SG11201610132RA - Aminoester derivatives - Google Patents

Aminoester derivatives

Info

Publication number
SG11201610132RA
SG11201610132RA SG11201610132RA SG11201610132RA SG11201610132RA SG 11201610132R A SG11201610132R A SG 11201610132RA SG 11201610132R A SG11201610132R A SG 11201610132RA SG 11201610132R A SG11201610132R A SG 11201610132RA SG 11201610132R A SG11201610132R A SG 11201610132RA
Authority
SG
Singapore
Prior art keywords
aminoester derivatives
aminoester
derivatives
Prior art date
Application number
SG11201610132RA
Other languages
English (en)
Inventor
Elisabetta Armani
Gabriele Amari
Carmelida Capaldi
Wesley Blackaby
Ian Linney
De Pöel Hervé Van
Charles Baker-Glenn
Naimisha Trivedi
Original Assignee
Chiesi Farma Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chiesi Farma Spa filed Critical Chiesi Farma Spa
Publication of SG11201610132RA publication Critical patent/SG11201610132RA/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4436Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/04Drugs for disorders of the respiratory system for throat disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
SG11201610132RA 2014-06-05 2015-06-03 Aminoester derivatives SG11201610132RA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP14171266 2014-06-05
PCT/EP2015/062417 WO2015185649A1 (fr) 2014-06-05 2015-06-03 Dérivés aminoesters

Publications (1)

Publication Number Publication Date
SG11201610132RA true SG11201610132RA (en) 2017-01-27

Family

ID=50884281

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201610132RA SG11201610132RA (en) 2014-06-05 2015-06-03 Aminoester derivatives

Country Status (32)

Country Link
US (2) US9763924B2 (fr)
EP (1) EP3152201B1 (fr)
JP (1) JP2017516824A (fr)
KR (1) KR102420323B1 (fr)
CN (1) CN106459020B (fr)
AR (1) AR100732A1 (fr)
AU (1) AU2015270539B2 (fr)
BR (1) BR112016026725B1 (fr)
CA (1) CA2953198C (fr)
CL (1) CL2016003117A1 (fr)
CY (1) CY1120698T1 (fr)
DK (1) DK3152201T3 (fr)
EA (1) EA032761B1 (fr)
ES (1) ES2688826T3 (fr)
GE (1) GEP20186922B (fr)
HR (1) HRP20181967T1 (fr)
HU (1) HUE042119T2 (fr)
IL (1) IL249325B (fr)
LT (1) LT3152201T (fr)
MA (1) MA39947B1 (fr)
MX (1) MX2016015958A (fr)
PE (1) PE20161557A1 (fr)
PH (1) PH12016502221A1 (fr)
PL (1) PL3152201T3 (fr)
PT (1) PT3152201T (fr)
RS (1) RS57787B1 (fr)
SG (1) SG11201610132RA (fr)
SI (1) SI3152201T1 (fr)
TN (1) TN2016000546A1 (fr)
TW (1) TW201625600A (fr)
WO (1) WO2015185649A1 (fr)
ZA (1) ZA201608331B (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3292118A1 (fr) 2015-05-07 2018-03-14 Chiesi Farmaceutici S.p.A. Dérivés d'aminoesters
AR104822A1 (es) * 2015-06-01 2017-08-16 Chiesi Farm Spa Derivado de aminoésteres
AR104829A1 (es) * 2015-06-01 2017-08-16 Chiesi Farm Spa Derivados de aminoésteres
CN106866474B (zh) * 2017-02-16 2018-12-28 陕西师范大学 一种手性α-芳基甘氨酸酯衍生物的合成方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2022783A1 (fr) * 2007-08-08 2009-02-11 CHIESI FARMACEUTICI S.p.A. Dérivés d'alcools 1-phényl-2-pyridinylalkyliques en tant qu'inhibiteurs de la phosphodiestérase
AR070562A1 (es) 2008-02-06 2010-04-21 Glaxo Group Ltd Farmacoforos duales - antagonistas muscarinicos de pde4
EP2216327A1 (fr) * 2009-02-06 2010-08-11 CHIESI FARMACEUTICI S.p.A. Benzoate de (1-Phenyl-2-Pyridin-4-yl)ethyle en tant qu'inhibiteurs de phosphodiestérase
WO2014086855A1 (fr) 2012-12-05 2014-06-12 Chiesi Farmaceutici S.P.A. Dérivés de phényléthylpyridine en tant qu'inhibiteurs de pde4
AR093797A1 (es) 2012-12-05 2015-06-24 Chiesi Farm Spa Derivados de feniletilpiridina inhibidores de pde-4
WO2014086852A1 (fr) 2012-12-05 2014-06-12 Chiesi Farmaceutici S.P.A. Dérivés de phényléthylpyridine comme inhibiteurs de pde4
RU2016121854A (ru) 2013-12-05 2017-12-07 КЬЕЗИ ФАРМАЧЕУТИЧИ С.п.А. Производные гетероарила
CN105814034A (zh) 2013-12-05 2016-07-27 奇斯药制品公司 用于治疗呼吸病的二苯甲基衍生物

Also Published As

Publication number Publication date
CN106459020B (zh) 2019-06-18
PE20161557A1 (es) 2017-02-07
CA2953198A1 (fr) 2015-12-10
AU2015270539B2 (en) 2018-11-08
ES2688826T3 (es) 2018-11-07
US10117860B2 (en) 2018-11-06
CL2016003117A1 (es) 2017-06-23
AR100732A1 (es) 2016-10-26
US20170340616A1 (en) 2017-11-30
BR112016026725A8 (pt) 2021-06-29
GEP20186922B (en) 2018-11-12
CA2953198C (fr) 2023-06-13
JP2017516824A (ja) 2017-06-22
MX2016015958A (es) 2017-04-10
PT3152201T (pt) 2018-10-26
CN106459020A (zh) 2017-02-22
US20150352091A1 (en) 2015-12-10
CY1120698T1 (el) 2019-12-11
WO2015185649A1 (fr) 2015-12-10
TW201625600A (zh) 2016-07-16
PL3152201T3 (pl) 2019-02-28
TN2016000546A1 (en) 2018-04-04
BR112016026725A2 (pt) 2017-08-15
HUE042119T2 (hu) 2019-06-28
LT3152201T (lt) 2018-10-10
US9763924B2 (en) 2017-09-19
DK3152201T3 (en) 2018-11-19
HRP20181967T1 (hr) 2019-02-08
AU2015270539A1 (en) 2016-12-22
BR112016026725B1 (pt) 2024-02-27
IL249325B (en) 2018-12-31
ZA201608331B (en) 2018-05-30
KR20170015294A (ko) 2017-02-08
PH12016502221A1 (en) 2017-02-06
WO2015185649A9 (fr) 2017-01-05
RS57787B1 (sr) 2018-12-31
IL249325A0 (en) 2017-02-28
EA032761B1 (ru) 2019-07-31
EP3152201B1 (fr) 2018-08-29
EP3152201A1 (fr) 2017-04-12
MA39947A (fr) 2017-04-12
KR102420323B1 (ko) 2022-07-13
SI3152201T1 (sl) 2018-10-30
MA39947B1 (fr) 2018-10-31
EA201692227A1 (ru) 2017-05-31

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