SG10201405568UA - 4-substituted pyridin-3-yl-carboxamide compounds and methods of use - Google Patents

4-substituted pyridin-3-yl-carboxamide compounds and methods of use

Info

Publication number
SG10201405568UA
SG10201405568UA SG10201405568UA SG10201405568UA SG10201405568UA SG 10201405568U A SG10201405568U A SG 10201405568UA SG 10201405568U A SG10201405568U A SG 10201405568UA SG 10201405568U A SG10201405568U A SG 10201405568UA SG 10201405568U A SG10201405568U A SG 10201405568UA
Authority
SG
Singapore
Prior art keywords
methods
carboxamide compounds
substituted pyridin
pyridin
substituted
Prior art date
Application number
SG10201405568UA
Other languages
English (en)
Inventor
Jr Allen J Ebens
Xiaojing Wang
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of SG10201405568UA publication Critical patent/SG10201405568UA/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
SG10201405568UA 2009-09-08 2010-09-07 4-substituted pyridin-3-yl-carboxamide compounds and methods of use SG10201405568UA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24047409P 2009-09-08 2009-09-08

Publications (1)

Publication Number Publication Date
SG10201405568UA true SG10201405568UA (en) 2014-11-27

Family

ID=43479412

Family Applications (2)

Application Number Title Priority Date Filing Date
SG10201405568UA SG10201405568UA (en) 2009-09-08 2010-09-07 4-substituted pyridin-3-yl-carboxamide compounds and methods of use
SG2012015350A SG178986A1 (en) 2009-09-08 2010-09-07 4-substituted pyridin-3-yl-carboxamide compounds and methods of use

Family Applications After (1)

Application Number Title Priority Date Filing Date
SG2012015350A SG178986A1 (en) 2009-09-08 2010-09-07 4-substituted pyridin-3-yl-carboxamide compounds and methods of use

Country Status (7)

Country Link
EP (1) EP2475659B1 (ja)
JP (1) JP5567136B2 (ja)
CN (1) CN102625807B (ja)
CA (1) CA2770252C (ja)
ES (1) ES2557316T3 (ja)
SG (2) SG10201405568UA (ja)
WO (1) WO2011029802A1 (ja)

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WO2013175388A1 (en) * 2012-05-21 2013-11-28 Novartis Ag Novel ring-substituted n-pyridinyl amides as kinase inhibitors
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JP6437452B2 (ja) 2013-01-14 2018-12-12 インサイト・ホールディングス・コーポレイションＩｎｃｙｔｅ Ｈｏｌｄｉｎｇｓ Ｃｏｒｐｏｒａｔｉｏｎ Ｐｉｍキナーゼ阻害剤として有用な二環式芳香族カルボキサミド化合物
ME03780B (me) 2013-01-15 2021-04-20 Incyte Holdings Corp Jedinjenja tiazolkarboksamida i piridinkarboksamida korisna kao inhibitori pim kinaze
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JP6851826B2 (ja) * 2013-07-19 2021-03-31 オニキス セラピューティクス， インク．Ｏｎｙｘ Ｔｈｅｒａｐｅｕｔｉｃｓ， Ｉｎｃ． がんの治療のためのｐｉｍキナーゼ阻害剤と組み合わせたペプチドエポキシケトンプロテアソーム阻害剤
ES2792549T3 (es) 2013-08-07 2020-11-11 Incyte Corp Formas de dosificación de liberación sostenida para un inhibidor de JAK1
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Also Published As

Publication number Publication date
SG178986A1 (en) 2012-04-27
CA2770252C (en) 2018-06-12
WO2011029802A1 (en) 2011-03-17
JP2013503837A (ja) 2013-02-04
JP5567136B2 (ja) 2014-08-06
EP2475659B1 (en) 2015-10-28
CN102625807A (zh) 2012-08-01
EP2475659A1 (en) 2012-07-18
CN102625807B (zh) 2016-03-09
CA2770252A1 (en) 2011-03-17
ES2557316T3 (es) 2016-01-25

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