SE454442B - Forfarande for framstellning av 4-metoxi-2'-(2-(1-metyl-2-piperidyl)etyl)-bensamid(enkainid) och 2-(2-pyridylacetyl)-p-anisanilid som mellanprodukt - Google Patents

Forfarande for framstellning av 4-metoxi-2'-(2-(1-metyl-2-piperidyl)etyl)-bensamid(enkainid) och 2-(2-pyridylacetyl)-p-anisanilid som mellanprodukt

Info

Publication number
SE454442B
SE454442B SE8207112A SE8207112A SE454442B SE 454442 B SE454442 B SE 454442B SE 8207112 A SE8207112 A SE 8207112A SE 8207112 A SE8207112 A SE 8207112A SE 454442 B SE454442 B SE 454442B
Authority
SE
Sweden
Prior art keywords
hydrogen
equivalents
anisanilide
pyridylacetyl
methyl
Prior art date
Application number
SE8207112A
Other languages
English (en)
Swedish (sv)
Other versions
SE8207112D0 (sv
SE8207112L (sv
Inventor
G D Madding
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of SE8207112D0 publication Critical patent/SE8207112D0/xx
Publication of SE8207112L publication Critical patent/SE8207112L/xx
Publication of SE454442B publication Critical patent/SE454442B/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/44Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
    • C07D213/46Oxygen atoms
    • C07D213/50Ketonic radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/26Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SE8207112A 1981-12-14 1982-12-13 Forfarande for framstellning av 4-metoxi-2'-(2-(1-metyl-2-piperidyl)etyl)-bensamid(enkainid) och 2-(2-pyridylacetyl)-p-anisanilid som mellanprodukt SE454442B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/330,298 US4394507A (en) 1981-12-14 1981-12-14 Process for production of encainide

Publications (3)

Publication Number Publication Date
SE8207112D0 SE8207112D0 (sv) 1982-12-13
SE8207112L SE8207112L (sv) 1983-06-15
SE454442B true SE454442B (sv) 1988-05-02

Family

ID=23289147

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8207112A SE454442B (sv) 1981-12-14 1982-12-13 Forfarande for framstellning av 4-metoxi-2'-(2-(1-metyl-2-piperidyl)etyl)-bensamid(enkainid) och 2-(2-pyridylacetyl)-p-anisanilid som mellanprodukt

Country Status (16)

Country Link
US (1) US4394507A (ko)
JP (1) JPS6058231B2 (ko)
KR (1) KR890000419B1 (ko)
AT (1) AT378182B (ko)
CA (1) CA1213282A (ko)
CH (1) CH655101A5 (ko)
DK (1) DK156648C (ko)
ES (2) ES517996A0 (ko)
FI (1) FI76561C (ko)
GR (1) GR77107B (ko)
HU (1) HU186190B (ko)
IT (1) IT1149399B (ko)
NL (1) NL8204775A (ko)
PT (1) PT75980B (ko)
SE (1) SE454442B (ko)
YU (1) YU44035B (ko)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4675409A (en) * 1986-02-25 1987-06-23 Bristol-Myers Company Process for the preparation of encainide
US4800226A (en) * 1986-02-25 1989-01-24 Bristol-Myers Company Process intermediate for the preparation of encainide

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2317303A (en) * 1940-12-07 1943-04-20 Merck & Co Inc Heterocyclic nitrogen containing compounds, and processes for making the same
US3931195A (en) * 1971-03-03 1976-01-06 Mead Johnson & Company Substituted piperidines
CA961038A (en) * 1971-03-03 1975-01-14 Joseph L. Minielli Substituted piperidines
US4064254A (en) * 1971-03-03 1977-12-20 Mead Johnson & Company Substituted piperidines therapeutic process and compositions
US4000143A (en) * 1971-03-03 1976-12-28 Mead Johnson & Company Substituted piperidines
SE7607114L (sv) * 1976-06-22 1977-12-23 Bofors Ab Sett att framstella hydrokloriden av n-metylpiperidin-2-karbonsyra-2,6-xyllidid

Also Published As

Publication number Publication date
YU271082A (en) 1985-03-20
SE8207112D0 (sv) 1982-12-13
DK156648B (da) 1989-09-18
KR840002355A (ko) 1984-06-25
CA1213282A (en) 1986-10-28
ES8506274A1 (es) 1985-07-01
ATA454082A (de) 1984-11-15
CH655101A5 (de) 1986-03-27
FI824234L (fi) 1983-06-15
US4394507A (en) 1983-07-19
YU44035B (en) 1990-02-28
IT8249608A0 (it) 1982-12-02
ES530218A0 (es) 1985-07-01
FI76561C (fi) 1988-11-10
GR77107B (ko) 1984-09-06
ES8405767A1 (es) 1984-06-16
PT75980A (en) 1983-01-01
JPS58105963A (ja) 1983-06-24
FI76561B (fi) 1988-07-29
SE8207112L (sv) 1983-06-15
AT378182B (de) 1985-06-25
IT1149399B (it) 1986-12-03
PT75980B (en) 1985-12-20
NL8204775A (nl) 1983-07-01
KR890000419B1 (ko) 1989-03-17
FI824234A0 (fi) 1982-12-09
HU186190B (en) 1985-06-28
DK551582A (da) 1983-06-15
ES517996A0 (es) 1984-06-16
DK156648C (da) 1990-03-05
JPS6058231B2 (ja) 1985-12-19

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