SE442867B - Forfarande for framstellning av karbamidderivat - Google Patents

Forfarande for framstellning av karbamidderivat

Info

Publication number
SE442867B
SE442867B SE7804596A SE7804596A SE442867B SE 442867 B SE442867 B SE 442867B SE 7804596 A SE7804596 A SE 7804596A SE 7804596 A SE7804596 A SE 7804596A SE 442867 B SE442867 B SE 442867B
Authority
SE
Sweden
Prior art keywords
butyl
urea
isoxazolyl
process according
reaction
Prior art date
Application number
SE7804596A
Other languages
English (en)
Swedish (sv)
Other versions
SE7804596L (sv
Inventor
Y Makisumi
T Sasatani
A Murabayashi
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of SE7804596L publication Critical patent/SE7804596L/xx
Publication of SE442867B publication Critical patent/SE442867B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/14—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D277/82—Nitrogen atoms
SE7804596A 1977-04-28 1978-04-21 Forfarande for framstellning av karbamidderivat SE442867B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP52049629A JPS6033109B2 (ja) 1977-04-28 1977-04-28 尿素誘導体の合成法

Publications (2)

Publication Number Publication Date
SE7804596L SE7804596L (sv) 1978-10-29
SE442867B true SE442867B (sv) 1986-02-03

Family

ID=12836505

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7804596A SE442867B (sv) 1977-04-28 1978-04-21 Forfarande for framstellning av karbamidderivat

Country Status (25)

Country Link
US (1) US4183856A (nl)
JP (1) JPS6033109B2 (nl)
AR (1) AR225666A1 (nl)
AU (1) AU513688B2 (nl)
BE (1) BE866581A (nl)
BG (1) BG33278A3 (nl)
BR (1) BR7802618A (nl)
CA (1) CA1093081A (nl)
CH (1) CH633542A5 (nl)
CS (1) CS198297B2 (nl)
DD (1) DD135905A5 (nl)
DE (1) DE2818947A1 (nl)
DK (1) DK144011C (nl)
ES (1) ES468897A1 (nl)
FR (1) FR2388802A1 (nl)
GB (1) GB1572976A (nl)
HU (1) HU176881B (nl)
IE (1) IE46769B1 (nl)
IL (1) IL54468A0 (nl)
IT (1) IT1111465B (nl)
NL (1) NL183513C (nl)
PL (1) PL110681B1 (nl)
SE (1) SE442867B (nl)
SU (1) SU1091853A3 (nl)
YU (1) YU40334B (nl)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8422461D0 (en) * 1984-09-05 1984-10-10 Wyeth John & Brother Ltd Pyridine derivatives
US4808722A (en) * 1985-10-31 1989-02-28 Fmc Corporation Pyridinylurea N-oxide compounds and agricultural uses
DE59005183D1 (de) * 1989-11-10 1994-05-05 Agrolinz Agrarchemikalien Verfahren zur Herstellung reiner, unsymmetrisch disubstituierter Harnstoffe.
DE3940261A1 (de) * 1989-12-06 1991-06-13 Agrolinz Agrarchemikalien Muen Verfahren zur herstellung reiner, unsymmetrisch disubstituierter harnstoffe
EP1458382A1 (en) * 2001-12-21 2004-09-22 Novo Nordisk A/S Amide derivatives as gk activators
KR101116627B1 (ko) * 2002-06-27 2012-10-09 노보 노르디스크 에이/에스 치료제로서 아릴 카르보닐 유도체
MXPA06007667A (es) * 2004-01-06 2006-09-01 Novo Nordisk As Heteroaril-ureas y su uso como activadores de glucocinasa.
ATE547396T1 (de) * 2005-07-08 2012-03-15 Novo Nordisk As Dicycloalkylcarbamoyl-harnstoffe als glucokinase- aktivatoren
KR20080024211A (ko) * 2005-07-08 2008-03-17 노보 노르디스크 에이/에스 디시클로알킬 우레아 글루코키나제 활성제
AU2006268589B2 (en) 2005-07-14 2011-09-29 Vtv Therapeutics Llc Urea glucokinase activators
EP2118083A1 (en) * 2007-01-09 2009-11-18 Novo Nordisk A/S Urea glucokinase activators
AU2008204530B2 (en) * 2007-01-11 2013-08-01 Vtv Therapeutics Llc Urea glucokinase activators
CN112040945A (zh) 2018-06-12 2020-12-04 Vtv治疗有限责任公司 葡萄糖激酶激活剂与胰岛素或胰岛素类似物组合的治疗用途

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2755285A (en) * 1956-07-17 I-xsubstituted
US2756135A (en) * 1955-07-13 1956-07-24 Du Pont 1-methyl-3-(2-benzothiazolyl)-ureas and their use as herbicides
DE1209801B (de) * 1963-05-11 1966-01-27 Bayer Ag Unkrautbekaempfung in Rueben
US3293257A (en) * 1964-09-14 1966-12-20 United States Borax Chem Pyridyl urea compounds
FR1533184A (fr) * 1965-04-06 1968-07-19 Pechiney Saint Gobain Dérivés du thiazole
DE1620448C3 (de) * 1965-05-08 1974-08-29 Schering Ag, 1000 Berlin Und 4619 Bergkamen Harnstoff- bzw. Thioharnstoffderivate des 3-Methylisothiazols
US3622593A (en) * 1967-08-09 1971-11-23 Fmc Corp 1,1-dimethyl-3-(isothiazol-5-yl)urea
US3547940A (en) * 1967-10-31 1970-12-15 Du Pont Substituted ureido isoxazoles
GB1266769A (nl) * 1969-08-15 1972-03-15
JPS5031039A (nl) * 1973-07-27 1975-03-27
US4062861A (en) * 1973-07-27 1977-12-13 Shionogi & Co., Ltd. 3-Isoxazolylurea derivatives
US4013706A (en) * 1973-11-14 1977-03-22 Sucreries Du Soissonnais Et Compagnie Sucriere Derivatives of substituted urea, acyl ureas, and sulphonyl ureas, and a process for producing the same
US4046770A (en) * 1974-08-30 1977-09-06 Eli Lilly And Company N-(6-acyloxybenzothiazol-2-yl)-N'-phenyl (or substituted phenyl)ureas
JPS5810361B2 (ja) * 1974-10-04 1983-02-25 塩野義製薬株式会社 ３−アルチルイソオキサゾ−ル系除草剤

Also Published As

Publication number Publication date
DK144011C (da) 1982-04-26
SE7804596L (sv) 1978-10-29
IE780707L (en) 1978-10-28
PL110681B1 (en) 1980-07-31
BR7802618A (pt) 1979-04-03
NL7804550A (nl) 1978-10-31
BE866581A (fr) 1978-08-14
CA1093081A (en) 1981-01-06
ES468897A1 (es) 1978-11-16
IT1111465B (it) 1986-01-13
YU103778A (en) 1982-10-31
AU513688B2 (en) 1980-12-18
NL183513B (nl) 1988-06-16
DE2818947A1 (de) 1978-11-02
IT7867959A0 (it) 1978-04-27
JPS6033109B2 (ja) 1985-08-01
SU1091853A3 (ru) 1984-05-07
DK180378A (da) 1978-10-29
FR2388802A1 (fr) 1978-11-24
AR225666A1 (es) 1982-04-15
HU176881B (en) 1981-05-28
IE46769B1 (en) 1983-09-21
GB1572976A (en) 1980-08-13
CS198297B2 (en) 1980-05-30
PL206450A1 (pl) 1979-03-26
BG33278A3 (en) 1983-01-14
YU40334B (en) 1985-12-31
NL183513C (nl) 1988-11-16
DE2818947C2 (nl) 1991-08-22
JPS53135972A (en) 1978-11-28
FR2388802B1 (nl) 1980-04-04
DK144011B (da) 1981-11-16
IL54468A0 (en) 1978-07-31
AU3546878A (en) 1979-11-01
DD135905A5 (de) 1979-06-06
US4183856A (en) 1980-01-15
CH633542A5 (de) 1982-12-15

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