SG11201503628YA - 3-aminocyclopentane carboxamide derivatives - Google Patents

3-aminocyclopentane carboxamide derivatives

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Publication number
SG11201503628YA
SG11201503628YA SG11201503628YA SG11201503628YA SG11201503628YA SG 11201503628Y A SG11201503628Y A SG 11201503628YA SG 11201503628Y A SG11201503628Y A SG 11201503628YA SG 11201503628Y A SG11201503628Y A SG 11201503628YA SG 11201503628Y A SG11201503628Y A SG 11201503628YA
Authority
SG
Singapore
Prior art keywords
aminocyclopentane
carboxamide derivatives
carboxamide
derivatives
aminocyclopentane carboxamide
Prior art date
Application number
SG11201503628YA
Other languages
English (en)
Inventor
Christos Tsaklakidis
Wolfgang Staehle
Brigitta Leuthner
Paul Czodrowski
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of SG11201503628YA publication Critical patent/SG11201503628YA/en

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    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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IL125954A (en) 1996-03-05 2003-06-24 Zeneca Ltd Quinazoline derivatives, processes for their preparation, pharmaceutical compositions containing them and use thereof in the manufacture of medicaments having an antiangiogenic and/or vascular permeability reducing effect
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CN104797553A (zh) 2015-07-22
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CA2891484A1 (en) 2014-05-22
US20160264517A1 (en) 2016-09-15
EP2920146A1 (en) 2015-09-23
HK1212671A1 (zh) 2016-06-17
JP2016504280A (ja) 2016-02-12
MX2015006037A (es) 2015-08-07
KR20150085045A (ko) 2015-07-22
EP2920146B1 (en) 2016-09-28
AR093461A1 (es) 2015-06-10
ES2608355T3 (es) 2017-04-10
RU2641913C2 (ru) 2018-01-23
US9732032B2 (en) 2017-08-15
WO2014075754A1 (en) 2014-05-22
CN104797553B (zh) 2017-07-21
BR112015010512A2 (pt) 2017-07-11
JP6316835B2 (ja) 2018-04-25
RU2015122801A (ru) 2017-01-10
AU2013347232A8 (en) 2015-08-06
ZA201504323B (en) 2017-09-27

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