1) MX9405217A (xx)
MY (1) MY113274A (xx)
NO (1) NO308702B1 (xx)
NZ (1) NZ268693A (xx)
PL (1) PL175999B1 (xx)
PT (1) PT707580E (xx)
RU (1) RU2139868C1 (xx)
SA (1) SA94150058B1 (xx)
SE (1) SE9302396D0 (xx)
SG (1) SG52464A1 (xx)
SI (1) SI0707580T1 (xx)
SK (1) SK281230B6 (xx)
TN (1) TNSN94079A1 (xx)
TW (1) TW504509B (xx)
UA (1) UA43343C2 (xx)
WO (1) WO1995001977A1 (xx)
YU (1) YU49193B (xx)
ZA (1) ZA944933B (xx)

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SE9302395D0 (sv) * 1993-07-09 1993-07-09 Ab Astra New pharmaceutical formulation
SE9302396D0 (sv) * 1993-07-09 1993-07-09 Ab Astra A novel compound form
EP0723436B1 (en) * 1994-07-08 2001-09-26 AstraZeneca AB Multiple unit tableted dosage form i
HUT78132A (hu) * 1994-07-08 2000-06-28 Astra Aktiebolag Omeprazol magnéziumsóját tartalmazó új orális gyógyszerforma
SE9500478D0 (sv) * 1995-02-09 1995-02-09 Astra Ab New pharmaceutical formulation and process
US5840737A (en) 1996-01-04 1998-11-24 The Curators Of The University Of Missouri Omeprazole solution and method for using same
US6489346B1 (en) 1996-01-04 2002-12-03 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
US6645988B2 (en) * 1996-01-04 2003-11-11 Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
US6699885B2 (en) 1996-01-04 2004-03-02 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and methods of using same
SE9600070D0 (sv) 1996-01-08 1996-01-08 Astra Ab New oral pharmaceutical dosage forms
SE508669C2 (sv) * 1996-04-26 1998-10-26 Astra Ab Nytt förfarande
US6623759B2 (en) * 1996-06-28 2003-09-23 Astrazeneca Ab Stable drug form for oral administration with benzimidazole derivatives as active ingredient and process for the preparation thereof
TW385306B (en) * 1996-11-14 2000-03-21 Takeda Chemical Industries Ltd Method for producing crystals of benzimidazole derivatives
SE510666C2 (sv) * 1996-12-20 1999-06-14 Astra Ab Nya Kristallmodifikationer
SE9702000D0 (sv) * 1997-05-28 1997-05-28 Astra Ab New pharmaceutical formulation
SE510650C2 (sv) 1997-05-30 1999-06-14 Astra Ab Ny förening
US6747155B2 (en) 1997-05-30 2004-06-08 Astrazeneca Ab Process
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US6096340A (en) * 1997-11-14 2000-08-01 Andrx Pharmaceuticals, Inc. Omeprazole formulation
SE9704870D0 (sv) 1997-12-22 1997-12-22 Astra Ab New pharmaceutical formulation I
FR2774288B1 (fr) * 1998-01-30 2001-09-07 Ethypharm Sa Microgranules d'omeprazole gastroproteges, procede d'obtention et preparations pharmaceutiques
US6048981A (en) * 1998-04-22 2000-04-11 Torcan Chemical Ltd. Magnesium omeprazole and process for its preparation
DE19843413C1 (de) 1998-08-18 2000-03-30 Byk Gulden Lomberg Chem Fab Neue Salzform von Pantoprazol
US6733778B1 (en) 1999-08-27 2004-05-11 Andrx Pharmaceuticals, Inc. Omeprazole formulation
SE9803772D0 (sv) 1998-11-05 1998-11-05 Astra Ab Pharmaceutical formulation
UA72748C2 (en) 1998-11-10 2005-04-15 Astrazeneca Ab A novel crystalline form of omeprazole
IL142703A (en) * 1998-11-10 2006-04-10 Astrazeneca Ab Crystalline form of omeprazole
IL142629A0 (en) * 1998-11-18 2002-03-10 Astra Ab Improved chemical process and pharmaceutical formulation
TWI243672B (en) 1999-06-01 2005-11-21 Astrazeneca Ab New use of compounds as antibacterial agents
US6316020B1 (en) * 1999-08-26 2001-11-13 Robert R. Whittle Pharmaceutical formulations
CA2290893C (en) * 1999-11-16 2007-05-01 Bernard Charles Sherman Magnesium omeprazole
SE0000774D0 (sv) 2000-03-08 2000-03-08 Astrazeneca Ab New formulation
US20030212274A1 (en) * 2000-05-15 2003-11-13 Bakthavathsalan Vijayaraghavan Novel amorphous form of omeprazole salts
CA2386716C (en) * 2002-05-17 2012-07-24 Bernard Charles Sherman Magnesium salt of s-omeprazole
CA2775616C (en) 2000-08-04 2013-09-17 Takeda Pharmaceutical Company Limited Salts of benzimidazole compound and application thereof
US6544556B1 (en) 2000-09-11 2003-04-08 Andrx Corporation Pharmaceutical formulations containing a non-steroidal antiinflammatory drug and a proton pump inhibitor
US20020064555A1 (en) * 2000-09-29 2002-05-30 Dan Cullen Proton pump inhibitor formulation
SE0101379D0 (sv) 2001-04-18 2001-04-18 Diabact Ab Komposition som hämmar utsöndring av magsyra
US8206741B2 (en) 2001-06-01 2012-06-26 Pozen Inc. Pharmaceutical compositions for the coordinated delivery of NSAIDs
SE0102993D0 (sv) 2001-09-07 2001-09-07 Astrazeneca Ab New self emulsifying drug delivery system
MXPA04007169A (es) * 2002-01-25 2004-10-29 Santarus Inc Suministro transmucosal de inhibidores de bomba de protones.
FR2836228B1 (fr) * 2002-02-21 2005-08-19 Inst Francais Du Petrole Methode et dispositif pour evaluer des parametres physiques d'un gisement souterrain a partir de debris de roche qui y sont preleves
US20030228363A1 (en) * 2002-06-07 2003-12-11 Patel Mahendra R. Stabilized pharmaceutical compositons containing benzimidazole compounds
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US20060024362A1 (en) * 2004-07-29 2006-02-02 Pawan Seth Composition comprising a benzimidazole and process for its manufacture
US8541026B2 (en) 2004-09-24 2013-09-24 Abbvie Inc. Sustained release formulations of opioid and nonopioid analgesics
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US20060160783A1 (en) * 2004-12-30 2006-07-20 Transform Pharmaceuticals, Inc. Novel omeprazole forms and related methods
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US7981908B2 (en) 2005-05-11 2011-07-19 Vecta, Ltd. Compositions and methods for inhibiting gastric acid secretion
US7803817B2 (en) 2005-05-11 2010-09-28 Vecta, Ltd. Composition and methods for inhibiting gastric acid secretion
CA2624179A1 (en) * 2005-10-06 2007-04-12 Auspex Pharmaceuticals, Inc. Deuterated inhibitors of gastric h+, k+-atpase with enhanced therapeutic properties
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US7553857B2 (en) 2005-12-23 2009-06-30 Lek Pharmaceuticals D.D. S-omeprazole magnesium
AU2007266574A1 (en) * 2006-06-01 2007-12-06 Dexcel Pharma Technologies Ltd. Multiple unit pharmaceutical formulation
RU2467747C2 (ru) 2006-07-25 2012-11-27 Векта Лтд. Композиции и способы для ингибирования секреции желудочной кислоты с использованием производных малых дикарбоновых кислот в сочетании с ppi
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EP2486910A3 (en) 2006-10-27 2012-08-22 The Curators Of The University Of Missouri Multi-chambered apparatus comprising a dispenser head
EP1947099A1 (en) 2007-01-18 2008-07-23 LEK Pharmaceuticals D.D. Process for solvent removal from omeprazole salts
US8911787B2 (en) 2008-02-26 2014-12-16 Ranbaxy Laboratories Limited Stable oral benzimidazole compositions and process of preparation thereof
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CN102993184A (zh) * 2013-01-08 2013-03-27 湖南方盛制药股份有限公司 一种埃索美拉唑及其镁盐三水合物的制备方法
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US10736855B2 (en) 2016-02-25 2020-08-11 Dexcel Pharma Technologies Ltd. Compositions comprising proton pump inhibitors
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WO2024075017A1 (en) 2022-10-04 2024-04-11 Zabirnyk Arsenii Inhibition of aortic valve calcification

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE7804231L (sv) * 1978-04-14 1979-10-15 Haessle Ab Magsyrasekretionsmedel
SE8301182D0 (sv) * 1983-03-04 1983-03-04 Haessle Ab Novel compounds
GB2189698A (en) * 1986-04-30 1987-11-04 Haessle Ab Coated omeprazole tablets
DE4035455A1 (de) * 1990-11-08 1992-05-14 Byk Gulden Lomberg Chem Fab Enantiomerentrennung
SE9302396D0 (sv) * 1993-07-09 1993-07-09 Ab Astra A novel compound form

Also Published As

Publication number Publication date
ES2100136T3 (es) 2002-09-01
HUT75314A (en) 1997-05-28
GR970300015T1 (en) 1997-05-31
DE69429774D1 (de) 2002-03-14
EE03127B1 (et) 1998-10-15
ATE212628T1 (de) 2002-02-15
SK2296A3 (en) 1996-10-02
SK281230B6 (sk) 2001-01-18
EP1164132A2 (en) 2001-12-19
HU226861B1 (en) 2009-12-28
DK0707580T3 (da) 2002-04-15
MX9405217A (es) 1995-01-31
HU9503873D0 (en) 1996-02-28
IS4186A (is) 1995-01-10
ES2100136T1 (es) 1997-06-16
FI960101A0 (fi) 1996-01-09
IL110190A0 (en) 1994-10-21
ZA944933B (en) 1995-02-20
HRP940385A2 (en) 1997-02-28
SI0707580T1 (en) 2002-06-30
CZ288933B6 (cs) 2001-09-12
NZ268693A (en) 1997-05-26
WO1995001977A1 (en) 1995-01-19
PL312440A1 (en) 1996-04-29
SA94150058B1 (ar) 2006-06-20
NO960068L (no) 1996-01-05
AU679766B2 (en) 1997-07-10
CZ6996A3 (en) 1996-05-15
FI960101A (fi) 1996-01-09
HRP940385B1 (en) 2003-06-30
TNSN94079A1 (fr) 1995-04-25
EP1164132A3 (en) 2002-01-02
JP2002105072A (ja) 2002-04-10
CN1126993A (zh) 1996-07-17
UA43343C2 (uk) 2001-12-17
NO960068D0 (no) 1996-01-05
BR9406940A (pt) 1996-09-10
CN1064680C (zh) 2001-04-18
FI114154B (fi) 2004-08-31
DE69429774T2 (de) 2002-11-14
HK1008329A1 (en) 1999-05-07
YU49193B (sh) 2004-09-03
KR100353783B1 (ko) 2004-04-03
US5900424A (en) 1999-05-04
IL110190A (en) 2000-07-26
PL175999B1 (pl) 1999-03-31
DZ1792A1 (fr) 2002-02-17
DE707580T1 (de) 1997-09-04
IS2075B (is) 2005-12-15
EG21437A (en) 2001-10-31
EP0707580A1 (en) 1996-04-24
YU43694A (sh) 1997-07-31
MY113274A (en) 2002-01-31
TW504509B (en) 2002-10-01
JPH08512315A (ja) 1996-12-24
PT707580E (pt) 2002-06-28
MA23257A1 (fr) 1995-04-01
NO308702B1 (no) 2000-10-16
RU2139868C1 (ru) 1999-10-20
AU7198194A (en) 1995-02-06
EP0707580B1 (en) 2002-01-30
JP3878826B2 (ja) 2007-02-07
JP3635432B2 (ja) 2005-04-06
SE9302396D0 (sv) 1993-07-09
CA2166794C (en) 1997-03-04

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