SG11201604787SA - Solid forms of an alpha, omega di-substituted dihydroxy cyclopentyl compound and methods for the preparation and use thereof - Google Patents

Solid forms of an alpha, omega di-substituted dihydroxy cyclopentyl compound and methods for the preparation and use thereof

Info

Publication number
SG11201604787SA
SG11201604787SA SG11201604787SA SG11201604787SA SG11201604787SA SG 11201604787S A SG11201604787S A SG 11201604787SA SG 11201604787S A SG11201604787S A SG 11201604787SA SG 11201604787S A SG11201604787S A SG 11201604787SA SG 11201604787S A SG11201604787S A SG 11201604787SA
Authority
SG
Singapore
Prior art keywords
omega
alpha
preparation
methods
solid forms
Prior art date
Application number
SG11201604787SA
Other languages
English (en)
Inventor
Ke Wu
Gyorgy Ambrus
Original Assignee
Allergan Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Allergan Inc filed Critical Allergan Inc
Publication of SG11201604787SA publication Critical patent/SG11201604787SA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/557Eicosanoids, e.g. leukotrienes or prostaglandins
    • A61K31/559Eicosanoids, e.g. leukotrienes or prostaglandins having heterocyclic rings containing hetero atoms other than oxygen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/28Halogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SG11201604787SA 2013-12-13 2014-12-12 Solid forms of an alpha, omega di-substituted dihydroxy cyclopentyl compound and methods for the preparation and use thereof SG11201604787SA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361915575P 2013-12-13 2013-12-13
PCT/US2014/070156 WO2015089475A1 (en) 2013-12-13 2014-12-12 Solid forms of an alpha, omega di-substituted dihydroxy cyclopentyl compound and methods for the preparation and use thereof

Publications (1)

Publication Number Publication Date
SG11201604787SA true SG11201604787SA (en) 2016-07-28

Family

ID=52282957

Family Applications (2)

Application Number Title Priority Date Filing Date
SG10201709702UA SG10201709702UA (en) 2013-12-13 2014-12-12 Solid forms of an alpha, omega di-substituted dihydroxy cyclopentyl compound and methods for the preparation and use thereof
SG11201604787SA SG11201604787SA (en) 2013-12-13 2014-12-12 Solid forms of an alpha, omega di-substituted dihydroxy cyclopentyl compound and methods for the preparation and use thereof

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SG10201709702UA SG10201709702UA (en) 2013-12-13 2014-12-12 Solid forms of an alpha, omega di-substituted dihydroxy cyclopentyl compound and methods for the preparation and use thereof

Country Status (16)

Country Link
US (2) US9353079B2 (es)
EP (1) EP3080096A1 (es)
JP (2) JP2016539994A (es)
KR (1) KR20160097310A (es)
CN (1) CN105814033B (es)
AU (1) AU2014361794B2 (es)
BR (1) BR112016013594A8 (es)
CA (1) CA2933556A1 (es)
CL (2) CL2016001448A1 (es)
IL (2) IL245917B (es)
MX (1) MX2016007717A (es)
RU (1) RU2730520C2 (es)
SA (1) SA516371307B1 (es)
SG (2) SG10201709702UA (es)
UA (1) UA121108C2 (es)
WO (1) WO2015089475A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10206813B2 (en) 2009-05-18 2019-02-19 Dose Medical Corporation Implants with controlled drug delivery features and methods of using same
WO2019023211A1 (en) 2017-07-25 2019-01-31 Allergan, Inc. SOLID COMPLEX COMPRISING (Z) -7 - ((1R, 2R, 3R, 5S) -2 - ((S, E) -5- (2,5-DICHLOROTHIOPHEN-3-YL) -3-HYDROXYPENT-1 EN-1-YL) -3,5-DIHYDROXYCYCLOPENTYL) HEPT-5-ENAMIDE, PREPARATION THEREOF AND USES THEREOF

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO143741C (no) * 1972-07-13 1981-04-08 Pfizer Analogifremgangsmaate for fremstilling av fysiologisk aktive prostaglandinforbindelser av e- og f-serien
US5296504A (en) * 1988-09-06 1994-03-22 Kabi Pharmacia Prostaglandin derivatives for the treatment of glaucoma or ocular hypertension
US6602900B2 (en) 1992-09-21 2003-08-05 Allergan, Inc. Cyclopentane heptan(ENE)oic acid, 2-heteroarylalkenyl derivatives as therapeutic agents
US5834498A (en) * 1992-09-21 1998-11-10 Allergan Cyclopentane heptan(ene)oic acid, 2-heteroarylalkenyl derivatives as therapeutic agents
US6124344A (en) * 1993-12-28 2000-09-26 Allergan Sales, Inc. Cyclopentane heptan(ene)oic acid, 2-heteroarylalkenyl derivatives as therapeutic agents
ES2159734T3 (es) * 1995-05-18 2001-10-16 Allergan Sales Inc Derivados 2-heteroarilalquenilicos del acido ciclopentano-heptan(en)oico como agentes terapeuticos para el tratamiento de la hipertension ocular.

Also Published As

Publication number Publication date
JP2020073513A (ja) 2020-05-14
AU2014361794B2 (en) 2019-04-04
CN105814033B (zh) 2019-10-25
CL2019000471A1 (es) 2019-07-12
UA121108C2 (uk) 2020-04-10
BR112016013594A2 (es) 2017-08-08
CL2016001448A1 (es) 2017-03-03
US20170087163A1 (en) 2017-03-30
MX2016007717A (es) 2016-09-09
IL283810A (en) 2021-07-29
BR112016013594A8 (pt) 2020-05-19
US20150166504A1 (en) 2015-06-18
AU2014361794A1 (en) 2016-06-16
CA2933556A1 (en) 2015-06-18
SG10201709702UA (en) 2018-01-30
WO2015089475A1 (en) 2015-06-18
US9353079B2 (en) 2016-05-31
EP3080096A1 (en) 2016-10-19
IL245917A0 (en) 2016-08-02
RU2730520C2 (ru) 2020-08-24
CN105814033A (zh) 2016-07-27
KR20160097310A (ko) 2016-08-17
JP2016539994A (ja) 2016-12-22
IL245917B (en) 2021-06-30
SA516371307B1 (ar) 2018-10-04

Similar Documents

Publication Publication Date Title
IL261602A (en) CD40 antibodies with increased agonistic activity
EP2951158A4 (en) PROCESS FOR THE PREPARATION OF IVACAFTOR AND SOLVATES THEREOF
EP2970418A4 (en) EZH2 PEPTIDE STABILIZED
HRP20181122T1 (hr) Postupak za pripremu jopamidola
PT3071247T (pt) Dispositivo para a construção de pele
HUE040294T2 (hu) Katalizátor foszgén elõállításához és eljárás foszgén elõállítására a katalizátor alkalmazásával
IL245474A0 (en) Process for the preparation of 5-fluoro-1h-pyrazoles
IL245476A0 (en) Process for preparing 5-fluoro-1h-pyrazoles
HK1202533A1 (en) Intermediates of ticagrelor and the preparation methods and for the preparation of ticagrelor
HK1220456A1 (zh) -乙酰嗎啡類似物,和其合成方法和用途
IL283810A (en) Solid forms of the compound alpha, omega-di-converted dihydroxy cyclopentyl and methods for their preparation and use
EP3065726A4 (en) Creatine analogs and the use thereof
ZA201603457B (en) Novel method for the synthesis of agomelatine
IL229326A (en) Process for making n-iodine-affluent
ZA201504080B (en) Combination medicament comprising phenylephrine and paracetamol
GB2510444B (en) Combination of phenylephrine and paracetamol
GB201323123D0 (en) Method for the preparation of biopolymers
HK1203297A2 (en) Mouse sticking structure with caution function
EP2983660A4 (en) MONO-ETHERS OF ISOHEXIDES AND METHOD FOR THE PRODUCTION THEREOF
IL246188A0 (en) A process for the preparation of tiacomycin
TH1401004311B (th) วิธีการสำหรับการผลิตวัตถุขึ้นรูปด้วยโฟมและวัตถุขึ้นรูปด้วยโฟม
CO6990721A2 (es) Proceso para la preparación de análogos de magnolol
TWM475359U (en) Improved structure of album