SG10201501054TA - Solid dispersion of rifaximin - Google Patents
Solid dispersion of rifaximinInfo
- Publication number
- SG10201501054TA SG10201501054TA SG10201501054TA SG10201501054TA SG10201501054TA SG 10201501054T A SG10201501054T A SG 10201501054TA SG 10201501054T A SG10201501054T A SG 10201501054TA SG 10201501054T A SG10201501054T A SG 10201501054TA SG 10201501054T A SG10201501054T A SG 10201501054TA
- Authority
- SG
- Singapore
- Prior art keywords
- rifaximin
- solid dispersion
- dispersion
- solid
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0043—Nose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0046—Ear
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Molecular Biology (AREA)
- Dispersion Chemistry (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Biophysics (AREA)
- Inorganic Chemistry (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Gynecology & Obstetrics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN1287KO2009 | 2009-10-27 |
Publications (1)
Publication Number | Publication Date |
---|---|
SG10201501054TA true SG10201501054TA (en) | 2015-04-29 |
Family
ID=43922730
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG10201501054TA SG10201501054TA (en) | 2009-10-27 | 2010-10-27 | Solid dispersion of rifaximin |
Country Status (22)
Country | Link |
---|---|
US (3) | US20120214833A1 (de) |
EP (1) | EP2493456B1 (de) |
JP (2) | JP6211768B2 (de) |
KR (5) | KR101972354B1 (de) |
CN (2) | CN113274355B (de) |
AU (2) | AU2010313078A1 (de) |
CA (1) | CA2778981C (de) |
CL (1) | CL2012001080A1 (de) |
ES (1) | ES2712080T3 (de) |
GE (1) | GEP201706693B (de) |
IL (1) | IL219508A (de) |
MA (1) | MA33761B1 (de) |
MX (1) | MX346660B (de) |
MY (1) | MY177151A (de) |
NZ (1) | NZ599944A (de) |
PE (1) | PE20121185A1 (de) |
RU (1) | RU2012121599A (de) |
SG (1) | SG10201501054TA (de) |
TN (1) | TN2012000195A1 (de) |
UA (1) | UA110199C2 (de) |
WO (1) | WO2011051971A2 (de) |
ZA (1) | ZA201203226B (de) |
Families Citing this family (24)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2522895T3 (es) | 2005-03-03 | 2014-11-19 | Alfa Wassermann S.P.A. | Nuevas formas polimorfas de rifaximina, procedimientos para su producción y uso de las mismas en preparados medicinales |
ITBO20050123A1 (it) | 2005-03-07 | 2005-06-06 | Alfa Wassermann Spa | Formulazioni farmaceutiche gastroresistenti contenenti rifaximina |
ITMI20061692A1 (it) | 2006-09-05 | 2008-03-06 | Alfa Wassermann Spa | Uso di polioli per ottenere forme polimorfe stabili di rifaximina |
US8486956B2 (en) | 2008-02-25 | 2013-07-16 | Salix Pharmaceuticals, Ltd | Forms of rifaximin and uses thereof |
KR101674382B1 (ko) | 2008-02-25 | 2016-11-09 | 샐릭스 파마슈티컬스 리미티드 | 리팍시민의 형태 및 이의 용도 |
SG10201501054TA (en) * | 2009-10-27 | 2015-04-29 | Lupin Ltd | Solid dispersion of rifaximin |
US9018684B2 (en) | 2009-11-23 | 2015-04-28 | California Institute Of Technology | Chemical sensing and/or measuring devices and methods |
EP2519108A4 (de) | 2009-12-31 | 2013-10-16 | Ira Milton Trachtman | Zusammensetzungen und verfahren zur behandlung und vorbeugung von chronisch-entzündlicher darmerkrankung |
IT1398550B1 (it) | 2010-03-05 | 2013-03-01 | Alfa Wassermann Spa | Formulazioni comprendenti rifaximina utili per ottenere un effetto prolungato nel tempo |
KR101887004B1 (ko) * | 2010-07-12 | 2018-08-09 | 샐릭스 파마슈티컬스 리미티드 | 리팍시민의 제형 및 이의 용도 |
PT2672970T (pt) | 2011-02-11 | 2018-10-11 | Salix Pharmaceuticals Ltd | Formas de rifaximina e suas utilizações |
CN102512358B (zh) * | 2011-12-16 | 2013-04-10 | 南京农业大学 | 家畜用利福昔明阴道栓剂及其制备方法 |
WO2013112809A2 (en) * | 2012-01-25 | 2013-08-01 | Salix Pharmaceuticals, Ltd | Rifaximin derivative and uses thereof |
ITBO20120368A1 (it) | 2012-07-06 | 2014-01-07 | Alfa Wassermann Spa | Composizioni comprendenti rifaximina e amminoacidi, cristalli di rifaximina derivanti da tali composizioni e loro uso. |
WO2014013498A1 (en) * | 2012-07-17 | 2014-01-23 | Symed Labs Limited | Amorphous coprecipitates of linezolid |
WO2015047941A2 (en) * | 2013-09-27 | 2015-04-02 | Trachtman Ira Milton | Compositions and methods for treatment and prophylaxis of gastrointestinal diseases |
US9938298B2 (en) | 2014-05-12 | 2018-04-10 | Alfa Wassermann S.P.A. | Solvated crystal form of rifaximin, production, compositions and uses thereof |
RS63751B1 (sr) | 2016-09-30 | 2022-12-30 | Salix Pharmaceuticals Inc | Čvrsti disperzioni oblici rifaksimina |
CN106491558A (zh) * | 2016-12-09 | 2017-03-15 | 福建生物工程职业技术学院 | 盐酸阿考替胺膜控型缓释制剂及其制备方法 |
CN106727350A (zh) * | 2016-12-28 | 2017-05-31 | 潍坊宇洋药业有限公司 | 一种林可霉素固体分散体制剂及其制备方法 |
CN109772234B (zh) | 2017-11-14 | 2024-01-05 | 中国石油化工股份有限公司 | 用于丙烯氨氧化反应器的原料气进料系统 |
WO2019157066A1 (en) * | 2018-02-06 | 2019-08-15 | Robert Niichel | A multiparticulate including pharmaceutical or probiotic active ingredients |
EP4034091A1 (de) * | 2019-09-24 | 2022-08-03 | Bausch Health Ireland Limited | Rifaximin-flüssigformulierungen |
WO2022090490A1 (en) * | 2020-10-29 | 2022-05-05 | Bausch Health Ireland Limited | Rifaximin liquid formulations for use in the treatment of sickle cell disease |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1154655B (it) | 1980-05-22 | 1987-01-21 | Alfa Farmaceutici Spa | Derivati imidazo-rifamicinici metodi per la loro preparazione e loro uso come sostanza ad azione antibatterica |
IT1253711B (it) * | 1991-12-17 | 1995-08-23 | Alfa Wassermann Spa | Formulazioni farmaceutiche vaginali contenenti rifaximin e loro uso nel trattamento delle infezioni vaginali |
WO1993011749A1 (en) * | 1991-12-18 | 1993-06-24 | Warner-Lambert Company | A process for the preparation of a solid dispersion |
IT1320176B1 (it) * | 2000-12-22 | 2003-11-26 | Nicox Sa | Dispersioni solide di principi attivi nitrati. |
ITMI20032144A1 (it) * | 2003-11-07 | 2005-05-08 | Alfa Wassermann Spa | Forme polimorfe di rifaximina, processi per ottenerle e |
JP2007516259A (ja) * | 2003-12-09 | 2007-06-21 | メッドクリスタルフォームズ、エルエルシー | 活性剤との混合相共結晶の調製方法 |
CA2687192C (en) * | 2007-06-04 | 2015-11-24 | Egalet A/S | Controlled release pharmaceutical compositions for prolonged effect |
AU2008273699A1 (en) * | 2007-07-06 | 2009-01-15 | Lupin Limited | Pharmaceutical compositions of rifaximin |
DK2011486T3 (da) * | 2007-07-06 | 2012-09-03 | Lupin Ltd | Farmaceutiske sammensætninger af rifaximin |
CN101502513A (zh) * | 2008-09-04 | 2009-08-12 | 山东淄博新达制药有限公司 | 一种利福昔明缓释制剂组合物及其制备方法 |
US8916193B2 (en) * | 2008-12-10 | 2014-12-23 | Cipla Limited | Rifaximin complexes |
SG10201501054TA (en) * | 2009-10-27 | 2015-04-29 | Lupin Ltd | Solid dispersion of rifaximin |
-
2010
- 2010-10-27 SG SG10201501054TA patent/SG10201501054TA/en unknown
- 2010-10-27 US US13/503,733 patent/US20120214833A1/en not_active Abandoned
- 2010-10-27 CN CN202110540088.6A patent/CN113274355B/zh active Active
- 2010-10-27 WO PCT/IN2010/000694 patent/WO2011051971A2/en active Application Filing
- 2010-10-27 KR KR1020177032267A patent/KR101972354B1/ko active IP Right Grant
- 2010-10-27 JP JP2012536017A patent/JP6211768B2/ja active Active
- 2010-10-27 MY MYPI2012001884A patent/MY177151A/en unknown
- 2010-10-27 KR KR1020217041533A patent/KR102456997B1/ko active IP Right Grant
- 2010-10-27 EP EP10790593.7A patent/EP2493456B1/de active Active
- 2010-10-27 ES ES10790593T patent/ES2712080T3/es active Active
- 2010-10-27 CN CN2010800554820A patent/CN102665693A/zh active Pending
- 2010-10-27 KR KR1020207023745A patent/KR20200100215A/ko not_active Application Discontinuation
- 2010-10-27 NZ NZ599944A patent/NZ599944A/en unknown
- 2010-10-27 PE PE2012000588A patent/PE20121185A1/es not_active Application Discontinuation
- 2010-10-27 AU AU2010313078A patent/AU2010313078A1/en not_active Abandoned
- 2010-10-27 RU RU2012121599/15A patent/RU2012121599A/ru unknown
- 2010-10-27 CA CA2778981A patent/CA2778981C/en active Active
- 2010-10-27 KR KR1020127012479A patent/KR20140015140A/ko active Application Filing
- 2010-10-27 MX MX2012004954A patent/MX346660B/es active IP Right Grant
- 2010-10-27 GE GEAP201012701A patent/GEP201706693B/en unknown
- 2010-10-27 UA UAA201206356A patent/UA110199C2/ru unknown
- 2010-10-27 KR KR1020187037658A patent/KR20190000931A/ko active Application Filing
-
2012
- 2012-04-26 TN TNP2012000195A patent/TN2012000195A1/en unknown
- 2012-04-26 CL CL2012001080A patent/CL2012001080A1/es unknown
- 2012-05-01 IL IL219508A patent/IL219508A/en active IP Right Grant
- 2012-05-04 ZA ZA2012/03226A patent/ZA201203226B/en unknown
- 2012-05-22 MA MA34885A patent/MA33761B1/fr unknown
-
2014
- 2014-01-09 US US14/151,515 patent/US20140221414A1/en not_active Abandoned
-
2015
- 2015-09-14 JP JP2015181131A patent/JP6234412B2/ja active Active
-
2016
- 2016-08-09 AU AU2016213722A patent/AU2016213722B2/en active Active
-
2020
- 2020-05-06 US US16/868,307 patent/US20200375959A1/en not_active Abandoned
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ZA201203226B (en) | Solid dispersion of rifaximin | |
IL222900A (en) | Forms of Rifaximin | |
PL2340960T3 (pl) | Przedział stanu naładowania | |
IL196456A0 (en) | Uderbelly of armord vehicle | |
HK1179608A1 (zh) | 利福昔明的晶型及其用途 | |
HUE064921T2 (hu) | Politiofén-részecskékbõl álló diszperz rendszer | |
EP2438246A4 (de) | Konstruktionsaspekte | |
EP2582707A4 (de) | Polymorphe formen von rifaximin | |
HK1165895A1 (zh) | 室調節 | |
ZA201102604B (en) | Alkylcyclohexylethers of dihydrotetraazabenzoazulenes | |
AU328140S (en) | Ring | |
ZA201108375B (en) | Solid preparation | |
PL2496340T3 (pl) | Dyspersja krzemionki | |
PL2133419T3 (pl) | Zastosowania beta-dipeptydów cyjanoficyny | |
EP2399463A4 (de) | Dispersion von phytosterolen | |
HK1163663A1 (en) | Rifamycin derivatives | |
GB0905702D0 (en) | Headset | |
EP2412366A4 (de) | Feste zubereitung | |
EP2412367A4 (de) | Feste zubereitung | |
GB2483195B (en) | Novel uses | |
TWM372743U (en) | Improved structure of Kendama | |
TWM365675U (en) | Improved structure of teapoy | |
EP2459540A4 (de) | Herstellung von fipamezol | |
GB0905956D0 (en) | Range assembly | |
GB0905280D0 (en) | Novel uses of VEGFxxxb |