SG11201601461RA - Pharmaceutical composition containing pyrimidine compound as active ingredient - Google Patents

Pharmaceutical composition containing pyrimidine compound as active ingredient

Info

Publication number
SG11201601461RA
SG11201601461RA SG11201601461RA SG11201601461RA SG11201601461RA SG 11201601461R A SG11201601461R A SG 11201601461RA SG 11201601461R A SG11201601461R A SG 11201601461RA SG 11201601461R A SG11201601461R A SG 11201601461RA SG 11201601461R A SG11201601461R A SG 11201601461RA
Authority
SG
Singapore
Prior art keywords
pharmaceutical composition
active ingredient
composition containing
pyrimidine compound
containing pyrimidine
Prior art date
Application number
SG11201601461RA
Other languages
English (en)
Inventor
Takashi Futami
Rumi Takeshita
Original Assignee
Astellas Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astellas Pharma Inc filed Critical Astellas Pharma Inc
Publication of SG11201601461RA publication Critical patent/SG11201601461RA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Dermatology (AREA)
SG11201601461RA 2013-08-28 2014-08-27 Pharmaceutical composition containing pyrimidine compound as active ingredient SG11201601461RA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2013176355 2013-08-28
PCT/JP2014/072349 WO2015030021A1 (ja) 2013-08-28 2014-08-27 ピリミジン化合物を有効成分とする医薬組成物

Publications (1)

Publication Number Publication Date
SG11201601461RA true SG11201601461RA (en) 2016-03-30

Family

ID=52586573

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201601461RA SG11201601461RA (en) 2013-08-28 2014-08-27 Pharmaceutical composition containing pyrimidine compound as active ingredient

Country Status (16)

Country Link
US (1) US20160199371A1 (es)
EP (1) EP3040072A4 (es)
JP (1) JPWO2015030021A1 (es)
KR (1) KR20160040719A (es)
CN (1) CN105492009A (es)
AR (1) AR097455A1 (es)
AU (1) AU2014312919A1 (es)
CA (1) CA2922352A1 (es)
HK (1) HK1219432A1 (es)
IL (1) IL244206A0 (es)
MX (1) MX2016002589A (es)
PH (1) PH12016500372A1 (es)
RU (1) RU2016106774A (es)
SG (1) SG11201601461RA (es)
TW (1) TW201605452A (es)
WO (1) WO2015030021A1 (es)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8754114B2 (en) 2010-12-22 2014-06-17 Incyte Corporation Substituted imidazopyridazines and benzimidazoles as inhibitors of FGFR3
PL3176170T3 (pl) 2012-06-13 2019-05-31 Incyte Holdings Corp Podstawione związki tricykliczne jako inhibitory fgfr
US9388185B2 (en) 2012-08-10 2016-07-12 Incyte Holdings Corporation Substituted pyrrolo[2,3-b]pyrazines as FGFR inhibitors
US9266892B2 (en) 2012-12-19 2016-02-23 Incyte Holdings Corporation Fused pyrazoles as FGFR inhibitors
CA2909207C (en) 2013-04-19 2021-11-02 Incyte Corporation Bicyclic heterocycles as fgfr inhibitors
CN110354128A (zh) 2013-10-18 2019-10-22 卫材R&D管理有限公司 嘧啶fgfr4抑制剂
PE20160546A1 (es) 2013-10-25 2016-05-26 Novartis Ag Compuestos derivados de piridilo biciclicos fusionados a anillo como inhibidores de fgfr4
JP6585167B2 (ja) 2014-10-03 2019-10-02 ノバルティス アーゲー Fgfr4阻害剤としての縮環二環式ピリジル誘導体の使用
US10851105B2 (en) 2014-10-22 2020-12-01 Incyte Corporation Bicyclic heterocycles as FGFR4 inhibitors
US9580423B2 (en) 2015-02-20 2017-02-28 Incyte Corporation Bicyclic heterocycles as FGFR4 inhibitors
MA41551A (fr) 2015-02-20 2017-12-26 Incyte Corp Hétérocycles bicycliques utilisés en tant qu'inhibiteurs de fgfr4
EP3617205B1 (en) 2015-02-20 2021-08-04 Incyte Corporation Bicyclic heterocycles as fgfr inhibitors
US9802917B2 (en) 2015-03-25 2017-10-31 Novartis Ag Particles of N-(5-cyano-4-((2-methoxyethyl)amino)pyridin-2-yl)-7-formyl-6-((4-methyl-2-oxopiperazin-1-yl)methyl)-3,4-dihydro-1,8-naphthyridine-1(2H)-carboxamide
KR102548229B1 (ko) 2015-04-14 2023-06-27 에자이 알앤드디 매니지먼트 가부시키가이샤 결정질 fgfr4 억제제 화합물 및 그의 용도
JP7372740B2 (ja) 2016-05-10 2023-11-01 エーザイ・アール・アンド・ディー・マネジメント株式会社 細胞生存性及び/又は細胞増殖を低減するための薬物の組み合わせ
CN107541495B (zh) * 2016-06-28 2022-04-26 上海市东方医院 一种fgf19过表达的人肝癌细胞系及其应用
WO2018055503A1 (en) 2016-09-20 2018-03-29 Novartis Ag Combination comprising a pd-1 antagonist and an fgfr4 inhibitor
JP7394623B2 (ja) 2016-11-02 2023-12-08 ノバルティス アーゲー Fgfr4インヒビターおよび胆汁酸捕捉薬の組合せ
AR111960A1 (es) 2017-05-26 2019-09-04 Incyte Corp Formas cristalinas de un inhibidor de fgfr y procesos para su preparación
CA3099287A1 (en) 2018-05-04 2019-11-07 Incyte Corporation Solid forms of an fgfr inhibitor and processes for preparing the same
WO2019213506A1 (en) 2018-05-04 2019-11-07 Incyte Corporation Salts of an fgfr inhibitor
US11628162B2 (en) 2019-03-08 2023-04-18 Incyte Corporation Methods of treating cancer with an FGFR inhibitor
WO2021007269A1 (en) 2019-07-09 2021-01-14 Incyte Corporation Bicyclic heterocycles as fgfr inhibitors
KR20220100879A (ko) 2019-10-14 2022-07-18 인사이트 코포레이션 Fgfr 저해제로서의 이환식 헤테로사이클
US11566028B2 (en) 2019-10-16 2023-01-31 Incyte Corporation Bicyclic heterocycles as FGFR inhibitors
MX2022006691A (es) 2019-12-04 2022-09-19 Incyte Corp Derivados de un inhibidor de receptores del factor de crecimiento de fibroblastos (fgfr).
EP4069696A1 (en) 2019-12-04 2022-10-12 Incyte Corporation Tricyclic heterocycles as fgfr inhibitors
US12012409B2 (en) 2020-01-15 2024-06-18 Incyte Corporation Bicyclic heterocycles as FGFR inhibitors
WO2021231928A1 (en) * 2020-05-15 2021-11-18 Eisai R&D Management Co., Ltd. A method for treating cancer with an oral dosage form of an fgfr4 inhibitor
WO2022261160A1 (en) 2021-06-09 2022-12-15 Incyte Corporation Tricyclic heterocycles as fgfr inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008533166A (ja) 2005-03-16 2008-08-21 ターゲジェン インコーポレーティッド ピリミジン化合物および使用法
WO2007056075A2 (en) 2005-11-02 2007-05-18 Targegen, Inc. Six membered heteroaromatic inhibitors targeting resistant kinase mutations
WO2008008234A1 (en) 2006-07-07 2008-01-17 Targegen, Inc. 2-amino-5-substituted pyrimidine inhibitors
EA026953B1 (ru) 2012-02-28 2017-06-30 Астеллас Фарма Инк. Азотсодержащее ароматическое гетероциклическое соединение
EA029140B1 (ru) * 2012-03-08 2018-02-28 Астеллас Фарма Инк. Новый слитый fgfr3

Also Published As

Publication number Publication date
PH12016500372A1 (en) 2016-05-02
MX2016002589A (es) 2016-06-14
KR20160040719A (ko) 2016-04-14
EP3040072A1 (en) 2016-07-06
HK1219432A1 (zh) 2017-04-07
JPWO2015030021A1 (ja) 2017-03-02
EP3040072A4 (en) 2017-03-29
WO2015030021A1 (ja) 2015-03-05
TW201605452A (zh) 2016-02-16
AU2014312919A1 (en) 2016-03-10
AR097455A1 (es) 2016-03-16
RU2016106774A (ru) 2017-10-03
US20160199371A1 (en) 2016-07-14
IL244206A0 (en) 2016-04-21
CN105492009A (zh) 2016-04-13
CA2922352A1 (en) 2015-03-05

Similar Documents

Publication Publication Date Title
IL244206A0 (en) A pharmaceutical preparation containing a pyrimidine compound as an active ingredient
ZA201406866B (en) Herbicidal composition comprising uracil compound as active ingredient
HK1211209A1 (en) Pharmaceutical formulation containing thienotriazolodiazepine compounds
LT3030262T (lt) Kombinuota farmacinė kompozicija
EP3082817A4 (en) Compositions for drug administration
EP3036231A4 (en) Substituted pyrimidine compounds, compositions and medicinal applications thereof
PL3043778T3 (pl) Kompozycje farmaceutyczne zawierające refametinib
HK1215191A1 (zh) 低劑量醫藥組合物
HK1205462A1 (en) Pharmaceutical preparation containing an antivirally active dihydroquinazoline derivative
HK1213182A1 (zh) 外用藥物組合物
EP3037090A4 (en) Composition containing monoacetyldiglyceride compound as active ingredient for preventing or treating rheumatoid arthritis
EP2990038A4 (en) SOLID PHARMACEUTICAL COMPOSITION
HUE043804T2 (hu) Kristályos macitentánt tartalmazó gyógyászati készítmény
EP2990039A4 (en) Solid pharmaceutical composition
EP3037092A4 (en) Composition containing monoacetyldiglyceride compound as active ingredient for inhibiting blood cancer or metastasis
IL240875A0 (en) Heterocyclic compounds and pharmaceutical preparations containing them
HK1243927A1 (zh) 含有茶皂醇衍生物作爲活性成分的組合物
IL249010A0 (en) A pharmaceutical preparation containing a pyrazine carboxamide compound as an active ingredient
IL243223B (en) History of imidazole, their preparation and pharmaceutical preparations containing them
EP2871187A4 (en) NOVEL COMPOUND OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT
HUP1300496A2 (hu) Stabil kombinációs gyógyszerkészítmény
PL3041837T3 (pl) Kryształ o specyficznym pokroju kryształu i kompozycja farmaceutyczna zawierająca ten kryształ jako składnik czynny
PL3043791T3 (pl) Środek przeciwnowotworowy zawierający związek aminoacetonitrylowy jako substancję czynną
EP2883546A4 (en) NOVEL DIFFERENTIALLY RELEASING PHARMACEUTICAL COMPOSITION CONTAINING THREE ACTIVE INGREDIENTS
HRP20171815T1 (hr) Stabilni farmaceutski pripravak koji sadrži amorfni rosuvastatin-kalcij