SE440352B - 4-(kinolinylaminobensoyl)piperaziner - Google Patents
4-(kinolinylaminobensoyl)piperazinerInfo
- Publication number
- SE440352B SE440352B SE7903820A SE7903820A SE440352B SE 440352 B SE440352 B SE 440352B SE 7903820 A SE7903820 A SE 7903820A SE 7903820 A SE7903820 A SE 7903820A SE 440352 B SE440352 B SE 440352B
- Authority
- SE
- Sweden
- Prior art keywords
- amino
- benzoyl
- quinolinyl
- piperazine
- trifluoromethyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/42—Nitrogen atoms attached in position 4
- C07D215/44—Nitrogen atoms attached in position 4 with aryl radicals attached to said nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/903,082 US4167567A (en) | 1978-05-05 | 1978-05-05 | Antihypertensive 4-aminoquinolines |
Publications (2)
Publication Number | Publication Date |
---|---|
SE7903820L SE7903820L (sv) | 1979-11-06 |
SE440352B true SE440352B (sv) | 1985-07-29 |
Family
ID=25416910
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE7903820A SE440352B (sv) | 1978-05-05 | 1979-05-02 | 4-(kinolinylaminobensoyl)piperaziner |
Country Status (16)
Country | Link |
---|---|
US (1) | US4167567A (it) |
JP (1) | JPS54145683A (it) |
AU (1) | AU522635B2 (it) |
BE (1) | BE876039A (it) |
CA (1) | CA1082707A (it) |
CH (1) | CH642964A5 (it) |
DE (1) | DE2914492A1 (it) |
ES (1) | ES480190A1 (it) |
FR (1) | FR2424913A1 (it) |
GB (1) | GB2021567B (it) |
HK (1) | HK60085A (it) |
IT (1) | IT1192349B (it) |
NL (1) | NL7902907A (it) |
SE (1) | SE440352B (it) |
SG (1) | SG38285G (it) |
ZA (1) | ZA791809B (it) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8424979D0 (en) * | 1984-10-03 | 1984-11-07 | Wyeth John & Brother Ltd | Benzenesulphonamide derivatives |
PH22302A (en) * | 1985-02-11 | 1988-07-22 | Fujisawa Pharmaceutical Co | Piperidine compounds |
GB8505430D0 (en) * | 1985-03-02 | 1985-04-03 | Wyeth John & Brother Ltd | Benzamide derivatives |
WO1986005489A1 (en) * | 1985-03-13 | 1986-09-25 | The Upjohn Company | Process for 4-amino quinolines |
US5212182A (en) * | 1990-10-03 | 1993-05-18 | American Home Products Corpooration | Substituted quinolinyl- and naphthalenylbenzamides or benzylamines and related compounds useful as analgesics |
US5438064A (en) * | 1991-12-23 | 1995-08-01 | American Home Products Corporation | Derivatives of 4-anilinoquinoline-3-carboxamide as analgesic agents |
IL115420A0 (en) | 1994-09-26 | 1995-12-31 | Zeneca Ltd | Aminoheterocyclic derivatives |
GB9516709D0 (en) * | 1995-08-15 | 1995-10-18 | Zeneca Ltd | Medicament |
US6313127B1 (en) | 1996-02-02 | 2001-11-06 | Zeneca Limited | Heterocyclic compounds useful as pharmaceutical agents |
GB9602166D0 (en) | 1996-02-02 | 1996-04-03 | Zeneca Ltd | Aminoheterocyclic derivatives |
CZ45699A3 (cs) * | 1996-08-14 | 1999-05-12 | Zeneca Limited | Substituované deriváty pyrimidinu, způsob jejich přípravy a farmaceutický prostředek, který je obsahuje |
UA56197C2 (uk) | 1996-11-08 | 2003-05-15 | Зенека Лімітед | Гетероциклічні похідні |
US6440972B1 (en) | 1997-02-13 | 2002-08-27 | Zeneca Limited | Heterocyclic compounds useful as oxido-squalene cyclase inhibitors |
DE69815509T2 (de) | 1997-02-13 | 2004-05-13 | Astrazeneca Ab | Heterozyklische verbindungen die als oxido-squalen-zyklase-inhibitoren anwendung finden |
GB9715895D0 (en) | 1997-07-29 | 1997-10-01 | Zeneca Ltd | Heterocyclic compounds |
US5922203A (en) * | 1997-10-07 | 1999-07-13 | Hydranautics | Amine monomers and their use in preparing interfacially synthesized membranes for reverse osmosis and nanofiltration |
GB9902989D0 (en) | 1999-02-11 | 1999-03-31 | Zeneca Ltd | Heterocyclic derivatives |
US6464873B1 (en) | 1999-06-15 | 2002-10-15 | Hydranautics | Interfacially polymerized, bipiperidine-polyamide membranes for reverse osmosis and/or nanofiltration and process for making the same |
US7842696B2 (en) * | 2007-06-21 | 2010-11-30 | Forest Laboratories Holdings Limited | Piperazine derivatives as inhibitors of stearoyl-CoA desaturase |
US9795928B2 (en) | 2014-06-24 | 2017-10-24 | Nano And Advanced Materials Institute Limited | Stepwise interfacial polymerization technique with different reagent solution designs to prepare hollow fiber nanofiltration membrane composites |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3362956A (en) * | 1965-08-19 | 1968-01-09 | Sterling Drug Inc | 1-[(heterocyclyl)-lower-alkyl]-4-substituted-piperazines |
BE754586A (fr) * | 1969-08-08 | 1971-02-08 | Upjohn Co | Preparations pharmaceutiques a base de p-(4-quinolylamino) benzamide etleur utilisation |
ZA742410B (en) * | 1973-05-04 | 1975-04-30 | Upjohn Co | A new chemical process for preparing 2-,3-and 4-(4-quinolyl)-aminobenzamides |
ZA743269B (en) * | 1973-06-15 | 1975-05-28 | Upjohn Co | Anti-hypertensive compounds |
US4025629A (en) * | 1974-01-07 | 1977-05-24 | The Upjohn Company | P-(trifluoromethylquinolylamino)benzamides, pharmaceutical dosage forms and method of treatment |
-
1978
- 1978-05-05 US US05/903,082 patent/US4167567A/en not_active Expired - Lifetime
-
1979
- 1979-03-29 CA CA324,413A patent/CA1082707A/en not_active Expired
- 1979-04-10 DE DE19792914492 patent/DE2914492A1/de not_active Ceased
- 1979-04-12 NL NL7902907A patent/NL7902907A/xx not_active Application Discontinuation
- 1979-04-17 ZA ZA791809A patent/ZA791809B/xx unknown
- 1979-04-23 IT IT22086/79A patent/IT1192349B/it active
- 1979-04-26 GB GB7914583A patent/GB2021567B/en not_active Expired
- 1979-05-02 AU AU46676/79A patent/AU522635B2/en not_active Ceased
- 1979-05-02 JP JP5356479A patent/JPS54145683A/ja active Pending
- 1979-05-02 SE SE7903820A patent/SE440352B/sv not_active IP Right Cessation
- 1979-05-03 ES ES480190A patent/ES480190A1/es not_active Expired
- 1979-05-04 FR FR7911265A patent/FR2424913A1/fr active Granted
- 1979-05-04 BE BE0/194991A patent/BE876039A/xx not_active IP Right Cessation
- 1979-05-04 CH CH422879A patent/CH642964A5/de not_active IP Right Cessation
-
1985
- 1985-05-23 SG SG382/85A patent/SG38285G/en unknown
- 1985-08-08 HK HK600/85A patent/HK60085A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
HK60085A (en) | 1985-08-16 |
DE2914492A1 (de) | 1979-11-08 |
US4167567A (en) | 1979-09-11 |
FR2424913B1 (it) | 1983-05-20 |
GB2021567A (en) | 1979-12-05 |
JPS54145683A (en) | 1979-11-14 |
SG38285G (en) | 1985-11-15 |
CA1082707A (en) | 1980-07-29 |
BE876039A (fr) | 1979-11-05 |
IT7922086A0 (it) | 1979-04-23 |
NL7902907A (nl) | 1979-11-07 |
ZA791809B (en) | 1980-05-28 |
AU522635B2 (en) | 1982-06-17 |
CH642964A5 (de) | 1984-05-15 |
ES480190A1 (es) | 1980-02-01 |
SE7903820L (sv) | 1979-11-06 |
GB2021567B (en) | 1982-09-02 |
FR2424913A1 (fr) | 1979-11-30 |
IT1192349B (it) | 1988-03-31 |
AU4667679A (en) | 1979-11-08 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
SE440352B (sv) | 4-(kinolinylaminobensoyl)piperaziner | |
SU1340589A3 (ru) | Способ получени 2-(4-замещенных пиперазино-4-амино-6,7-диметокси)хинолинов или их гидрохлоридов | |
KR100443850B1 (ko) | 헤테로시클릭 화합물의 도파민-d3 리간드로서의 용도 | |
EP0079545B1 (en) | Benzimidazole derivatives, process for the preparation thereof and pharmaceutical composition containing the same | |
US4159331A (en) | Antihypertensive 4-aminoquinolines | |
EP0017484B1 (en) | 2-imidazoline derivatives, process for the preparation thereof and the pharmaceutical composition of the same | |
HU188852B (en) | Process for producing thiazolidine derivatives active against gastric ulcer and intestinal ulcer | |
US4166853A (en) | Antihypertensive 7-trifluoromethyl-4-aminoquinolones | |
US4315940A (en) | Antidiabetic 1-piperidine-sulfonylureas | |
RU2245334C2 (ru) | Производные пиперазинилалкилтиопиримидина, содержащие их фармацевтические композиции и способ получения | |
EP0228959B1 (en) | Aminostyryl compound, leukotriene antagonistic composition containing the same as effective ingredients and method of antagonizing srs by employing the same | |
EP0104614B1 (en) | Phenylpiperazine derivatives and process for producing the same | |
JPS58206588A (ja) | 抗潰瘍性2−グアニジノ−4−(2−置換−アミノ−4−イミダゾリル)チアゾ−ル類およびそれらの製造方法 | |
US3998953A (en) | 1,3,7-Trisubstitued xanthine peripheral vasodilators | |
EP0027895A1 (en) | 1-(2-(Alkyl and arylsulfonyl)-2-propenyl and propyl) substituted piperidines and pharmaceutical and antimicrobial compositions comprising the same | |
US4128643A (en) | 4-Quinazolinyl-guanidines | |
JPH01157979A (ja) | 1―アシル―3―[4―(2―ピリミジニル)―1―ピペラジニル]プロパン類 | |
US4140775A (en) | Piperazino methyl phenyl aminoquinolines | |
CA1285945C (en) | N-¬¬¬1-(2)naphthylenemethyl or quinol-6-ylmethyl)-4- piperidinyl|amino|-carbonyl|-6-quinolinecarboxamide compounds | |
US3470185A (en) | 2-(piperazino)methyl-2,3-dihydro-benzofurans | |
US2837522A (en) | Substituted alkylenedipiperazines | |
NO874958L (no) | Analogifremgangsmaate for fremstilling av 1-aryloksy-3-amino-2-propanoler. | |
US4997833A (en) | Aryloxy-aminoalkanes, and antihypertensive use thereof | |
KR900001188B1 (ko) | 치환된 페닐알킬(피페라지닐 또는 호모피페라지닐)알킬-티올 및-티오카바메이트의 제조방법 | |
EP0187639A1 (en) | Novel piperazine derivatives, processes for production thereof, and pharmaceutical compositions comprising said compounds as active ingredient |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
NUG | Patent has lapsed |
Ref document number: 7903820-4 Effective date: 19890525 Format of ref document f/p: F |