BE810266R - Acides 6-(alpha-(amidino- et imidoylaminoalcanoylamino)-aracylamino) penicillaniques et leur preparation - Google Patents

Acides 6-(alpha-(amidino- et imidoylaminoalcanoylamino)-aracylamino) penicillaniques et leur preparation

Info

Publication number
BE810266R
BE810266R BE1005676A BE1005676A BE810266R BE 810266 R BE810266 R BE 810266R BE 1005676 A BE1005676 A BE 1005676A BE 1005676 A BE1005676 A BE 1005676A BE 810266 R BE810266 R BE 810266R
Authority
BE
Belgium
Prior art keywords
imidoylaminoalcanoylamino
aracylamino
amidino
alpha
preparation
Prior art date
Application number
BE1005676A
Other languages
English (en)
French (fr)
Inventor
E S Hamanaka
J G Stam
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/424,891 external-priority patent/US3951952A/en
Application filed filed Critical
Application granted granted Critical
Publication of BE810266R publication Critical patent/BE810266R/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/881—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with a hydrogen atom or an unsubstituted hydrocarbon radical, attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/429—Thiazoles condensed with heterocyclic ring systems
    • A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE1005676A 1973-12-14 1974-01-29 Acides 6-(alpha-(amidino- et imidoylaminoalcanoylamino)-aracylamino) penicillaniques et leur preparation BE810266R (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/424,891 US3951952A (en) 1972-08-02 1973-12-14 Broad spectrum antibiotics

Publications (1)

Publication Number Publication Date
BE810266R true BE810266R (fr) 1974-07-29

Family

ID=23684297

Family Applications (1)

Application Number Title Priority Date Filing Date
BE1005676A BE810266R (fr) 1973-12-14 1974-01-29 Acides 6-(alpha-(amidino- et imidoylaminoalcanoylamino)-aracylamino) penicillaniques et leur preparation

Country Status (31)

Country Link
US (1) US4073783A (xx)
JP (3) JPS5089393A (xx)
KR (1) KR780000354B1 (xx)
AR (1) AR202472A1 (xx)
AT (1) AT326821B (xx)
BE (1) BE810266R (xx)
BG (1) BG24955A3 (xx)
CA (1) CA1023348A (xx)
CH (1) CH596218A5 (xx)
CS (1) CS194205B2 (xx)
DD (1) DD113008A6 (xx)
DE (1) DE2403512C2 (xx)
DK (1) DK150856C (xx)
EG (1) EG11025A (xx)
ES (1) ES422732A2 (xx)
FI (1) FI62840C (xx)
FR (1) FR2254310B2 (xx)
GB (1) GB1462421A (xx)
HU (1) HU167158B (xx)
IE (1) IE39964B1 (xx)
IL (1) IL44033A (xx)
IN (1) IN139932B (xx)
LU (1) LU69290A1 (xx)
NL (1) NL7401174A (xx)
NO (1) NO145794C (xx)
PH (1) PH15634A (xx)
RO (1) RO67596A (xx)
SE (1) SE421797B (xx)
SU (1) SU609468A3 (xx)
YU (1) YU22674A (xx)
ZA (1) ZA74509B (xx)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4024130A (en) * 1975-03-31 1977-05-17 Pfizer Inc. Process for the manufacture of alkali metal salts of 6-[2-phenyl-2-(imidoylaminoalkanoylamino)acetamido]penicillanic acids
CN102190598A (zh) * 2011-03-28 2011-09-21 浙江工业大学 环丙烷肟酯衍生物及其制备方法和用途

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4168266A (en) * 1978-05-30 1979-09-18 E. R. Squibb & Sons, Inc. 6-[[[(2-Cyanomethyl)amino]-1,2-dioxoethyl]-amino]acyl penicillins

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3634405A (en) * 1969-08-01 1972-01-11 Bristol Myers Co Synthetic penicillins
US3579501A (en) * 1969-08-22 1971-05-18 Bristol Myers Co 6-(alpha-(3 - guanyl - 1 - ureido)phenyl- or thienyl-acetamido)penicillanic acids
DE2104580C3 (de) * 1971-02-01 1981-04-02 Bayer Ag, 5090 Leverkusen Acylureidopenicilline
BE790441A (fr) * 1971-10-23 1973-04-24 Bayer Ag Nouvelles penicillines, leur procede de preparation et medicament les contenant
BE794886A (fr) * 1972-02-22 1973-08-02 Pfizer Acides 6-(alpha-(omega-guanidinoalcanoylamino)acylamino)-penicillaniques
US3838153A (en) * 1972-05-16 1974-09-24 Pfizer 6-(alpha-(guanylureidoalkanoylamino)aracylamino)penicillanic acids

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4024130A (en) * 1975-03-31 1977-05-17 Pfizer Inc. Process for the manufacture of alkali metal salts of 6-[2-phenyl-2-(imidoylaminoalkanoylamino)acetamido]penicillanic acids
CN102190598A (zh) * 2011-03-28 2011-09-21 浙江工业大学 环丙烷肟酯衍生物及其制备方法和用途
CN102190598B (zh) * 2011-03-28 2014-01-29 浙江工业大学 环丙烷肟酯衍生物及其制备方法和用途

Also Published As

Publication number Publication date
FR2254310A2 (xx) 1975-07-11
NO145794B (no) 1982-02-22
DE2403512C2 (de) 1983-01-13
RO67596A (ro) 1980-02-15
FI62840C (fi) 1983-03-10
JPS5089393A (xx) 1975-07-17
SU609468A3 (ru) 1978-05-30
JPS6043072B2 (ja) 1985-09-26
DE2403512A1 (de) 1975-06-19
YU22674A (en) 1982-02-28
SE7400501L (xx) 1975-06-16
US4073783A (en) 1978-02-14
LU69290A1 (xx) 1974-09-25
FR2254310B2 (xx) 1977-04-22
JPS5756483A (en) 1982-04-05
BG24955A3 (en) 1978-06-15
CS194205B2 (en) 1979-11-30
AT326821B (de) 1975-12-29
JPS6048519B2 (ja) 1985-10-28
DK150856B (da) 1987-07-06
CA1023348A (en) 1977-12-27
DK45574A (xx) 1975-08-11
IN139932B (xx) 1976-08-21
IE39964B1 (en) 1979-02-14
IE39964L (en) 1975-06-14
FI740226A0 (xx) 1975-06-15
SE421797B (sv) 1982-02-01
HU167158B (xx) 1975-08-28
ATA73374A (de) 1975-03-15
PH15634A (en) 1983-03-11
ZA74509B (en) 1974-12-24
EG11025A (en) 1976-11-30
AR202472A1 (es) 1975-06-13
NO740281L (xx) 1975-07-14
IL44033A (en) 1977-10-31
NO145794C (no) 1982-06-09
NL7401174A (nl) 1975-06-17
AU6463674A (en) 1975-07-17
ES422732A2 (es) 1977-07-01
FI62840B (fi) 1982-11-30
JPS5874688A (ja) 1983-05-06
GB1462421A (en) 1977-01-26
DK150856C (da) 1987-11-16
KR780000354B1 (en) 1978-09-16
CH596218A5 (xx) 1978-03-15
DD113008A6 (xx) 1975-05-12

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: PFIZER INC.

Effective date: 19920831