SG10201506873WA - Fast-dissolve dosage forms of 5-ht2c agonists - Google Patents

Fast-dissolve dosage forms of 5-ht2c agonists

Info

Publication number
SG10201506873WA
SG10201506873WA SG10201506873WA SG10201506873WA SG10201506873WA SG 10201506873W A SG10201506873W A SG 10201506873WA SG 10201506873W A SG10201506873W A SG 10201506873WA SG 10201506873W A SG10201506873W A SG 10201506873WA SG 10201506873W A SG10201506873W A SG 10201506873WA
Authority
SG
Singapore
Prior art keywords
fast
dosage forms
ht2c agonists
dissolve dosage
dissolve
Prior art date
Application number
SG10201506873WA
Other languages
English (en)
Inventor
Anthony C Blackburn
Scott Stirn
Yun Shan
Anna Shifrina
Original Assignee
Arena Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arena Pharm Inc filed Critical Arena Pharm Inc
Publication of SG10201506873WA publication Critical patent/SG10201506873WA/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16—Benzazepines; Hydrogenated benzazepines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Child & Adolescent Psychology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SG10201506873WA 2010-09-01 2011-08-31 Fast-dissolve dosage forms of 5-ht2c agonists SG10201506873WA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US40258910P 2010-09-01 2010-09-01

Publications (1)

Publication Number Publication Date
SG10201506873WA true SG10201506873WA (en) 2015-10-29

Family

ID=44645827

Family Applications (2)

Application Number Title Priority Date Filing Date
SG10201506873WA SG10201506873WA (en) 2010-09-01 2011-08-31 Fast-dissolve dosage forms of 5-ht2c agonists
SG2013015607A SG188363A1 (en) 2010-09-01 2011-08-31 Fast-dissolve dosage forms of 5-ht2c agonists

Family Applications After (1)

Application Number Title Priority Date Filing Date
SG2013015607A SG188363A1 (en) 2010-09-01 2011-08-31 Fast-dissolve dosage forms of 5-ht2c agonists

Country Status (11)

Country Link
US (1) US20140148442A1 (enExample)
EP (1) EP2611781A1 (enExample)
JP (1) JP2013536858A (enExample)
KR (1) KR20130138768A (enExample)
CN (1) CN103189358A (enExample)
AU (1) AU2011296027A1 (enExample)
CA (1) CA2808900A1 (enExample)
IN (1) IN2013DN02552A (enExample)
MX (1) MX2013002430A (enExample)
SG (2) SG10201506873WA (enExample)
WO (1) WO2012030951A1 (enExample)

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EP2611433A2 (en) 2010-09-01 2013-07-10 Arena Pharmaceuticals, Inc. Non-hygroscopic salts of 5-ht2c agonists
KR20130138770A (ko) 2010-09-01 2013-12-19 아레나 파마슈티칼스, 인크. 광학적으로 활성 산을 갖는 로르카세린의 염
JP2015534563A (ja) 2012-10-09 2015-12-03 アリーナ ファーマシューティカルズ， インコーポレイテッド 体重管理の方法
WO2014135545A1 (en) * 2013-03-05 2014-09-12 Sandoz Ag Solid dispersion comprising amorphous lorcaserin hydrochloride
CN105431415A (zh) * 2013-05-20 2016-03-23 斯洛文尼亚莱柯制药股份有限公司 通过烯烃的弗瑞德-克来福特烷基化进行的8-氯-3-苯并[d]氮杂*的新合成方法
EP2868656A1 (en) * 2013-11-05 2015-05-06 LEK Pharmaceuticals d.d. Stabilized amorphous lorcaserin hydrochloride
WO2015096119A1 (zh) * 2013-12-27 2015-07-02 杭州普晒医药科技有限公司 氯卡色林盐及其晶体、其制备方法和用途
US9981912B2 (en) 2014-04-21 2018-05-29 Hangzhou Pushai Pharmaceutical Technology Co., Ltd. Cocrystal of lorcaserin, preparation methods, pharmaceutical compositions and uses thereof
CN103901151A (zh) * 2014-04-23 2014-07-02 湖北朗昕生化药业有限公司 一种hplc法检测氯卡色林盐酸盐含量的方法
WO2016069875A1 (en) 2014-10-30 2016-05-06 Arena Pharmaceuticals, Inc. Compositions and methods for ceasing tobacco smoking
US10143706B2 (en) 2016-06-29 2018-12-04 Cannscience Innovations, Inc. Decarboxylated cannabis resins, uses thereof and methods of making same

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Also Published As

Publication number Publication date
AU2011296027A1 (en) 2013-04-04
CA2808900A1 (en) 2012-03-08
CN103189358A (zh) 2013-07-03
JP2013536858A (ja) 2013-09-26
WO2012030951A1 (en) 2012-03-08
IN2013DN02552A (enExample) 2015-08-07
SG188363A1 (en) 2013-04-30
MX2013002430A (es) 2013-07-22
KR20130138768A (ko) 2013-12-19
US20140148442A1 (en) 2014-05-29
EP2611781A1 (en) 2013-07-10

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