SG11201601461RA - Pharmaceutical composition containing pyrimidine compound as active ingredient - Google Patents
Pharmaceutical composition containing pyrimidine compound as active ingredientInfo
- Publication number
- SG11201601461RA SG11201601461RA SG11201601461RA SG11201601461RA SG11201601461RA SG 11201601461R A SG11201601461R A SG 11201601461RA SG 11201601461R A SG11201601461R A SG 11201601461RA SG 11201601461R A SG11201601461R A SG 11201601461RA SG 11201601461R A SG11201601461R A SG 11201601461RA
- Authority
- SG
- Singapore
- Prior art keywords
- pharmaceutical composition
- active ingredient
- composition containing
- pyrimidine compound
- containing pyrimidine
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Gastroenterology & Hepatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Dermatology (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2013176355 | 2013-08-28 | ||
PCT/JP2014/072349 WO2015030021A1 (ja) | 2013-08-28 | 2014-08-27 | ピリミジン化合物を有効成分とする医薬組成物 |
Publications (1)
Publication Number | Publication Date |
---|---|
SG11201601461RA true SG11201601461RA (en) | 2016-03-30 |
Family
ID=52586573
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG11201601461RA SG11201601461RA (en) | 2013-08-28 | 2014-08-27 | Pharmaceutical composition containing pyrimidine compound as active ingredient |
Country Status (16)
Country | Link |
---|---|
US (1) | US20160199371A1 (es) |
EP (1) | EP3040072A4 (es) |
JP (1) | JPWO2015030021A1 (es) |
KR (1) | KR20160040719A (es) |
CN (1) | CN105492009A (es) |
AR (1) | AR097455A1 (es) |
AU (1) | AU2014312919A1 (es) |
CA (1) | CA2922352A1 (es) |
HK (1) | HK1219432A1 (es) |
IL (1) | IL244206A0 (es) |
MX (1) | MX2016002589A (es) |
PH (1) | PH12016500372A1 (es) |
RU (1) | RU2016106774A (es) |
SG (1) | SG11201601461RA (es) |
TW (1) | TW201605452A (es) |
WO (1) | WO2015030021A1 (es) |
Families Citing this family (30)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8754114B2 (en) | 2010-12-22 | 2014-06-17 | Incyte Corporation | Substituted imidazopyridazines and benzimidazoles as inhibitors of FGFR3 |
PL3176170T3 (pl) | 2012-06-13 | 2019-05-31 | Incyte Holdings Corp | Podstawione związki tricykliczne jako inhibitory fgfr |
US9388185B2 (en) | 2012-08-10 | 2016-07-12 | Incyte Holdings Corporation | Substituted pyrrolo[2,3-b]pyrazines as FGFR inhibitors |
US9266892B2 (en) | 2012-12-19 | 2016-02-23 | Incyte Holdings Corporation | Fused pyrazoles as FGFR inhibitors |
CA2909207C (en) | 2013-04-19 | 2021-11-02 | Incyte Corporation | Bicyclic heterocycles as fgfr inhibitors |
CN110354128A (zh) | 2013-10-18 | 2019-10-22 | 卫材R&D管理有限公司 | 嘧啶fgfr4抑制剂 |
PE20160546A1 (es) | 2013-10-25 | 2016-05-26 | Novartis Ag | Compuestos derivados de piridilo biciclicos fusionados a anillo como inhibidores de fgfr4 |
JP6585167B2 (ja) | 2014-10-03 | 2019-10-02 | ノバルティス アーゲー | Fgfr4阻害剤としての縮環二環式ピリジル誘導体の使用 |
US10851105B2 (en) | 2014-10-22 | 2020-12-01 | Incyte Corporation | Bicyclic heterocycles as FGFR4 inhibitors |
US9580423B2 (en) | 2015-02-20 | 2017-02-28 | Incyte Corporation | Bicyclic heterocycles as FGFR4 inhibitors |
MA41551A (fr) | 2015-02-20 | 2017-12-26 | Incyte Corp | Hétérocycles bicycliques utilisés en tant qu'inhibiteurs de fgfr4 |
EP3617205B1 (en) | 2015-02-20 | 2021-08-04 | Incyte Corporation | Bicyclic heterocycles as fgfr inhibitors |
US9802917B2 (en) | 2015-03-25 | 2017-10-31 | Novartis Ag | Particles of N-(5-cyano-4-((2-methoxyethyl)amino)pyridin-2-yl)-7-formyl-6-((4-methyl-2-oxopiperazin-1-yl)methyl)-3,4-dihydro-1,8-naphthyridine-1(2H)-carboxamide |
KR102548229B1 (ko) | 2015-04-14 | 2023-06-27 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 결정질 fgfr4 억제제 화합물 및 그의 용도 |
JP7372740B2 (ja) | 2016-05-10 | 2023-11-01 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 細胞生存性及び/又は細胞増殖を低減するための薬物の組み合わせ |
CN107541495B (zh) * | 2016-06-28 | 2022-04-26 | 上海市东方医院 | 一种fgf19过表达的人肝癌细胞系及其应用 |
WO2018055503A1 (en) | 2016-09-20 | 2018-03-29 | Novartis Ag | Combination comprising a pd-1 antagonist and an fgfr4 inhibitor |
JP7394623B2 (ja) | 2016-11-02 | 2023-12-08 | ノバルティス アーゲー | Fgfr4インヒビターおよび胆汁酸捕捉薬の組合せ |
AR111960A1 (es) | 2017-05-26 | 2019-09-04 | Incyte Corp | Formas cristalinas de un inhibidor de fgfr y procesos para su preparación |
CA3099287A1 (en) | 2018-05-04 | 2019-11-07 | Incyte Corporation | Solid forms of an fgfr inhibitor and processes for preparing the same |
WO2019213506A1 (en) | 2018-05-04 | 2019-11-07 | Incyte Corporation | Salts of an fgfr inhibitor |
US11628162B2 (en) | 2019-03-08 | 2023-04-18 | Incyte Corporation | Methods of treating cancer with an FGFR inhibitor |
WO2021007269A1 (en) | 2019-07-09 | 2021-01-14 | Incyte Corporation | Bicyclic heterocycles as fgfr inhibitors |
KR20220100879A (ko) | 2019-10-14 | 2022-07-18 | 인사이트 코포레이션 | Fgfr 저해제로서의 이환식 헤테로사이클 |
US11566028B2 (en) | 2019-10-16 | 2023-01-31 | Incyte Corporation | Bicyclic heterocycles as FGFR inhibitors |
MX2022006691A (es) | 2019-12-04 | 2022-09-19 | Incyte Corp | Derivados de un inhibidor de receptores del factor de crecimiento de fibroblastos (fgfr). |
EP4069696A1 (en) | 2019-12-04 | 2022-10-12 | Incyte Corporation | Tricyclic heterocycles as fgfr inhibitors |
US12012409B2 (en) | 2020-01-15 | 2024-06-18 | Incyte Corporation | Bicyclic heterocycles as FGFR inhibitors |
WO2021231928A1 (en) * | 2020-05-15 | 2021-11-18 | Eisai R&D Management Co., Ltd. | A method for treating cancer with an oral dosage form of an fgfr4 inhibitor |
WO2022261160A1 (en) | 2021-06-09 | 2022-12-15 | Incyte Corporation | Tricyclic heterocycles as fgfr inhibitors |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2008533166A (ja) | 2005-03-16 | 2008-08-21 | ターゲジェン インコーポレーティッド | ピリミジン化合物および使用法 |
WO2007056075A2 (en) | 2005-11-02 | 2007-05-18 | Targegen, Inc. | Six membered heteroaromatic inhibitors targeting resistant kinase mutations |
WO2008008234A1 (en) | 2006-07-07 | 2008-01-17 | Targegen, Inc. | 2-amino-5-substituted pyrimidine inhibitors |
EA026953B1 (ru) | 2012-02-28 | 2017-06-30 | Астеллас Фарма Инк. | Азотсодержащее ароматическое гетероциклическое соединение |
EA029140B1 (ru) * | 2012-03-08 | 2018-02-28 | Астеллас Фарма Инк. | Новый слитый fgfr3 |
-
2014
- 2014-08-26 AR ARP140103193A patent/AR097455A1/es unknown
- 2014-08-26 TW TW103129371A patent/TW201605452A/zh unknown
- 2014-08-27 RU RU2016106774A patent/RU2016106774A/ru not_active Application Discontinuation
- 2014-08-27 KR KR1020167007640A patent/KR20160040719A/ko not_active Application Discontinuation
- 2014-08-27 WO PCT/JP2014/072349 patent/WO2015030021A1/ja active Application Filing
- 2014-08-27 EP EP14840047.6A patent/EP3040072A4/en not_active Withdrawn
- 2014-08-27 MX MX2016002589A patent/MX2016002589A/es unknown
- 2014-08-27 CN CN201480047119.2A patent/CN105492009A/zh active Pending
- 2014-08-27 SG SG11201601461RA patent/SG11201601461RA/en unknown
- 2014-08-27 AU AU2014312919A patent/AU2014312919A1/en not_active Abandoned
- 2014-08-27 US US14/914,955 patent/US20160199371A1/en not_active Abandoned
- 2014-08-27 JP JP2015534246A patent/JPWO2015030021A1/ja active Pending
- 2014-08-27 CA CA2922352A patent/CA2922352A1/en not_active Abandoned
-
2016
- 2016-02-21 IL IL244206A patent/IL244206A0/en unknown
- 2016-02-24 PH PH12016500372A patent/PH12016500372A1/en unknown
- 2016-06-29 HK HK16107576.9A patent/HK1219432A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
PH12016500372A1 (en) | 2016-05-02 |
MX2016002589A (es) | 2016-06-14 |
KR20160040719A (ko) | 2016-04-14 |
EP3040072A1 (en) | 2016-07-06 |
HK1219432A1 (zh) | 2017-04-07 |
JPWO2015030021A1 (ja) | 2017-03-02 |
EP3040072A4 (en) | 2017-03-29 |
WO2015030021A1 (ja) | 2015-03-05 |
TW201605452A (zh) | 2016-02-16 |
AU2014312919A1 (en) | 2016-03-10 |
AR097455A1 (es) | 2016-03-16 |
RU2016106774A (ru) | 2017-10-03 |
US20160199371A1 (en) | 2016-07-14 |
IL244206A0 (en) | 2016-04-21 |
CN105492009A (zh) | 2016-04-13 |
CA2922352A1 (en) | 2015-03-05 |
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