SE421797B - Forfarande for framstellning av 6-(2-aryl-2-(imidoylamino)-acetamido)-penicillansyra - Google Patents

Forfarande for framstellning av 6-(2-aryl-2-(imidoylamino)-acetamido)-penicillansyra

Info

Publication number
SE421797B
SE421797B SE7400501A SE7400501A SE421797B SE 421797 B SE421797 B SE 421797B SE 7400501 A SE7400501 A SE 7400501A SE 7400501 A SE7400501 A SE 7400501A SE 421797 B SE421797 B SE 421797B
Authority
SE
Sweden
Prior art keywords
imidoylamino
acetamido
aryl
preparing
penicillanic acid
Prior art date
Application number
SE7400501A
Other languages
English (en)
Other versions
SE7400501L (sv
Inventor
E S Hamanaka
J G Stam
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/424,891 external-priority patent/US3951952A/en
Application filed by Pfizer filed Critical Pfizer
Publication of SE7400501L publication Critical patent/SE7400501L/xx
Publication of SE421797B publication Critical patent/SE421797B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/881—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with a hydrogen atom or an unsubstituted hydrocarbon radical, attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/429—Thiazoles condensed with heterocyclic ring systems
    • A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SE7400501A 1973-12-14 1974-01-15 Forfarande for framstellning av 6-(2-aryl-2-(imidoylamino)-acetamido)-penicillansyra SE421797B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/424,891 US3951952A (en) 1972-08-02 1973-12-14 Broad spectrum antibiotics

Publications (2)

Publication Number Publication Date
SE7400501L SE7400501L (sv) 1975-06-16
SE421797B true SE421797B (sv) 1982-02-01

Family

ID=23684297

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7400501A SE421797B (sv) 1973-12-14 1974-01-15 Forfarande for framstellning av 6-(2-aryl-2-(imidoylamino)-acetamido)-penicillansyra

Country Status (31)

Country Link
US (1) US4073783A (sv)
JP (3) JPS5089393A (sv)
KR (1) KR780000354B1 (sv)
AR (1) AR202472A1 (sv)
AT (1) AT326821B (sv)
BE (1) BE810266R (sv)
BG (1) BG24955A3 (sv)
CA (1) CA1023348A (sv)
CH (1) CH596218A5 (sv)
CS (1) CS194205B2 (sv)
DD (1) DD113008A6 (sv)
DE (1) DE2403512C2 (sv)
DK (1) DK150856C (sv)
EG (1) EG11025A (sv)
ES (1) ES422732A2 (sv)
FI (1) FI62840C (sv)
FR (1) FR2254310B2 (sv)
GB (1) GB1462421A (sv)
HU (1) HU167158B (sv)
IE (1) IE39964B1 (sv)
IL (1) IL44033A (sv)
IN (1) IN139932B (sv)
LU (1) LU69290A1 (sv)
NL (1) NL7401174A (sv)
NO (1) NO145794C (sv)
PH (1) PH15634A (sv)
RO (1) RO67596A (sv)
SE (1) SE421797B (sv)
SU (1) SU609468A3 (sv)
YU (1) YU22674A (sv)
ZA (1) ZA74509B (sv)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4024130A (en) * 1975-03-31 1977-05-17 Pfizer Inc. Process for the manufacture of alkali metal salts of 6-[2-phenyl-2-(imidoylaminoalkanoylamino)acetamido]penicillanic acids
US4168266A (en) * 1978-05-30 1979-09-18 E. R. Squibb & Sons, Inc. 6-[[[(2-Cyanomethyl)amino]-1,2-dioxoethyl]-amino]acyl penicillins
CN102190598B (zh) * 2011-03-28 2014-01-29 浙江工业大学 环丙烷肟酯衍生物及其制备方法和用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3634405A (en) * 1969-08-01 1972-01-11 Bristol Myers Co Synthetic penicillins
US3579501A (en) * 1969-08-22 1971-05-18 Bristol Myers Co 6-(alpha-(3 - guanyl - 1 - ureido)phenyl- or thienyl-acetamido)penicillanic acids
DE2104580C3 (de) * 1971-02-01 1981-04-02 Bayer Ag, 5090 Leverkusen Acylureidopenicilline
BE790441A (fr) * 1971-10-23 1973-04-24 Bayer Ag Nouvelles penicillines, leur procede de preparation et medicament les contenant
BE794886A (fr) * 1972-02-22 1973-08-02 Pfizer Acides 6-(alpha-(omega-guanidinoalcanoylamino)acylamino)-penicillaniques
US3838153A (en) * 1972-05-16 1974-09-24 Pfizer 6-(alpha-(guanylureidoalkanoylamino)aracylamino)penicillanic acids

Also Published As

Publication number Publication date
DD113008A6 (sv) 1975-05-12
DK150856B (da) 1987-07-06
US4073783A (en) 1978-02-14
FI62840B (fi) 1982-11-30
AU6463674A (en) 1975-07-17
GB1462421A (en) 1977-01-26
JPS6043072B2 (ja) 1985-09-26
SU609468A3 (ru) 1978-05-30
DK45574A (sv) 1975-08-11
NO145794B (no) 1982-02-22
NO740281L (sv) 1975-07-14
LU69290A1 (sv) 1974-09-25
IN139932B (sv) 1976-08-21
ZA74509B (en) 1974-12-24
ES422732A2 (es) 1977-07-01
JPS5089393A (sv) 1975-07-17
IE39964B1 (en) 1979-02-14
DE2403512A1 (de) 1975-06-19
IL44033A (en) 1977-10-31
JPS6048519B2 (ja) 1985-10-28
BE810266R (fr) 1974-07-29
FI62840C (fi) 1983-03-10
DK150856C (da) 1987-11-16
AR202472A1 (es) 1975-06-13
RO67596A (ro) 1980-02-15
DE2403512C2 (de) 1983-01-13
SE7400501L (sv) 1975-06-16
YU22674A (en) 1982-02-28
BG24955A3 (en) 1978-06-15
KR780000354B1 (en) 1978-09-16
FR2254310A2 (sv) 1975-07-11
PH15634A (en) 1983-03-11
IE39964L (en) 1975-06-14
CH596218A5 (sv) 1978-03-15
FR2254310B2 (sv) 1977-04-22
CS194205B2 (en) 1979-11-30
AT326821B (de) 1975-12-29
EG11025A (en) 1976-11-30
NL7401174A (nl) 1975-06-17
ATA73374A (de) 1975-03-15
HU167158B (sv) 1975-08-28
JPS5756483A (en) 1982-04-05
CA1023348A (en) 1977-12-27
NO145794C (no) 1982-06-09
FI740226A0 (sv) 1975-06-15
JPS5874688A (ja) 1983-05-06

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