SE378109B - - Google Patents

Info

Publication number
SE378109B
SE378109B SE7206644A SE664472A SE378109B SE 378109 B SE378109 B SE 378109B SE 7206644 A SE7206644 A SE 7206644A SE 664472 A SE664472 A SE 664472A SE 378109 B SE378109 B SE 378109B
Authority
SE
Sweden
Application number
SE7206644A
Inventor
R L Brattsand
K G Claeson
Af Ekenstam B Thuresson
B A Thalen
Original Assignee
Bofors Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20269234&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SE378109(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority to SE7206644A priority Critical patent/SE378109B/xx
Application filed by Bofors Ab filed Critical Bofors Ab
Priority to IL42155A priority patent/IL42155A/en
Priority to ZA732955A priority patent/ZA732955B/xx
Priority to AU55253/73A priority patent/AU487812B2/en
Priority to GB2219473A priority patent/GB1429922A/en
Priority to DE2323215A priority patent/DE2323215C3/de
Priority to CY1013A priority patent/CY1013A/xx
Priority to ES414673A priority patent/ES414673A1/es
Priority to US360051A priority patent/US3929768A/en
Priority to FI731542A priority patent/FI50631C/fi
Priority to YU1291/73A priority patent/YU35896B/xx
Priority to CH699973A priority patent/CH595400A5/xx
Priority to DK277273AA priority patent/DK134783B/da
Priority to DD170888A priority patent/DD104295A5/xx
Priority to AT436573A priority patent/AT328630B/de
Priority to BE131270A priority patent/BE799727A/xx
Priority to SU1923451A priority patent/SU470954A3/ru
Priority to PL1973162650A priority patent/PL87765B1/pl
Priority to CS3590A priority patent/CS178129B2/cs
Priority to NO2059/73A priority patent/NO139640C/no
Priority to HUBO1438A priority patent/HU166680B/hu
Priority to NLAANVRAGE7306978,A priority patent/NL177493C/xx
Priority to CA171,785A priority patent/CA1002938A/en
Priority to FR7318125A priority patent/FR2185405B1/fr
Priority to JP5623373A priority patent/JPS5521760B2/ja
Publication of SE378109B publication Critical patent/SE378109B/xx
Priority to US05/629,389 priority patent/US3983233A/en
Priority to KE2970A priority patent/KE2970A/xx
Priority to HK491/79A priority patent/HK49179A/xx
Priority to NL930025C priority patent/NL930025I1/nl
Priority to NO1994013C priority patent/NO1994013I1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/0026—Oxygen-containing hetero ring cyclic ketals
    • C07J71/0031—Oxygen-containing hetero ring cyclic ketals at positions 16, 17
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SE7206644A 1972-05-19 1972-05-19 SE378109B (fi)

Priority Applications (30)

Application Number Priority Date Filing Date Title
SE7206644A SE378109B (fi) 1972-05-19 1972-05-19
IL42155A IL42155A (en) 1972-05-19 1973-05-01 16alpha,17alpha-alkylidenedioxy-11beta,21-dihydroxy-pregna-1,4-diene-3,20-diones their manufacture and preparations containing same
ZA732955A ZA732955B (en) 1972-05-19 1973-05-01 New steroids,processes for their manufacture and preparations containing same
AU55253/73A AU487812B2 (en) 1972-05-19 1973-05-04 New Steroids, processes for their manufacture and preparations containing same
GB2219473A GB1429922A (en) 1972-05-19 1973-05-09 Steroid acetals processes for their manufacture and preparations containing them
DE2323215A DE2323215C3 (de) 1972-05-19 1973-05-09 Pregna-l,4-dien-ll-ol-3,20-dione, Verfahren zu deren Herstellung und sie enthaltende Arzneimittel
CY1013A CY1013A (en) 1972-05-19 1973-05-09 Steroid acetals, processes for their manufacture and preparations containing them
ES414673A ES414673A1 (es) 1972-05-19 1973-05-11 Procedimiento para preparar esteroides.
FI731542A FI50631C (fi) 1972-05-19 1973-05-14 Menetelmä pregnadieenijohdannaisten valmistamiseksi.
US360051A US3929768A (en) 1972-05-19 1973-05-14 Steroids, processes for their manufacture and preparations containing same
YU1291/73A YU35896B (en) 1972-05-19 1973-05-16 Process for obtaining steroids
CH699973A CH595400A5 (fi) 1972-05-19 1973-05-16
DK277273AA DK134783B (da) 1972-05-19 1973-05-17 Analogifremgangsmåde til fremstilling af 16alfa,17alfa-alkylidendioxypregna-1,4-dien-11beta,21-diol-3,20-dioner.
DD170888A DD104295A5 (fi) 1972-05-19 1973-05-17
BE131270A BE799727A (fr) 1972-05-19 1973-05-18 Nouveaux steroides physiologiquement actifs, et procede pour leur preparation.
AT436573A AT328630B (de) 1972-05-19 1973-05-18 Verfahren zur herstellung neuer steroide
FR7318125A FR2185405B1 (fi) 1972-05-19 1973-05-18
SU1923451A SU470954A3 (ru) 1972-05-19 1973-05-18 Способ получени производных кортикостероидов
PL1973162650A PL87765B1 (fi) 1972-05-19 1973-05-18
CS3590A CS178129B2 (fi) 1972-05-19 1973-05-18
NO2059/73A NO139640C (no) 1972-05-19 1973-05-18 Analogifremgangsmaate for fremstilling av fysiologisk virksomme 16alfa,17alfa-alkylidendioksypregna-1,4-dien-3,20-dioner
HUBO1438A HU166680B (fi) 1972-05-19 1973-05-18
NLAANVRAGE7306978,A NL177493C (nl) 1972-05-19 1973-05-18 Werkwijze voor de bereiding van steroiden en werkwijze ter bereiding van een farmaceutisch preparaat tegen ontstekingen.
CA171,785A CA1002938A (en) 1972-05-19 1973-05-18 Steroids, processes for their manufacture and preparations containing same
JP5623373A JPS5521760B2 (fi) 1972-05-19 1973-05-19
US05/629,389 US3983233A (en) 1972-05-19 1975-11-06 Compositions and method of treating with stereoisomeric mixtures of 2-unsymmetrical 16,17-methylenedioxy steroids
KE2970A KE2970A (en) 1972-05-19 1979-06-20 New steriod acetals, process for their manufacture and preparations containing them
HK491/79A HK49179A (en) 1972-05-19 1979-07-19 New steroid acetals, processes for their manufacture and preparations containing them
NL930025C NL930025I1 (nl) 1972-05-19 1993-04-13 Werkwijze voor de bereiding van steroïden en werkwijze ter bereiding van een farmaceutisch preparaattegen ontstekingen
NO1994013C NO1994013I1 (no) 1972-05-19 1994-08-31 Budenosid/ 16¿, 17¿-alkyldendioksypregna-1,4-dien-3,20-dioner

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE7206644A SE378109B (fi) 1972-05-19 1972-05-19

Publications (1)

Publication Number Publication Date
SE378109B true SE378109B (fi) 1975-08-18

Family

ID=20269234

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7206644A SE378109B (fi) 1972-05-19 1972-05-19

Country Status (26)

Country Link
US (2) US3929768A (fi)
JP (1) JPS5521760B2 (fi)
AT (1) AT328630B (fi)
BE (1) BE799727A (fi)
CA (1) CA1002938A (fi)
CH (1) CH595400A5 (fi)
CS (1) CS178129B2 (fi)
CY (1) CY1013A (fi)
DD (1) DD104295A5 (fi)
DE (1) DE2323215C3 (fi)
DK (1) DK134783B (fi)
ES (1) ES414673A1 (fi)
FI (1) FI50631C (fi)
FR (1) FR2185405B1 (fi)
GB (1) GB1429922A (fi)
HK (1) HK49179A (fi)
HU (1) HU166680B (fi)
IL (1) IL42155A (fi)
KE (1) KE2970A (fi)
NL (2) NL177493C (fi)
NO (2) NO139640C (fi)
PL (1) PL87765B1 (fi)
SE (1) SE378109B (fi)
SU (1) SU470954A3 (fi)
YU (1) YU35896B (fi)
ZA (1) ZA732955B (fi)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0170642A2 (en) * 1984-07-30 1986-02-05 Aktiebolaget Draco Liposomes containing steroid esters
EP0197018A1 (en) * 1985-04-04 1986-10-08 Aktiebolaget Draco 16,17-Acetal-substituted androstane-17-beta-carboxylic-acid esters, process for their preparation and pharmaceutical compound containing them
EP0232690A1 (en) * 1985-12-19 1987-08-19 Aktiebolaget Draco Novel 16,17-acetalsubstituted pregnane-21-oic acid derivatives, process for the preparation thereof and pharmaceutical preparation containing them
US5215979A (en) * 1985-12-19 1993-06-01 Aktiebolaget Draco 16,17-acetalsubstituted pregnane 21-oic acid derivatives

Families Citing this family (136)

* Cited by examiner, † Cited by third party
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SE8004580L (sv) * 1980-06-19 1981-12-20 Draco Ab Farmaceutisk beredning
SE8008524L (sv) * 1980-12-04 1982-06-05 Draco Ab 4-pregnen-derivat, ett forfarande for deras framstellning, beredning och metod for behandling av inflammatoriska tillstand
IT1196142B (it) * 1984-06-11 1988-11-10 Sicor Spa Procedimento per la preparazione di 16,17-acetali di derivati pregnanici e nuovi composti ottenuti
SE8604059D0 (sv) * 1986-09-25 1986-09-25 Astra Pharma Prod A method of controlling the epimeric distribution in the preparation of 16,17-acetals of pregnane derivatives
LV5274A3 (lv) * 1988-02-29 1993-10-10 Richter Gedeon Vegyeszet 22(R,S)-11 beta,21-dihidroksi-16 alpha,17-butilidenbisoksipregna-1,4-dien-3,20-diona iegusanas panemiens
HU203769B (en) * 1989-03-09 1991-09-30 Richter Gedeon Vegyeszet Process for producing new steroide derivatives and pharmaceutical compositions containing them
SE8903219D0 (sv) * 1989-10-02 1989-10-02 Astra Ab Process for the manufacture of budesonide
SE8903914D0 (sv) 1989-11-22 1989-11-22 Draco Ab Oral composition for the treatment of inflammatory bowel diseases
US5643602A (en) * 1989-11-22 1997-07-01 Astra Aktiebolag Oral composition for the treatment of inflammatory bowel disease
GR1001529B (el) * 1990-09-07 1994-03-31 Elmuquimica Farm Sl Μέ?οδος για την λήψη νέων 21-εστέρων της 16-17-ακετάλης της πρ να-1,4-διενο-3,20-διόνης.
SE9100342D0 (sv) * 1991-02-04 1991-02-04 Astra Ab Novel steroid esters
US5888995A (en) * 1991-02-04 1999-03-30 Astra Aktiebolag Steroid esters
SE9100341D0 (sv) * 1991-02-04 1991-02-04 Astra Ab Novel steroids
IE67345B1 (en) * 1991-03-12 1996-03-20 Akzo Nv Low dose dry pharmaceutical preparations
FR2675146A1 (fr) * 1991-04-10 1992-10-16 Roussel Uclaf Nouveaux derives sterouides de la pregna-1,4-diene-3,20-dione, leur preparation, leur application a la preparation de derives 16,17-methylene dioxy substitues et nouveaux intermediaires.
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Cited By (8)

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EP0170642A3 (en) * 1984-07-30 1986-10-29 Aktiebolaget Draco Liposomes containing steroid esters
US4693999A (en) * 1984-07-30 1987-09-15 Aktiebolaget Draco Liposomes containing steroid esters
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EP0355859A1 (en) * 1985-04-04 1990-02-28 Aktiebolaget Draco Process for the preparation of intermediates for 11-beta,16-alpha,17-alpha,21-tetrahydroxypregna-3,20-dione 16-alpha,17-alpha-acetals and 21-esters thereof
US4950659A (en) * 1985-04-04 1990-08-21 Aktiebolaget Draco 16,17-acetalsubstituted androstane-17β-carboxylic acid esters prossessing high binding affinity to the glucocorticosteroid receptor
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US5215979A (en) * 1985-12-19 1993-06-01 Aktiebolaget Draco 16,17-acetalsubstituted pregnane 21-oic acid derivatives

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YU35896B (en) 1981-08-31
NO139640B (no) 1979-01-08
US3929768A (en) 1975-12-30
FI50631B (fi) 1976-02-02
BE799727A (fr) 1973-09-17
GB1429922A (en) 1976-03-31
YU129173A (en) 1981-02-28
AT328630B (de) 1976-03-25
CY1013A (en) 1979-11-23
ZA732955B (en) 1974-04-24
SU470954A3 (ru) 1975-05-15
PL87765B1 (fi) 1976-07-31
JPS4941378A (fi) 1974-04-18
NL177493B (nl) 1985-05-01
DE2323215B2 (de) 1977-08-11
NO139640C (no) 1979-04-18
DE2323215A1 (de) 1973-11-29
HU166680B (fi) 1975-05-28
DD104295A5 (fi) 1974-03-05
US3983233A (en) 1976-09-28
DE2323215C3 (de) 1978-03-30
IL42155A0 (en) 1973-07-30
CS178129B2 (fi) 1977-08-31
CA1002938A (en) 1977-01-04
NL930025I1 (nl) 1993-06-01
FR2185405A1 (fi) 1974-01-04
IL42155A (en) 1977-06-30
JPS5521760B2 (fi) 1980-06-12
NL7306978A (fi) 1973-11-21
DK134783B (da) 1977-01-17
ATA436573A (de) 1975-06-15
NO1994013I1 (no) 1994-08-31
AU5525373A (en) 1974-11-07
FR2185405B1 (fi) 1976-12-31
CH595400A5 (fi) 1978-02-15
KE2970A (en) 1979-07-20
DK134783C (fi) 1977-06-06
HK49179A (en) 1979-07-27
ES414673A1 (es) 1976-07-01
NL177493C (nl) 1985-10-01
FI50631C (fi) 1976-05-10

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