SE7705744L - PROCEDURES AND INTERMEDIATES FOR THE PREPARATION OF KINOXALIN-1,4-DIOXIDES - Google Patents
PROCEDURES AND INTERMEDIATES FOR THE PREPARATION OF KINOXALIN-1,4-DIOXIDESInfo
- Publication number
- SE7705744L SE7705744L SE7705744A SE7705744A SE7705744L SE 7705744 L SE7705744 L SE 7705744L SE 7705744 A SE7705744 A SE 7705744A SE 7705744 A SE7705744 A SE 7705744A SE 7705744 L SE7705744 L SE 7705744L
- Authority
- SE
- Sweden
- Prior art keywords
- formula
- dioxides
- kinoxalin
- intermediates
- procedures
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
- C07D241/50—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to ring nitrogen atoms
- C07D241/52—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Tropical Medicine & Parasitology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Physical Or Chemical Processes And Apparatus (AREA)
- Saccharide Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
The carbazates of formula I are obtained by reacting the quinoxaline N<1>,N<4>-dioxides carrying in position 2 a chloromethyl or bromomethyl group with one to two equivalents of an alkali metal carbonate and one to two equivalents of a hydrazine of formula R''NH-NH-COOCH3 at a temperature of between 75 and 85 DEG C and in an inert solvent. This hydrazine is prepared by reaction of methyl carbazate with a corresponding acid anhydride or sulphonyl halide which introduces the radical R''. The meaning of the symbols is explained in Claim 1. The compounds of formula I are strong antibacterial agents. <IMAGE>
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US69626376A | 1976-06-15 | 1976-06-15 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| SE7705744L true SE7705744L (en) | 1977-12-16 |
| SE428925B SE428925B (en) | 1983-08-01 |
Family
ID=24796354
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE7705744A SE428925B (en) | 1976-06-15 | 1977-05-16 | IMPROVED PROCEDURE FOR THE PREPARATION OF METHYL-3- (2-KINOXALINYLMETHYIN) -CARBAZATE-N? 721, N? 724-DIOXIDE |
| SE8003393A SE437985B (en) | 1976-06-15 | 1980-05-06 | NEW N-METOXICARBONYL-N? 721-SUBSTITUTED HYDRAZINE USED AS AN INTERMEDIATE FOR THE PREPARATION OF METHYL-3- (2-CHINOXALINYLMETHYL) -CARBAZATE-N? 721, N? 724-DI |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE8003393A SE437985B (en) | 1976-06-15 | 1980-05-06 | NEW N-METOXICARBONYL-N? 721-SUBSTITUTED HYDRAZINE USED AS AN INTERMEDIATE FOR THE PREPARATION OF METHYL-3- (2-CHINOXALINYLMETHYL) -CARBAZATE-N? 721, N? 724-DI |
Country Status (31)
| Country | Link |
|---|---|
| JP (2) | JPS52153986A (en) |
| AR (1) | AR221207A1 (en) |
| AT (1) | AT357562B (en) |
| BG (1) | BG35595A3 (en) |
| CA (1) | CA1087616A (en) |
| CH (1) | CH620911A5 (en) |
| CS (1) | CS200218B2 (en) |
| DD (2) | DD131371A5 (en) |
| DE (1) | DE2725023A1 (en) |
| DK (1) | DK142497B (en) |
| ES (2) | ES459745A1 (en) |
| FI (1) | FI771742A (en) |
| GB (3) | GB1591872A (en) |
| GR (1) | GR72289B (en) |
| HK (3) | HK1883A (en) |
| IE (1) | IE44684B1 (en) |
| IL (1) | IL52166A0 (en) |
| IT (1) | IT1078874B (en) |
| LU (1) | LU77474A1 (en) |
| MY (2) | MY8300230A (en) |
| NL (2) | NL166685C (en) |
| NO (2) | NO146864C (en) |
| NZ (1) | NZ184167A (en) |
| PH (2) | PH14866A (en) |
| PL (1) | PL105555B1 (en) |
| PT (1) | PT66618B (en) |
| SE (2) | SE428925B (en) |
| SG (1) | SG49282G (en) |
| SU (1) | SU657746A3 (en) |
| YU (1) | YU39492B (en) |
| ZA (1) | ZA772979B (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS60164410A (en) * | 1984-02-08 | 1985-08-27 | 株式会社石井製作所 | Threshing and sorting apparatus |
-
1977
- 1977-05-16 SE SE7705744A patent/SE428925B/en not_active IP Right Cessation
- 1977-05-17 CA CA278,574A patent/CA1087616A/en not_active Expired
- 1977-05-18 GB GB20800/77A patent/GB1591872A/en not_active Expired
- 1977-05-18 GB GB764/80A patent/GB1591873A/en not_active Expired
- 1977-05-18 GB GB765/80A patent/GB1591874A/en not_active Expired
- 1977-05-18 ZA ZA00772979A patent/ZA772979B/en unknown
- 1977-05-20 NZ NZ184167A patent/NZ184167A/en unknown
- 1977-05-20 GR GR53522A patent/GR72289B/el unknown
- 1977-05-20 IE IE1040/77A patent/IE44684B1/en not_active IP Right Cessation
- 1977-05-25 IL IL52166A patent/IL52166A0/en unknown
- 1977-05-26 CH CH650777A patent/CH620911A5/en not_active IP Right Cessation
- 1977-05-26 PH PH19820A patent/PH14866A/en unknown
- 1977-05-27 YU YU1327/77A patent/YU39492B/en unknown
- 1977-05-30 JP JP6315177A patent/JPS52153986A/en active Granted
- 1977-05-31 NL NL7705938.A patent/NL166685C/en not_active IP Right Cessation
- 1977-05-31 CS CS773581A patent/CS200218B2/en unknown
- 1977-05-31 DE DE19772725023 patent/DE2725023A1/en active Pending
- 1977-05-31 PT PT66618A patent/PT66618B/en unknown
- 1977-05-31 IT IT49637/77A patent/IT1078874B/en active
- 1977-05-31 NO NO771903A patent/NO146864C/en unknown
- 1977-06-01 DK DK240777AA patent/DK142497B/en unknown
- 1977-06-01 FI FI771742A patent/FI771742A/fi not_active Application Discontinuation
- 1977-06-01 AT AT387077A patent/AT357562B/en not_active IP Right Cessation
- 1977-06-02 AR AR267928A patent/AR221207A1/en active
- 1977-06-02 DD DD7700199261A patent/DD131371A5/en unknown
- 1977-06-02 DD DD77204377A patent/DD135080A5/en not_active IP Right Cessation
- 1977-06-02 LU LU77474A patent/LU77474A1/xx unknown
- 1977-06-13 BG BG7736608A patent/BG35595A3/en unknown
- 1977-06-14 ES ES459745A patent/ES459745A1/en not_active Expired
- 1977-06-14 ES ES459750A patent/ES459750A1/en not_active Expired
- 1977-06-14 SU SU772494213A patent/SU657746A3/en active
- 1977-06-15 PL PL1977198873A patent/PL105555B1/en unknown
- 1977-11-09 PH PH20413A patent/PH14481A/en unknown
-
1979
- 1979-11-10 JP JP14596079A patent/JPS5589256A/en active Granted
-
1980
- 1980-05-06 SE SE8003393A patent/SE437985B/en not_active IP Right Cessation
- 1980-12-10 NL NL8006697A patent/NL8006697A/en not_active Application Discontinuation
-
1981
- 1981-09-22 NO NO813221A patent/NO147422C/en unknown
-
1982
- 1982-10-11 SG SG49282A patent/SG49282G/en unknown
-
1983
- 1983-01-13 HK HK18/83A patent/HK1883A/en unknown
- 1983-01-13 HK HK19/83A patent/HK1983A/en unknown
- 1983-01-13 HK HK20/83A patent/HK2083A/en unknown
- 1983-12-30 MY MY230/83A patent/MY8300230A/en unknown
- 1983-12-30 MY MY229/83A patent/MY8300229A/en unknown
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| NUG | Patent has lapsed |
Ref document number: 7705744-6 Effective date: 19941210 Format of ref document f/p: F |
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| NUG | Patent has lapsed |
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