SG10201700493XA - Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists - Google Patents

Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists

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Publication number
SG10201700493XA
SG10201700493XA SG10201700493XA SG10201700493XA SG10201700493XA SG 10201700493X A SG10201700493X A SG 10201700493XA SG 10201700493X A SG10201700493X A SG 10201700493XA SG 10201700493X A SG10201700493X A SG 10201700493XA SG 10201700493X A SG10201700493X A SG 10201700493XA
Authority
SG
Singapore
Prior art keywords
pyrazol
benzene sulfonamides
ccr9 antagonists
ccr9
antagonists
Prior art date
Application number
SG10201700493XA
Other languages
English (en)
Inventor
Xi Chen
Junfa Fan
Pingchen Fan
Antoni Krasinski
Lianfa Li
Rebecca M Lui
Jeffrey P Mcmahon
Jay P Powers
Yibin Zeng
Penglie Zhang
Original Assignee
Chemocentryx Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chemocentryx Inc filed Critical Chemocentryx Inc
Publication of SG10201700493XA publication Critical patent/SG10201700493XA/en

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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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SG10201700493XA 2012-02-29 2013-02-28 Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists SG10201700493XA (en)

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AU (3) AU2013225938B2 (zh)
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US10827315B2 (en) * 2006-04-07 2020-11-03 Groupon, Inc. Facilitating user interactions based on proximity
CN107266425B (zh) * 2012-02-29 2020-03-03 坎莫森特里克斯公司 作为ccr9拮抗剂的吡唑-1-基苯磺酰胺
WO2014088113A1 (en) 2012-12-04 2014-06-12 Millennium Pharmaceuticals, Inc. Prophylactic or therapeutic method for sjogren's syndrome using specific ccr9 receptor inhibitors/antagonists
GB201308978D0 (en) 2013-05-17 2013-07-03 Imp Innovations Ltd Method for producing polymers and block copolymers
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