RU94044438A - Применение 2-фенил-3-ароилбензтиофенов для подавления способности к зачатию у женщин - Google Patents
Применение 2-фенил-3-ароилбензтиофенов для подавления способности к зачатию у женщинInfo
- Publication number
- RU94044438A RU94044438A RU94044438/14A RU94044438A RU94044438A RU 94044438 A RU94044438 A RU 94044438A RU 94044438/14 A RU94044438/14 A RU 94044438/14A RU 94044438 A RU94044438 A RU 94044438A RU 94044438 A RU94044438 A RU 94044438A
- Authority
- RU
- Russia
- Prior art keywords
- women
- aroylbenzthiophenes
- contraception
- suppression
- phenyl
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4535—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom, e.g. pizotifen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Метод подавления способности и зачатию у женщин, включающий введение женщинам эффективного количества соединения формулы, приведенной в описании, и его фармацевтически приемлемых солей и сольватов.
Claims (1)
- Метод подавления способности и зачатию у женщин, включающий введение женщинам эффективного количества соединения формулы, приведенной в описании, и его фармацевтически приемлемых солей и сольватов.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08/170,945 US5462949A (en) | 1993-12-21 | 1993-12-21 | Methods of inhibiting fertility in women |
US08/170945 | 1993-12-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
RU94044438A true RU94044438A (ru) | 1996-10-20 |
Family
ID=22621919
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU94044438/14A RU94044438A (ru) | 1993-12-21 | 1994-12-19 | Применение 2-фенил-3-ароилбензтиофенов для подавления способности к зачатию у женщин |
Country Status (15)
Country | Link |
---|---|
US (1) | US5462949A (ru) |
EP (1) | EP0659429A1 (ru) |
JP (1) | JPH07215870A (ru) |
KR (1) | KR950016747A (ru) |
CN (1) | CN1108091A (ru) |
AU (1) | AU8154594A (ru) |
CA (1) | CA2138456A1 (ru) |
CZ (1) | CZ322994A3 (ru) |
HU (1) | HUT71328A (ru) |
IL (1) | IL112030A (ru) |
NO (1) | NO944916L (ru) |
NZ (1) | NZ270188A (ru) |
PH (1) | PH31268A (ru) |
RU (1) | RU94044438A (ru) |
ZA (1) | ZA9410099B (ru) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6515009B1 (en) | 1991-09-27 | 2003-02-04 | Neorx Corporation | Therapeutic inhibitor of vascular smooth muscle cells |
US5811447A (en) | 1993-01-28 | 1998-09-22 | Neorx Corporation | Therapeutic inhibitor of vascular smooth muscle cells |
USRE39049E1 (en) | 1992-07-28 | 2006-03-28 | Eli Lilly And Company | Methods for inhibiting bone loss |
TW366342B (en) * | 1992-07-28 | 1999-08-11 | Lilly Co Eli | The use of 2-phenyl-3-aroylbenzothiophenes in inhibiting bone loss |
USRE38968E1 (en) | 1992-07-28 | 2006-02-07 | Eli Lilly And Company | Methods for inhibiting bone loss using 6-hydroxy-2-(4-hydroxyphenyl)-benzo[b]thien-3-yl-4-[2-(piperidin-1-yl) ethoxyphenylimethanone hydrochloride |
US5847007A (en) | 1993-05-13 | 1998-12-08 | Neorx Corporation | Prevention and treatment of pathologies associated with abnormally proliferative smooth muscle cells |
US6491938B2 (en) | 1993-05-13 | 2002-12-10 | Neorx Corporation | Therapeutic inhibitor of vascular smooth muscle cells |
US5595722A (en) | 1993-01-28 | 1997-01-21 | Neorx Corporation | Method for identifying an agent which increases TGF-beta levels |
US5478847A (en) | 1994-03-02 | 1995-12-26 | Eli Lilly And Company | Methods of use for inhibiting bone loss and lowering serum cholesterol |
US5569459A (en) * | 1995-02-15 | 1996-10-29 | Bio-Virus Research Incorporated | Pharmaceutical compositions for the management of premenstrual syndrome and alleviation of menopausal disorders |
IL120266A (en) | 1996-02-28 | 2005-05-17 | Pfizer | Use of estrogen antagonists and estrogen agonists in the preparation of medicaments for inhibiting pathological conditions |
TW442286B (en) * | 1996-02-28 | 2001-06-23 | Pfizer | New therapeutic uses of estrogen agonists |
AU6959898A (en) * | 1997-04-11 | 1998-11-11 | David J. Grainger | Compounds and therapies for the prevention of vascular and non-vascular pathol ogies |
US20020169205A1 (en) * | 1998-09-29 | 2002-11-14 | Krzysztof Chwalisz | Implantation rates after in vitro fertilization, and treatment of infertility and early pregnancy loss with a nitric oxide donor or substrate alone or in combination with progesterone, and a method for contraception with nitric oxide inhibitors in combination with antiprogestins or other agents |
US20060106010A1 (en) * | 2003-05-27 | 2006-05-18 | Black Larry J | Methods for inhibiting bone loss |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4133814A (en) * | 1975-10-28 | 1979-01-09 | Eli Lilly And Company | 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents |
US4418068A (en) * | 1981-04-03 | 1983-11-29 | Eli Lilly And Company | Antiestrogenic and antiandrugenic benzothiophenes |
IL65379A0 (en) * | 1981-04-03 | 1982-05-31 | Lilly Co Eli | Process for preparing acylated benzothiophenes |
US4380635A (en) * | 1981-04-03 | 1983-04-19 | Eli Lilly And Company | Synthesis of acylated benzothiophenes |
US5075321A (en) * | 1987-03-24 | 1991-12-24 | University Of Pennsylvania | Methods of treating diseases characterized by interactions of IgG-containing immune complexes with macrophage Fc receptors using antiestrogenic benzothiophenes |
US5395842A (en) * | 1988-10-31 | 1995-03-07 | Endorecherche Inc. | Anti-estrogenic compounds and compositions |
JP3157882B2 (ja) * | 1991-11-15 | 2001-04-16 | 帝国臓器製薬株式会社 | 新規なベンゾチオフエン誘導体 |
-
1993
- 1993-12-21 US US08/170,945 patent/US5462949A/en not_active Expired - Fee Related
-
1994
- 1994-12-19 RU RU94044438/14A patent/RU94044438A/ru unknown
- 1994-12-19 CA CA002138456A patent/CA2138456A1/en not_active Abandoned
- 1994-12-19 EP EP94309487A patent/EP0659429A1/en not_active Withdrawn
- 1994-12-19 PH PH40590A patent/PH31268A/en unknown
- 1994-12-19 HU HU9403678A patent/HUT71328A/hu unknown
- 1994-12-19 CZ CZ943229A patent/CZ322994A3/cs unknown
- 1994-12-19 AU AU81545/94A patent/AU8154594A/en not_active Abandoned
- 1994-12-19 KR KR1019940034938A patent/KR950016747A/ko not_active Application Discontinuation
- 1994-12-19 NZ NZ270188A patent/NZ270188A/en unknown
- 1994-12-19 JP JP6314582A patent/JPH07215870A/ja active Pending
- 1994-12-19 ZA ZA9410099A patent/ZA9410099B/xx unknown
- 1994-12-19 NO NO944916A patent/NO944916L/no unknown
- 1994-12-19 CN CN94119733A patent/CN1108091A/zh active Pending
- 1994-12-19 IL IL112030A patent/IL112030A/en active IP Right Revival
Also Published As
Publication number | Publication date |
---|---|
PH31268A (en) | 1998-06-18 |
JPH07215870A (ja) | 1995-08-15 |
HUT71328A (en) | 1995-11-28 |
HU9403678D0 (en) | 1995-02-28 |
CZ322994A3 (en) | 1995-08-16 |
KR950016747A (ko) | 1995-07-20 |
CA2138456A1 (en) | 1995-06-22 |
CN1108091A (zh) | 1995-09-13 |
IL112030A0 (en) | 1995-03-15 |
NZ270188A (en) | 1997-01-29 |
NO944916D0 (no) | 1994-12-19 |
US5462949A (en) | 1995-10-31 |
ZA9410099B (en) | 1996-06-19 |
EP0659429A1 (en) | 1995-06-28 |
NO944916L (no) | 1995-06-22 |
IL112030A (en) | 1998-03-10 |
AU8154594A (en) | 1995-06-29 |
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