DE707580T1 - Magnesium-omeprazol - Google Patents

Magnesium-omeprazol

Info

Publication number
DE707580T1
DE707580T1 DE0707580T DE94921154T DE707580T1 DE 707580 T1 DE707580 T1 DE 707580T1 DE 0707580 T DE0707580 T DE 0707580T DE 94921154 T DE94921154 T DE 94921154T DE 707580 T1 DE707580 T1 DE 707580T1
Authority
DE
Germany
Prior art keywords
magnesium
omeprazol
crystallinity
manufacture
useful
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE0707580T
Other languages
English (en)
Inventor
Lars Kaellstroem
Monica Nygren
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AstraZeneca AB
Original Assignee
Astra AB
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20390588&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE707580(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astra AB filed Critical Astra AB
Publication of DE707580T1 publication Critical patent/DE707580T1/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
DE0707580T 1993-07-09 1994-07-08 Magnesium-omeprazol Pending DE707580T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE19939302396A SE9302396D0 (sv) 1993-07-09 1993-07-09 A novel compound form
PCT/SE1994/000680 WO1995001977A1 (en) 1993-07-09 1994-07-08 Magnesium omeprazole

Publications (1)

Publication Number Publication Date
DE707580T1 true DE707580T1 (de) 1997-09-04

Family

ID=20390588

Family Applications (2)

Application Number Title Priority Date Filing Date
DE69429774T Expired - Lifetime DE69429774T2 (de) 1993-07-09 1994-07-08 Magnesium-omeprazol
DE0707580T Pending DE707580T1 (de) 1993-07-09 1994-07-08 Magnesium-omeprazol

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DE69429774T Expired - Lifetime DE69429774T2 (de) 1993-07-09 1994-07-08 Magnesium-omeprazol

Country Status (42)

Country Link
US (1) US5900424A (de)
EP (2) EP1164132A3 (de)
JP (2) JP3635432B2 (de)
KR (1) KR100353783B1 (de)
CN (1) CN1064680C (de)
AT (1) ATE212628T1 (de)
AU (1) AU679766B2 (de)
BR (1) BR9406940A (de)
CA (1) CA2166794C (de)
CZ (1) CZ288933B6 (de)
DE (2) DE69429774T2 (de)
DK (1) DK0707580T3 (de)
DZ (1) DZ1792A1 (de)
EE (1) EE03127B1 (de)
EG (1) EG21437A (de)
ES (1) ES2100136T3 (de)
FI (1) FI114154B (de)
GR (1) GR970300015T1 (de)
HK (1) HK1008329A1 (de)
HR (1) HRP940385B1 (de)
HU (1) HU226861B1 (de)
IL (1) IL110190A (de)
IS (1) IS2075B (de)
MA (1) MA23257A1 (de)
MX (1) MX9405217A (de)
MY (1) MY113274A (de)
NO (1) NO308702B1 (de)
NZ (1) NZ268693A (de)
PL (1) PL175999B1 (de)
PT (1) PT707580E (de)
RU (1) RU2139868C1 (de)
SA (1) SA94150058B1 (de)
SE (1) SE9302396D0 (de)
SG (1) SG52464A1 (de)
SI (1) SI0707580T1 (de)
SK (1) SK281230B6 (de)
TN (1) TNSN94079A1 (de)
TW (1) TW504509B (de)
UA (1) UA43343C2 (de)
WO (1) WO1995001977A1 (de)
YU (1) YU49193B (de)
ZA (1) ZA944933B (de)

Families Citing this family (92)

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EE03305B1 (et) 1994-07-08 2000-12-15 Astra Aktiebolag Paljuosaline tableteeritud annusvorm I
BR9508261A (pt) * 1994-07-08 1997-12-23 Astra Ab Formulação oral entericamente revestida uso da mesma processo para preparer a formulação inibir a secreção de ácido gástrico em mamíferos e no ser humano e tratar doenças relacionadas ao ácido gástrico em maníferos e no ser humano e pacote de empola de pressão transversal
SE9500478D0 (sv) * 1995-02-09 1995-02-09 Astra Ab New pharmaceutical formulation and process
US6699885B2 (en) 1996-01-04 2004-03-02 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and methods of using same
US6489346B1 (en) 1996-01-04 2002-12-03 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
US6645988B2 (en) 1996-01-04 2003-11-11 Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
US5840737A (en) 1996-01-04 1998-11-24 The Curators Of The University Of Missouri Omeprazole solution and method for using same
SE9600070D0 (sv) 1996-01-08 1996-01-08 Astra Ab New oral pharmaceutical dosage forms
SE508669C2 (sv) * 1996-04-26 1998-10-26 Astra Ab Nytt förfarande
US6623759B2 (en) 1996-06-28 2003-09-23 Astrazeneca Ab Stable drug form for oral administration with benzimidazole derivatives as active ingredient and process for the preparation thereof
TW385306B (en) * 1996-11-14 2000-03-21 Takeda Chemical Industries Ltd Method for producing crystals of benzimidazole derivatives
SE510666C2 (sv) * 1996-12-20 1999-06-14 Astra Ab Nya Kristallmodifikationer
SE9702000D0 (sv) * 1997-05-28 1997-05-28 Astra Ab New pharmaceutical formulation
SE510650C2 (sv) * 1997-05-30 1999-06-14 Astra Ab Ny förening
US6747155B2 (en) 1997-05-30 2004-06-08 Astrazeneca Ab Process
US6096340A (en) * 1997-11-14 2000-08-01 Andrx Pharmaceuticals, Inc. Omeprazole formulation
US6174548B1 (en) 1998-08-28 2001-01-16 Andrx Pharmaceuticals, Inc. Omeprazole formulation
SE9704870D0 (sv) 1997-12-22 1997-12-22 Astra Ab New pharmaceutical formulation I
FR2774288B1 (fr) * 1998-01-30 2001-09-07 Ethypharm Sa Microgranules d'omeprazole gastroproteges, procede d'obtention et preparations pharmaceutiques
US6048981A (en) * 1998-04-22 2000-04-11 Torcan Chemical Ltd. Magnesium omeprazole and process for its preparation
DE19843413C1 (de) 1998-08-18 2000-03-30 Byk Gulden Lomberg Chem Fab Neue Salzform von Pantoprazol
US6733778B1 (en) 1999-08-27 2004-05-11 Andrx Pharmaceuticals, Inc. Omeprazole formulation
SE9803772D0 (sv) 1998-11-05 1998-11-05 Astra Ab Pharmaceutical formulation
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UA72748C2 (en) * 1998-11-10 2005-04-15 Astrazeneca Ab A novel crystalline form of omeprazole
CN100503598C (zh) * 1998-11-18 2009-06-24 阿斯特拉曾尼卡有限公司 改进的化学方法和药物制剂
TWI243672B (en) 1999-06-01 2005-11-21 Astrazeneca Ab New use of compounds as antibacterial agents
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SE0000774D0 (sv) 2000-03-08 2000-03-08 Astrazeneca Ab New formulation
US20030212274A1 (en) * 2000-05-15 2003-11-13 Bakthavathsalan Vijayaraghavan Novel amorphous form of omeprazole salts
WO2002012225A1 (fr) 2000-08-04 2002-02-14 Takeda Chemical Industries, Ltd. Sels de composé à base de benzimidazole et leurs applications
CA2386716C (en) * 2002-05-17 2012-07-24 Bernard Charles Sherman Magnesium salt of s-omeprazole
US6544556B1 (en) 2000-09-11 2003-04-08 Andrx Corporation Pharmaceutical formulations containing a non-steroidal antiinflammatory drug and a proton pump inhibitor
WO2002026210A2 (en) * 2000-09-29 2002-04-04 Geneva Pharmaceuticals Inc. Proton pump inhibitor formulation
SE0101379D0 (sv) 2001-04-18 2001-04-18 Diabact Ab Komposition som hämmar utsöndring av magsyra
US8206741B2 (en) 2001-06-01 2012-06-26 Pozen Inc. Pharmaceutical compositions for the coordinated delivery of NSAIDs
SE0102993D0 (sv) 2001-09-07 2001-09-07 Astrazeneca Ab New self emulsifying drug delivery system
MXPA04007169A (es) * 2002-01-25 2004-10-29 Santarus Inc Suministro transmucosal de inhibidores de bomba de protones.
FR2836228B1 (fr) * 2002-02-21 2005-08-19 Inst Francais Du Petrole Methode et dispositif pour evaluer des parametres physiques d'un gisement souterrain a partir de debris de roche qui y sont preleves
US20030228363A1 (en) * 2002-06-07 2003-12-11 Patel Mahendra R. Stabilized pharmaceutical compositons containing benzimidazole compounds
SE0203065D0 (sv) 2002-10-16 2002-10-16 Diabact Ab Gastric acid secretion inhibiting composition
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EP1633736A1 (de) * 2003-05-05 2006-03-15 Ranbaxy Laboratories Limited Barium salz eines benzimidazol-derivats
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US20060024362A1 (en) * 2004-07-29 2006-02-02 Pawan Seth Composition comprising a benzimidazole and process for its manufacture
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US7981908B2 (en) 2005-05-11 2011-07-19 Vecta, Ltd. Compositions and methods for inhibiting gastric acid secretion
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CA2624179A1 (en) * 2005-10-06 2007-04-12 Auspex Pharmaceuticals, Inc. Deuterated inhibitors of gastric h+, k+-atpase with enhanced therapeutic properties
EP1801110A1 (de) 2005-12-22 2007-06-27 KRKA, tovarna zdravil, d.d., Novo mesto Argininsalz des Esomeprazols
US7553857B2 (en) 2005-12-23 2009-06-30 Lek Pharmaceuticals D.D. S-omeprazole magnesium
US20100297226A1 (en) * 2006-06-01 2010-11-25 Dexcel Pharma Technologies Ltd. Multiple unit pharmaceutical formulation
ES2511792T3 (es) 2006-07-25 2014-10-23 Vecta Ltd. Composiciones y métodos para la inhibición de la secreción de ácido gástrico usando derivados de pequeños ácidos dicarboxílicos en combinación con IBP
US20090092658A1 (en) * 2007-10-05 2009-04-09 Santarus, Inc. Novel formulations of proton pump inhibitors and methods of using these formulations
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US8911787B2 (en) 2008-02-26 2014-12-16 Ranbaxy Laboratories Limited Stable oral benzimidazole compositions and process of preparation thereof
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Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE7804231L (sv) * 1978-04-14 1979-10-15 Haessle Ab Magsyrasekretionsmedel
SE8301182D0 (sv) * 1983-03-04 1983-03-04 Haessle Ab Novel compounds
GB2189698A (en) * 1986-04-30 1987-11-04 Haessle Ab Coated omeprazole tablets
DE4035455A1 (de) * 1990-11-08 1992-05-14 Byk Gulden Lomberg Chem Fab Enantiomerentrennung
SE9302396D0 (sv) * 1993-07-09 1993-07-09 Ab Astra A novel compound form

Also Published As

Publication number Publication date
EP0707580A1 (de) 1996-04-24
HK1008329A1 (en) 1999-05-07
HU9503873D0 (en) 1996-02-28
HUT75314A (en) 1997-05-28
YU43694A (sh) 1997-07-31
UA43343C2 (uk) 2001-12-17
RU2139868C1 (ru) 1999-10-20
JP2002105072A (ja) 2002-04-10
HRP940385A2 (en) 1997-02-28
SK2296A3 (en) 1996-10-02
SK281230B6 (sk) 2001-01-18
WO1995001977A1 (en) 1995-01-19
ATE212628T1 (de) 2002-02-15
CA2166794C (en) 1997-03-04
IL110190A0 (en) 1994-10-21
NO960068L (no) 1996-01-05
CZ288933B6 (cs) 2001-09-12
HU226861B1 (en) 2009-12-28
IS2075B (is) 2005-12-15
PL312440A1 (en) 1996-04-29
DK0707580T3 (da) 2002-04-15
SI0707580T1 (en) 2002-06-30
EP1164132A2 (de) 2001-12-19
JPH08512315A (ja) 1996-12-24
MA23257A1 (fr) 1995-04-01
NZ268693A (en) 1997-05-26
MY113274A (en) 2002-01-31
HRP940385B1 (en) 2003-06-30
FI114154B (fi) 2004-08-31
SG52464A1 (en) 1998-09-28
IL110190A (en) 2000-07-26
JP3878826B2 (ja) 2007-02-07
EP1164132A3 (de) 2002-01-02
YU49193B (sh) 2004-09-03
CN1126993A (zh) 1996-07-17
BR9406940A (pt) 1996-09-10
NO308702B1 (no) 2000-10-16
JP3635432B2 (ja) 2005-04-06
US5900424A (en) 1999-05-04
FI960101A0 (fi) 1996-01-09
EG21437A (en) 2001-10-31
KR100353783B1 (ko) 2004-04-03
NO960068D0 (no) 1996-01-05
TNSN94079A1 (fr) 1995-04-25
EE03127B1 (et) 1998-10-15
ES2100136T1 (es) 1997-06-16
PL175999B1 (pl) 1999-03-31
IS4186A (is) 1995-01-10
MX9405217A (es) 1995-01-31
ZA944933B (en) 1995-02-20
FI960101A (fi) 1996-01-09
SE9302396D0 (sv) 1993-07-09
CN1064680C (zh) 2001-04-18
TW504509B (en) 2002-10-01
ES2100136T3 (es) 2002-09-01
DE69429774D1 (de) 2002-03-14
EP0707580B1 (de) 2002-01-30
CZ6996A3 (en) 1996-05-15
SA94150058B1 (ar) 2006-06-20
PT707580E (pt) 2002-06-28
AU7198194A (en) 1995-02-06
DE69429774T2 (de) 2002-11-14
GR970300015T1 (en) 1997-05-31
DZ1792A1 (fr) 2002-02-17
AU679766B2 (en) 1997-07-10

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