SE8604059D0 - A method of controlling the epimeric distribution in the preparation of 16,17-acetals of pregnane derivatives - Google Patents
A method of controlling the epimeric distribution in the preparation of 16,17-acetals of pregnane derivativesInfo
- Publication number
- SE8604059D0 SE8604059D0 SE8604059A SE8604059A SE8604059D0 SE 8604059 D0 SE8604059 D0 SE 8604059D0 SE 8604059 A SE8604059 A SE 8604059A SE 8604059 A SE8604059 A SE 8604059A SE 8604059 D0 SE8604059 D0 SE 8604059D0
- Authority
- SE
- Sweden
- Prior art keywords
- acetals
- preparation
- controlling
- hydrocarbon solvent
- epimeric distribution
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/0026—Oxygen-containing hetero ring cyclic ketals
- C07J71/0031—Oxygen-containing hetero ring cyclic ketals at positions 16, 17
Priority Applications (13)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE8604059A SE8604059D0 (sv) | 1986-09-25 | 1986-09-25 | A method of controlling the epimeric distribution in the preparation of 16,17-acetals of pregnane derivatives |
US07/096,598 US4925933A (en) | 1986-09-25 | 1987-09-11 | Method of controlling the epimeric distribution in the preparation of 16,17-acetals of pregnane derivatives |
DE8787850282T DE3774987D1 (de) | 1986-09-25 | 1987-09-18 | Verfahren zur kontrolle der epimerischen verteilung in der herstellung von pregnane-16,17-acetal oder ketal derivaten. |
ES198787850282T ES2026576T3 (es) | 1986-09-25 | 1987-09-18 | Un metodo para controlar la distribucion epimera en la preparacion de 16,17-acetales o cetales de derivados de pregnano. |
AT87850282T ATE70066T1 (de) | 1986-09-25 | 1987-09-18 | Verfahren zur kontrolle der epimerischen verteilung in der herstellung von pregnane-16,17- acetal oder ketal derivaten. |
EP87850282A EP0262108B1 (en) | 1986-09-25 | 1987-09-18 | A method of controlling the empimeric distribution in the preparation of 16,17-acetals or ketals of pregnane derivatives |
IL83994A IL83994A (en) | 1986-09-25 | 1987-09-23 | Method of controlling the epimeric distribution in the preparation of 16,17-acetals of pregnane derivatives |
FI874189A FI90345C (sv) | 1986-09-25 | 1987-09-24 | Förfarande för kontroll av epimerdistributionen vid framställning av 16,17-acetaler av pregnanderivat |
KR1019870010561A KR950014460B1 (ko) | 1986-09-25 | 1987-09-24 | 프레그난 유도체의 16, 17-아세탈 또는 케탈의 제조에 있어서 에피머 분배를 조절하는 방법 |
JP62237588A JP2668000B2 (ja) | 1986-09-25 | 1987-09-24 | プレグナン誘導体の16,17−アセタール製造におけるエピマー分配の調整法 |
GR91401949T GR3003332T3 (en) | 1986-09-25 | 1991-12-12 | A method of controlling the empimeric distribution in the preparation of 16,17-acetals or ketals of pregnane derivatives |
HK46194A HK46194A (en) | 1986-09-25 | 1994-05-12 | A method of controlling the empimeric distribution in the preparation of 16,17-acetals or ketals of pregnane derivatives |
CY179195A CY1791A (en) | 1986-09-25 | 1995-10-20 | A method of controlling the empimeric distribution in the preparation of 16,17-acetals or ketals of pregnane derivatives |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE8604059A SE8604059D0 (sv) | 1986-09-25 | 1986-09-25 | A method of controlling the epimeric distribution in the preparation of 16,17-acetals of pregnane derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
SE8604059D0 true SE8604059D0 (sv) | 1986-09-25 |
Family
ID=20365704
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE8604059A SE8604059D0 (sv) | 1986-09-25 | 1986-09-25 | A method of controlling the epimeric distribution in the preparation of 16,17-acetals of pregnane derivatives |
Country Status (13)
Country | Link |
---|---|
US (1) | US4925933A (sv) |
EP (1) | EP0262108B1 (sv) |
JP (1) | JP2668000B2 (sv) |
KR (1) | KR950014460B1 (sv) |
AT (1) | ATE70066T1 (sv) |
CY (1) | CY1791A (sv) |
DE (1) | DE3774987D1 (sv) |
ES (1) | ES2026576T3 (sv) |
FI (1) | FI90345C (sv) |
GR (1) | GR3003332T3 (sv) |
HK (1) | HK46194A (sv) |
IL (1) | IL83994A (sv) |
SE (1) | SE8604059D0 (sv) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE8903219D0 (sv) * | 1989-10-02 | 1989-10-02 | Astra Ab | Process for the manufacture of budesonide |
GR1001529B (el) * | 1990-09-07 | 1994-03-31 | Elmuquimica Farm Sl | Μέ?οδος για την λήψη νέων 21-εστέρων της 16-17-ακετάλης της πρ να-1,4-διενο-3,20-διόνης. |
SE9100341D0 (sv) * | 1991-02-04 | 1991-02-04 | Astra Ab | Novel steroids |
FR2675146A1 (fr) * | 1991-04-10 | 1992-10-16 | Roussel Uclaf | Nouveaux derives sterouides de la pregna-1,4-diene-3,20-dione, leur preparation, leur application a la preparation de derives 16,17-methylene dioxy substitues et nouveaux intermediaires. |
GB9423919D0 (en) * | 1994-11-26 | 1995-01-11 | Rhone Poulenc Rorer Ltd | Chemical process |
DE19635498A1 (de) * | 1996-09-03 | 1998-03-26 | Byk Gulden Lomberg Chem Fab | Verfahren zur Epimerenanreicherung |
IT1291288B1 (it) * | 1997-04-30 | 1999-01-07 | Farmabios Srl | Processo per la preparazione di 16,17 acetali di derivati pregnanici con controllo della distribuzione epimerica al c-22. |
US6266556B1 (en) | 1998-04-27 | 2001-07-24 | Beth Israel Deaconess Medical Center, Inc. | Method and apparatus for recording an electroencephalogram during transcranial magnetic stimulation |
IT1302657B1 (it) * | 1998-10-13 | 2000-09-29 | Farmabios Srl | Processo stereoselettivo per la preparazione di budesonide nella formadi epimero 22-r. |
CA2430196C (en) * | 2000-11-10 | 2010-01-26 | Altana Pharma Ag | Process for the production of 16,17-[(cyclohexylmethylen)bis(oxy)]-11,21-dihydroxy-pregna-1,4-dien-3,20-dion or its 21-isobutyrat by transketalisation |
EP1465915A1 (en) | 2001-09-25 | 2004-10-13 | PHARMACIA & UPJOHN COMPANY | Stereoselective transacetalization of steroidal c-22 acetonide |
US20040235811A1 (en) * | 2002-10-08 | 2004-11-25 | Sepracor Inc. | Fatty acid modified forms of glucocorticoids |
CA2622640A1 (en) * | 2005-11-02 | 2007-05-18 | Sicor Inc. | Improved process for the preparation of ciclesonide |
US20070232578A1 (en) * | 2006-02-15 | 2007-10-04 | Pierluigi Rossetto | Crystalline forms of ciclesonide |
WO2016120891A1 (en) * | 2015-01-30 | 2016-08-04 | Coral Drugs Pvt. Ltd. | Novel process for preparation of glucocorticoid steroids |
JP7330101B2 (ja) | 2016-11-08 | 2023-08-21 | レゲネロン ファーマシューティカルス,インコーポレーテッド | ステロイド及びそのタンパク質コンジュゲート |
EP3624894A1 (en) | 2017-05-18 | 2020-03-25 | Regeneron Pharmaceuticals, Inc. | Cyclodextrin protein drug conjugates |
JP2021523147A (ja) | 2018-05-09 | 2021-09-02 | レゲネロン ファーマシューティカルス,インコーポレーテッド | 抗msr1抗体及びその使用方法 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE378109B (sv) * | 1972-05-19 | 1975-08-18 | Bofors Ab | |
SE378110B (sv) * | 1972-05-19 | 1975-08-18 | Bofors Ab | |
SE8008524L (sv) * | 1980-12-04 | 1982-06-05 | Draco Ab | 4-pregnen-derivat, ett forfarande for deras framstellning, beredning och metod for behandling av inflammatoriska tillstand |
IT1196142B (it) * | 1984-06-11 | 1988-11-10 | Sicor Spa | Procedimento per la preparazione di 16,17-acetali di derivati pregnanici e nuovi composti ottenuti |
-
1986
- 1986-09-25 SE SE8604059A patent/SE8604059D0/sv unknown
-
1987
- 1987-09-11 US US07/096,598 patent/US4925933A/en not_active Expired - Lifetime
- 1987-09-18 DE DE8787850282T patent/DE3774987D1/de not_active Expired - Fee Related
- 1987-09-18 EP EP87850282A patent/EP0262108B1/en not_active Expired - Lifetime
- 1987-09-18 ES ES198787850282T patent/ES2026576T3/es not_active Expired - Lifetime
- 1987-09-18 AT AT87850282T patent/ATE70066T1/de not_active IP Right Cessation
- 1987-09-23 IL IL83994A patent/IL83994A/xx unknown
- 1987-09-24 FI FI874189A patent/FI90345C/sv not_active IP Right Cessation
- 1987-09-24 KR KR1019870010561A patent/KR950014460B1/ko not_active IP Right Cessation
- 1987-09-24 JP JP62237588A patent/JP2668000B2/ja not_active Expired - Fee Related
-
1991
- 1991-12-12 GR GR91401949T patent/GR3003332T3/el unknown
-
1994
- 1994-05-12 HK HK46194A patent/HK46194A/xx not_active IP Right Cessation
-
1995
- 1995-10-20 CY CY179195A patent/CY1791A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
GR3003332T3 (en) | 1993-02-17 |
CY1791A (en) | 1995-10-20 |
FI90345B (sv) | 1993-10-15 |
JP2668000B2 (ja) | 1997-10-27 |
ATE70066T1 (de) | 1991-12-15 |
EP0262108A1 (en) | 1988-03-30 |
EP0262108B1 (en) | 1991-12-04 |
KR880003969A (ko) | 1988-06-01 |
IL83994A (en) | 1992-02-16 |
DE3774987D1 (de) | 1992-01-16 |
FI90345C (sv) | 1994-01-25 |
FI874189A (sv) | 1988-03-26 |
IL83994A0 (en) | 1988-02-29 |
US4925933A (en) | 1990-05-15 |
KR950014460B1 (ko) | 1995-11-28 |
FI874189A0 (sv) | 1987-09-24 |
ES2026576T3 (es) | 1992-05-01 |
HK46194A (en) | 1994-05-20 |
JPS6393795A (ja) | 1988-04-25 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
SE8604059D0 (sv) | A method of controlling the epimeric distribution in the preparation of 16,17-acetals of pregnane derivatives | |
ATE15206T1 (de) | 3-beta,7-beta,15-alpha-trihydroxy-5-androsten-1 - one, ihre 3,15-trimethylessigsaeure-ester und ihre herstellung. | |
NO932159L (no) | Gallesyrederivater, fremgangsmaate for fremstilling av dem og anvendelse av forbindelsene som legemidler | |
PT79997A (en) | Process for preparing complex compounds of piroxicam with cyclodextrins | |
ES2103433T3 (es) | Procedimiento para preparar derivados de 1-halo-2-desoxi-2,2-difluoro-d-ribofuranosilo enriquecidos en anomero alfa. | |
ES446411A1 (es) | Un metodo para preparar 17 alfa-ester-21-halo-pregnanos | |
IE40078L (en) | 1,2-benzisoxazole derivatives | |
ATE128111T1 (de) | Verfahren zur oxidation paraffinischer verbindungen mit sauerstoff. | |
DE68927103T2 (de) | Verfahren zur herstellung von gamma- und delta-lactonen | |
DK0843680T3 (da) | Isomeriseringsfremgangsmåde | |
ATE8788T1 (de) | Verfahren zur herstellung 3-bromosubstituierter desacetoxycephalosporansaeure-sulfoxyd-derivate. | |
FR2506305A1 (fr) | Nouveaux agents de deshydrogenation a base de derives organiques du selenium | |
AU501748B2 (en) | Substituted 2h-pyran-2, 6(3h) dione derivatives | |
ATE151428T1 (de) | Verfahren zur herstellung von 3- exomethylencephamsulfoxydderivate und zwischenverbindungen | |
AU499324B2 (en) | D-homo pregna 1, 4 diene-3, 11, 20 trione derivatives | |
SE7601753L (sv) | Sett att framstella 3-enoletrar av 11beta-hydroxi-delta?724-pregnen-3-oner och derivat derav | |
JPS51143646A (en) | Process for preparation of cyclohexanone and cyclopentanone derivative s | |
JPS5312493A (en) | Oxidation of steriod by microorganisms | |
DE3764457D1 (de) | Empfaengnisverhuetende, waessrig-saure zusammensetzung und verfahren zu ihrer herstellung. | |
ATE68487T1 (de) | Verfahren zur herstellung eines 2,3dihydroxychinoxalins. | |
SE8402755L (sv) | Forfarande for framstellning av 4-keto-9-metyl-fenazin | |
JPS55164700A (en) | 1alpha,25-dihydroxy-24-oxocholesterol, and its preparation | |
JPS5273890A (en) | Synthesis of 6-amino-penicillanic acid derivatives |